IN2006DE01793A - - Google Patents
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- Publication number
- IN2006DE01793A IN2006DE01793A IN1793DE2006A IN2006DE01793A IN 2006DE01793 A IN2006DE01793 A IN 2006DE01793A IN 1793DE2006 A IN1793DE2006 A IN 1793DE2006A IN 2006DE01793 A IN2006DE01793 A IN 2006DE01793A
- Authority
- IN
- India
- Prior art keywords
- sup
- formula
- preparing
- esters
- dihalomethylpyrazoles
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/30—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and unsaturated
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/34—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings
- C07C229/36—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton containing six-membered aromatic rings with at least one amino group and one carboxyl group bound to the same carbon atom of the carbon skeleton
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/14—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10349500A DE10349500A1 (de) | 2003-10-23 | 2003-10-23 | Verfahren zum Herstellen von 2-Dihalogenacyl-3-amino-acrylsäureestern und 3-Dihalogenmethyl-pyrazol-4-carbonsäureestern |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IN2006DE01793A true IN2006DE01793A (enExample) | 2007-08-10 |
Family
ID=34529740
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IN1793DE2006 IN2006DE01793A (enExample) | 2003-10-23 | 2006-04-03 |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US7358387B2 (enExample) |
| EP (1) | EP1678119B1 (enExample) |
| JP (1) | JP4725977B2 (enExample) |
| KR (1) | KR101116686B1 (enExample) |
| CN (1) | CN100422141C (enExample) |
| AT (1) | ATE494274T1 (enExample) |
| BR (1) | BRPI0415855B1 (enExample) |
| DE (2) | DE10349500A1 (enExample) |
| DK (1) | DK1678119T3 (enExample) |
| IL (1) | IL175024A (enExample) |
| IN (1) | IN2006DE01793A (enExample) |
| MX (1) | MXPA06004339A (enExample) |
| TW (1) | TWI363050B (enExample) |
| WO (1) | WO2005042468A1 (enExample) |
Families Citing this family (63)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2003261796B2 (en) | 2003-08-28 | 2010-01-21 | Universal Can Corporation | Apparatus for producing bottle can |
| DE10352082A1 (de) * | 2003-10-23 | 2005-05-25 | Bayer Cropscience Ag | Hexylcarboxanilide |
| DE102006039909A1 (de) | 2006-08-25 | 2008-03-13 | Bayer Cropscience Ag | Verfahren zum Herstellen von 3-Dihalomethyl-pyrazol-4-carbonsäurederivaten |
| CN101627008A (zh) * | 2006-12-28 | 2010-01-13 | 三井化学Agro株式会社 | 2-含氟酰基-3-氨基丙烯腈衍生物及其制备方法 |
| RU2459807C2 (ru) * | 2007-05-31 | 2012-08-27 | Зингента Партисипейшнс Аг | Способ получения пиразолов |
| EP1997808A1 (en) * | 2007-05-31 | 2008-12-03 | Syngeta Participations AG | Process for the production of pyrazoles |
| EA016615B1 (ru) | 2007-06-01 | 2012-06-29 | Басф Се | Способ получения n-замещенных (3-дигалометил-1-метилпиразол-4-ил)карбоксамидов |
| JP5559678B2 (ja) | 2007-06-15 | 2014-07-23 | ビーエーエスエフ ソシエタス・ヨーロピア | ジフルオロメチル置換ピラゾール化合物の製造方法 |
| EP2008996A1 (en) * | 2007-06-27 | 2008-12-31 | Syngeta Participations AG | Process for the production of pyrazoles |
| EP2042482A1 (de) * | 2007-09-26 | 2009-04-01 | Bayer CropScience AG | Verfahren zur Herstellung von 2-Dihalogenacyl-3-amino-acrylsäure-Derivaten |
| EP2072497A1 (de) | 2007-12-21 | 2009-06-24 | Bayer CropScience AG | Verfahren zum Herstellen von 2-Fluoracyl-3-amino-acrylsäure-Derivaten |
| EP2133341A1 (de) * | 2008-02-25 | 2009-12-16 | Bayer CropScience AG | Verfahren zur regioselektiven Synthese von 1-Alkyl-3-haloalkyl-pyrazol-4-carbonsäure-Derivaten |
| EP2100883A1 (de) | 2008-03-10 | 2009-09-16 | Bayer CropScience AG | Verfahren zur regioselektiven Synthese von 1-Alkyl-3-haloalkyl-pyrazol-4carbonsäure-Derivaten |
| KR101211264B1 (ko) * | 2008-03-18 | 2012-12-18 | 미쓰이가가쿠 아그로 가부시키가이샤 | 함불소 아실아세트산 유도체의 제조방법, 함불소 피라졸카르복실산에스테르 유도체의 제조방법 및 함불소 피라졸카르복실산 유도체의 제조방법 |
| JP2009227643A (ja) * | 2008-03-25 | 2009-10-08 | Mitsui Chemicals Agro Inc | 含フッ素アルキルカルボン酸誘導体を利用した含フッ素ピラゾール誘導体の製造方法 |
| WO2009133178A1 (de) * | 2008-05-02 | 2009-11-05 | Basf Se | Verfahren zur herstellung von 2-(aminomethyliden)-4,4-difluor-3-oxobuttersäureestern |
| WO2009133179A2 (de) * | 2008-05-02 | 2009-11-05 | Basf Se | Verfahren zur herstellung halogensubstituierter 2-(aminomethyliden)-3-oxobuttersäureester |
| DK2288597T3 (en) * | 2008-05-05 | 2015-01-26 | Basf Se | PROCESS FOR THE PREPARATION OF 1,3,4-SUBSTITUTED pyrazole |
| US7601864B1 (en) * | 2008-05-08 | 2009-10-13 | Ufc Corporation | Method for synthesizing 4,4-dihalogen-2-(dialkylamino)methylene-3-oxy-alkylbutyrate and derivatives thereof |
| JP5558467B2 (ja) | 2008-07-21 | 2014-07-23 | ビーエーエスエフ ソシエタス・ヨーロピア | １，３−二置換ピラゾールカルボン酸エステルの調製方法 |
| KR101772610B1 (ko) | 2008-07-25 | 2017-09-12 | 비이브 헬쓰케어 컴퍼니 | 화합물 |
| JP5228817B2 (ja) * | 2008-11-12 | 2013-07-03 | セントラル硝子株式会社 | ピラゾール化合物の製造方法 |
| JP5572168B2 (ja) | 2008-12-11 | 2014-08-13 | ビーブ・ヘルスケア・カンパニー | カルバモイルピリドンｈｉｖインテグラーゼ阻害剤の製造方法および中間体 |
| US8624023B2 (en) | 2008-12-11 | 2014-01-07 | Shionogi & Co., Ltd. | Synthesis of carbamoylpyridone HIV integrase inhibitors and intermediates |
| TWI518084B (zh) | 2009-03-26 | 2016-01-21 | 鹽野義製藥股份有限公司 | 哌喃酮與吡啶酮衍生物之製造方法 |
| AR077503A1 (es) * | 2009-07-28 | 2011-08-31 | Syngenta Participations Ag | Procesos relacionados con la alquilacion de pirazoles |
| US8362272B2 (en) | 2009-11-05 | 2013-01-29 | Basf Se | Process for preparing 1,3-disubstituted pyrazole compounds |
| US8362273B2 (en) | 2009-11-05 | 2013-01-29 | Basf Se | Process for preparing aminale and their use for preparing 1,3-disubstituted pyrazole compounds |
| TWI582097B (zh) | 2010-03-23 | 2017-05-11 | Ｖｉｉｖ醫療保健公司 | 製備胺甲醯吡啶酮衍生物及中間體之方法 |
| AU2011288601B2 (en) * | 2010-08-10 | 2014-08-07 | Syngenta Crop Protection Ag | Process for the preparation of 3-haloalkylpyrazoles |
| JP5605104B2 (ja) * | 2010-09-10 | 2014-10-15 | セントラル硝子株式会社 | ピラゾール化合物の製造方法 |
| JP5790195B2 (ja) * | 2011-06-22 | 2015-10-07 | セントラル硝子株式会社 | ピラゾール化合物の製造方法 |
| DE112012002522T5 (de) * | 2011-06-22 | 2014-03-13 | Central Glass Co., Ltd. | Verfahren zur Herstellung einer Pyrazol-Verbindung |
| JP5793983B2 (ja) * | 2011-06-22 | 2015-10-14 | セントラル硝子株式会社 | ピラゾール化合物の製造方法 |
| JP5830957B2 (ja) * | 2011-06-22 | 2015-12-09 | セントラル硝子株式会社 | ピラゾール化合物の製造方法 |
| JP5915004B2 (ja) * | 2011-06-22 | 2016-05-11 | セントラル硝子株式会社 | ピラゾール化合物の製造方法 |
| EP2623496A1 (de) | 2012-02-01 | 2013-08-07 | Bayer CropScience AG | Verfahren zur Herstellung von 3,5-bis (fluoralkyl)-pyrazol-4-carbonsäure-Derivaten und 3,5-bis(fluoralkyl)-pyrazolen |
| CN102731402A (zh) * | 2012-06-29 | 2012-10-17 | 上海康鹏化学有限公司 | 3-三氟甲基吡唑-4-羧酸和3-二氟甲基吡唑-4-羧酸的制备方法 |
| US8871947B2 (en) | 2013-02-04 | 2014-10-28 | KingChem LLC | Preparation of alkyl 3-difluoromethyl-1-methyl-1H-pyrazole-4-carboxylic acid ester |
| ES2627739T3 (es) | 2013-05-22 | 2017-07-31 | Bayer Cropscience Aktiengesellschaft | Procedimiento de preparación de derivados de 3,5-bis(fluoroalquil)pirazol a partir de alfa,alfa-dihaloaminas |
| KR102233203B1 (ko) | 2013-05-22 | 2021-03-26 | 바이엘 크롭사이언스 악티엔게젤샤프트 | 3,5-비스(플루오로알킬)피라졸 유도체의 제조방법 |
| TWI647215B (zh) * | 2013-11-11 | 2019-01-11 | 德商拜耳作物科學股份有限公司 | 自α,α－二鹵胺製備３,５－雙鹵烷基吡唑衍生物之方法 |
| US9139507B2 (en) | 2013-12-09 | 2015-09-22 | KingChem LLC. | Process for the preparation of alkyl 3-difluoromethyl-1-methyl-1H-pyrazole-4-carboxylate and its analogs |
| JPWO2015105129A1 (ja) | 2014-01-10 | 2017-03-23 | 旭硝子株式会社 | エーテル性酸素原子含有ペルフルオロアルキル基置換ピラゾール環化合物およびその製造方法 |
| KR102410034B1 (ko) * | 2014-03-24 | 2022-06-15 | 바이엘 크롭사이언스 악티엔게젤샤프트 | α,α-디할로아민 및 케트이민으로부터 3,5-비스(할로알킬)피라졸 유도체의 제조방법 |
| EP3015458A1 (en) | 2014-11-03 | 2016-05-04 | Bayer CropScience AG | Process for preparing 3,5-bis(haloalkyl)pyrazole derivatives from a,a-dihaloamines and ketimines |
| ES2672577T3 (es) | 2014-06-11 | 2018-06-15 | Bayer Cropscience Aktiengesellschaft | Proceso para preparar derivados de 3,5-bis(haloalquil)pirazol por medio de la acilación de Hidrazonas |
| MX383114B (es) | 2014-06-11 | 2025-03-13 | Bayer Cropscience Ag | Proceso para la preparación de 3,5-bis(haloalquil)pirazoles por medio de la acilación de cetiminas. |
| EP2987782A1 (en) | 2014-08-22 | 2016-02-24 | Solvay SA | Distillation process comprising at least two distillation steps to obtain purified halogenated carboxylic acid halide, and use of the purified halogenated carboxylic acid halide |
| JP2017533941A (ja) | 2014-11-17 | 2017-11-16 | ソルヴェイ（ソシエテ アノニム） | 精製ハロゲン化カルボン酸ハロゲン化物を得るための少なくとも２つの蒸留ステップを含む蒸留プロセス、および精製ハロゲン化カルボン酸ハロゲン化物の使用 |
| CN104529899A (zh) * | 2014-12-19 | 2015-04-22 | 浙江泰达作物科技有限公司 | 高区域选择性制备1-烷基-3-卤代烷基吡唑衍生物的方法 |
| CN105541716B (zh) * | 2015-03-26 | 2024-02-23 | Ａｇｃ株式会社 | 吡唑衍生物的制造方法 |
| KR20160120009A (ko) | 2015-04-07 | 2016-10-17 | (주)부흥산업사 | 4,4-디플루오로-((2-디알킬아미노)메틸렌)-3-옥소부탄산 알킬에스테르의 새로운 제조방법 |
| CN107960078A (zh) | 2015-06-26 | 2018-04-24 | 拜耳作物科学股份公司 | 由α,α-二卤代烷基胺和酮亚胺制备含有卤代烷氧基和卤代烷硫基的取代的吡唑的方法 |
| EP3178813A1 (en) | 2015-12-09 | 2017-06-14 | Basf Se | Method for preparing halogenated 3-oxocarboxylates carrying a 2-alkoxymethylidene or a 2-dialkylaminomethylidene group |
| JP2019515938A (ja) * | 2016-05-10 | 2019-06-13 | ソルヴェイ（ソシエテ アノニム） | ３−（ハロアルキルまたはホルミル）−１ｈ−ピラゾール−４−カルボン酸またはエステルを含む組成物、その製造、およびカルボキサミド調製のためのその使用 |
| ES2849960T3 (es) | 2016-09-21 | 2021-08-24 | Bayer Cropscience Ag | Procedimiento para la preparación de 3-fluoroalquil-5-pirazolcarboxilatos y ácidos 3-fluoroalquil-5-pirazolcarboxílicos |
| CN111372908A (zh) | 2017-09-04 | 2020-07-03 | 索尔维公司 | 用于制造二氟乙酰氯的方法和中间体 |
| CN111116364B (zh) * | 2019-12-30 | 2022-11-11 | 浙江本立科技股份有限公司 | 2-多卤代乙酰基-3-烷氧基丙烯酸酯的制备方法 |
| CN113912541A (zh) * | 2021-10-29 | 2022-01-11 | 南通宝凯药业有限公司 | 一种3-二氟甲基-1-甲基-1h-吡唑-4-羧酸的制备方法 |
| CN114195715B (zh) * | 2021-12-31 | 2024-05-10 | 福建永晶科技股份有限公司 | 1-甲基-3-二氟甲基-4-吡唑酸和1-甲基-3-三氟甲基-4-吡唑酸的制备方法 |
| CN117447401B (zh) * | 2023-12-26 | 2024-04-19 | 山东国邦药业有限公司 | 一种二氟吡唑酸的合成方法 |
| CN120118034A (zh) * | 2025-05-14 | 2025-06-10 | 辽宁龙田化工科技有限公司 | 一种3-二氟甲基-1-甲基吡唑-4-羧酸的合成方法 |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5093347A (en) * | 1991-01-28 | 1992-03-03 | Monsanto Company | 3-difluoromethylpyrazolecarboxamide fungicides, compositions and use |
| US5223526A (en) * | 1991-12-06 | 1993-06-29 | Monsanto Company | Pyrazole carboxanilide fungicides and use |
| US5498624A (en) * | 1995-05-03 | 1996-03-12 | Monsanto Company | Selected pyrazolyl derivatives |
| KR20000035081A (ko) * | 1998-11-10 | 2000-06-26 | 마크 에스. 아들러 | 2-(트리할로아세틸)-3-(치환된 아미노)-2-프로페노에이트 제조방법 |
| CN1308044A (zh) * | 2000-01-28 | 2001-08-15 | 住友化学工业株式会社 | 二卤代化合物和制备维生素a衍生物的方法 |
| DE10161978A1 (de) * | 2001-12-17 | 2003-06-26 | Bayer Ag | Verfahren zur Herstellung von 2-Halogenacyl-3-amino-acrylsäure-derivate |
-
2003
- 2003-10-23 DE DE10349500A patent/DE10349500A1/de not_active Withdrawn
-
2004
- 2004-10-12 CN CNB2004800312031A patent/CN100422141C/zh not_active Expired - Lifetime
- 2004-10-12 DE DE502004012095T patent/DE502004012095D1/de not_active Expired - Lifetime
- 2004-10-12 EP EP04790277A patent/EP1678119B1/de not_active Expired - Lifetime
- 2004-10-12 WO PCT/EP2004/011376 patent/WO2005042468A1/de not_active Ceased
- 2004-10-12 BR BRPI0415855-5B1A patent/BRPI0415855B1/pt not_active IP Right Cessation
- 2004-10-12 DK DK04790277.0T patent/DK1678119T3/da active
- 2004-10-12 KR KR1020067009068A patent/KR101116686B1/ko not_active Expired - Lifetime
- 2004-10-12 MX MXPA06004339A patent/MXPA06004339A/es active IP Right Grant
- 2004-10-12 AT AT04790277T patent/ATE494274T1/de active
- 2004-10-12 JP JP2006535992A patent/JP4725977B2/ja not_active Expired - Lifetime
- 2004-10-12 US US10/576,059 patent/US7358387B2/en not_active Expired - Lifetime
- 2004-10-22 TW TW093132065A patent/TWI363050B/zh not_active IP Right Cessation
-
2006
- 2006-04-03 IN IN1793DE2006 patent/IN2006DE01793A/en unknown
- 2006-04-20 IL IL175024A patent/IL175024A/en active IP Right Grant
Also Published As
| Publication number | Publication date |
|---|---|
| TWI363050B (en) | 2012-05-01 |
| MXPA06004339A (es) | 2006-06-05 |
| WO2005042468A1 (de) | 2005-05-12 |
| DE10349500A1 (de) | 2005-06-02 |
| US7358387B2 (en) | 2008-04-15 |
| TW200526550A (en) | 2005-08-16 |
| JP2007509850A (ja) | 2007-04-19 |
| KR101116686B1 (ko) | 2012-02-22 |
| US20060252944A1 (en) | 2006-11-09 |
| BRPI0415855A (pt) | 2007-01-09 |
| EP1678119A1 (de) | 2006-07-12 |
| ATE494274T1 (de) | 2011-01-15 |
| IL175024A (en) | 2011-05-31 |
| DE502004012095D1 (de) | 2011-02-17 |
| JP4725977B2 (ja) | 2011-07-13 |
| KR20060109901A (ko) | 2006-10-23 |
| CN1871204A (zh) | 2006-11-29 |
| DK1678119T3 (da) | 2011-05-02 |
| EP1678119B1 (de) | 2011-01-05 |
| CN100422141C (zh) | 2008-10-01 |
| IL175024A0 (en) | 2006-08-20 |
| BRPI0415855B1 (pt) | 2013-11-05 |
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