JP2000504685A - タマリンド種子多糖で粘稠化された点眼液 - Google Patents
タマリンド種子多糖で粘稠化された点眼液Info
- Publication number
- JP2000504685A JP2000504685A JP9528356A JP52835697A JP2000504685A JP 2000504685 A JP2000504685 A JP 2000504685A JP 9528356 A JP9528356 A JP 9528356A JP 52835697 A JP52835697 A JP 52835697A JP 2000504685 A JP2000504685 A JP 2000504685A
- Authority
- JP
- Japan
- Prior art keywords
- ophthalmic
- weight
- polysaccharide fraction
- tamarind gum
- tamarind
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0048—Eye, e.g. artificial tears
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Inorganic Chemistry (AREA)
- Ophthalmology & Optometry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
- Polysaccharides And Polysaccharide Derivatives (AREA)
- Medicines Containing Plant Substances (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
Description
Claims (1)
- 【特許請求の範囲】 1.人工涙液または局所投与眼用医薬のビヒクルとして使用する粘稠化点眼液 の製造のためのタマリンドゴムの多糖分画の使用. 2.局所投与眼用医薬は持続放出性医薬である「請求項1」記載の使用. 3.点眼液は,タマリンドゴムの多糖分画 0.1〜5.0 重量%を含有する「請求 項1または2」記載の使用. 4.点眼液はタマリンドゴムの多糖分画 0.7〜1.5 重量%を含有する人工涙液 として用いる製剤である「請求項1」記載の使用. 5.製剤は1重量%のタマリンドゴムの多糖分画を含有する「請求項4」記載 の使用. 6.点眼液はタマリンドゴムの多糖分画1〜4重量%を含有する持続放出性の 局所投与眼用医薬のビヒクルである「請求項1」記載の使用. 7.ビヒクルは液体型で,タマリンドゴムの多糖分画 1.5〜2.5 重量%を含有 する「請求項6」記載の使用. 8.ビヒクルはゲル型で,タマリンドゴムの多糖分画3〜4重量%を含有する 「請求項6」記載の使用. 9.1種または2種以上の医薬的に活性な成分の有効量およびデリバリーシス テムとして多糖分画を含有する持続放出性の局所投与眼用医薬の製造のためのタ マリンドゴムの多糖分画の使用. 10.眼用医薬は1〜4重量%のタマリンドゴムの多糖分画を含有する「請求項 9」記載の使用. 11.1種または2種以上の医薬的に活性な成分はピロカルピン,チモロール, オフロキサシンおよびゲンタマイシンからなる群より選択される「請求項10」記 載の使用. 12.タマリンドゴムの多糖分画は市販のタマリンドゴムから精製して得られる 「請求項1〜11」のいずれか1項に記載の使用. 13.増粘剤およびムコ接着剤としてタマリンドゴムの多糖分画を含有する人工 涙液または局所投与眼用医薬のビヒクルとしての使用のための点眼液. 14.タマリンドゴムの多糖分画 0.1〜5.0 重量%を含有する「請求項13」記載 の点眼液. 15.タマリンドゴムの多糖分画 0.7〜1.5 重量%を含有する人工涙液として使 用するための「請求項13」記載の点眼液. 16.タマリンドゴムの多糖分画1〜4重量%を含有する持続放出性の局所投与 眼用医薬のビヒクルとして使用するための「請求項13」記載の点眼液. 17.1種または2種以上の医薬的に活性な成分の有効量およびデリバリーシス テムとしてタマリンドゴムの多糖分画を含有する持続放出性の局所投与眼用医薬 . 18.タマリンドゴムの多糖分画1〜4重量%を含有する「請求項17」記載の眼 用医薬. 19.1種または2種以上の医薬的に活性な成分はピロカルピン,チモロール, オフロキサシンおよびゲンタマイシンからなる群より選択される「請求項18」記 載の眼用医薬. 20.タマリンドゴムの多糖分画は市販のタマリンドゴムから精製して得られる 「請求項13〜19」のいずれか1項に記載の点眼液または眼用医薬.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IT96RM000075A IT1283911B1 (it) | 1996-02-05 | 1996-02-05 | Soluzioni oftalmiche viscosizzate con polisaccaridi della gomma di tamarindo |
IT96A000075 | 1996-02-05 | ||
PCT/IT1997/000026 WO1997028787A1 (en) | 1996-02-05 | 1997-02-04 | Ophthalmic solutions viscosified with tamarind seed polysaccharide |
Publications (2)
Publication Number | Publication Date |
---|---|
JP2000504685A true JP2000504685A (ja) | 2000-04-18 |
JP3872515B2 JP3872515B2 (ja) | 2007-01-24 |
Family
ID=11403863
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP52835697A Expired - Fee Related JP3872515B2 (ja) | 1996-02-05 | 1997-02-04 | タマリンド種子多糖で粘稠化された点眼液 |
Country Status (14)
Country | Link |
---|---|
US (1) | US6056950A (ja) |
EP (1) | EP0892636B1 (ja) |
JP (1) | JP3872515B2 (ja) |
KR (1) | KR100430260B1 (ja) |
AT (1) | ATE204745T1 (ja) |
AU (1) | AU1617897A (ja) |
CA (1) | CA2245617C (ja) |
DE (1) | DE69706410T2 (ja) |
DK (1) | DK0892636T3 (ja) |
EA (1) | EA001067B1 (ja) |
ES (1) | ES2164327T3 (ja) |
IT (1) | IT1283911B1 (ja) |
PT (1) | PT892636E (ja) |
WO (1) | WO1997028787A1 (ja) |
Cited By (6)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JP2007501799A (ja) * | 2003-08-07 | 2007-02-01 | アラーガン、インコーポレイテッド | 眼内に医薬を送達するための組成物ならびにその調製方法および使用方法 |
JP2010540619A (ja) * | 2007-10-02 | 2010-12-24 | エルエムエフアー・トレーディング・エス・アー | タマリンド種子多糖およびヒアルロン酸に基づく点眼組成物 |
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- 1997-02-04 JP JP52835697A patent/JP3872515B2/ja not_active Expired - Fee Related
- 1997-02-04 PT PT97902574T patent/PT892636E/pt unknown
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Cited By (8)
Publication number | Priority date | Publication date | Assignee | Title |
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JP2007501799A (ja) * | 2003-08-07 | 2007-02-01 | アラーガン、インコーポレイテッド | 眼内に医薬を送達するための組成物ならびにその調製方法および使用方法 |
JP2010540619A (ja) * | 2007-10-02 | 2010-12-24 | エルエムエフアー・トレーディング・エス・アー | タマリンド種子多糖およびヒアルロン酸に基づく点眼組成物 |
JP2013510844A (ja) * | 2009-11-16 | 2013-03-28 | エイチエムエフアールエイ ハンガリー リミテッド ライアビリティー カンパニー | Bdnf(脳由来神経栄養因子)をベースとする眼科用製剤およびそれらの使用 |
JP2016026229A (ja) * | 2009-11-16 | 2016-02-12 | エイチエムエフアールエイ ハンガリー リミテッド ライアビリティー カンパニーHmfra Hungary Limited Liability Company | Bdnf(脳由来神経栄養因子)をベースとする眼科用製剤およびそれらの使用 |
JP2013526594A (ja) * | 2010-05-24 | 2013-06-24 | インデナ エッセ ピ ア | 微生物感染の治療に使用するためのタマリンド種子多糖 |
JP2012012328A (ja) * | 2010-06-30 | 2012-01-19 | Dsp Gokyo Food & Chemical Co Ltd | キシログルカン−カチオン複合体及びそれを含有する安定化組成物 |
JP2022095972A (ja) * | 2015-07-13 | 2022-06-28 | 株式会社 東北テクノアーチ | 視神経保護用組成物 |
JP7270222B2 (ja) | 2015-07-13 | 2023-05-10 | 株式会社 東北テクノアーチ | 視神経保護用組成物 |
Also Published As
Publication number | Publication date |
---|---|
JP3872515B2 (ja) | 2007-01-24 |
EA001067B1 (ru) | 2000-10-30 |
WO1997028787A1 (en) | 1997-08-14 |
CA2245617C (en) | 2005-07-12 |
ES2164327T3 (es) | 2002-02-16 |
US6056950A (en) | 2000-05-02 |
ITRM960075A1 (it) | 1997-08-05 |
DE69706410T2 (de) | 2002-06-06 |
EA199800689A1 (ru) | 1999-02-25 |
EP0892636A1 (en) | 1999-01-27 |
KR100430260B1 (ko) | 2004-07-30 |
CA2245617A1 (en) | 1997-08-14 |
DK0892636T3 (da) | 2001-12-17 |
PT892636E (pt) | 2002-02-28 |
ITRM960075A0 (it) | 1996-02-05 |
DE69706410D1 (de) | 2001-10-04 |
KR19990082244A (ko) | 1999-11-25 |
AU1617897A (en) | 1997-08-28 |
ATE204745T1 (de) | 2001-09-15 |
IT1283911B1 (it) | 1998-05-07 |
EP0892636B1 (en) | 2001-08-29 |
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