IN2003KO00001A - - Google Patents

Info

Publication number
IN2003KO00001A
IN2003KO00001A IN1KO2003A IN2003KO00001A IN 2003KO00001 A IN2003KO00001 A IN 2003KO00001A IN 1KO2003 A IN1KO2003 A IN 1KO2003A IN 2003KO00001 A IN2003KO00001 A IN 2003KO00001A
Authority
IN
India
Application number
Other languages
English (en)
Inventor
Mark R Schmitt
Donald R Kirsch
Jane E Harris
Carl F Beyer
Klaus-Juergen Pees
Paul Carter
Waldemar Pfrengle
Guido Albert
Original Assignee
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Home Prod filed Critical American Home Prod
Publication of IN2003KO00001A publication Critical patent/IN2003KO00001A/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IN1KO2003 2000-06-30 2003-01-01 IN2003KO00001A (ja)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US21558500P 2000-06-30 2000-06-30

Publications (1)

Publication Number Publication Date
IN2003KO00001A true IN2003KO00001A (ja) 2005-12-02

Family

ID=22803554

Family Applications (1)

Application Number Title Priority Date Filing Date
IN1KO2003 IN2003KO00001A (ja) 2000-06-30 2003-01-01

Country Status (24)

Country Link
US (1) US7329663B2 (ja)
EP (1) EP1307200A2 (ja)
JP (1) JP2004502691A (ja)
KR (1) KR20030013475A (ja)
CN (1) CN1592624A (ja)
AR (1) AR034553A1 (ja)
AU (2) AU7306201A (ja)
BG (1) BG107277A (ja)
BR (1) BR0112038A (ja)
CA (1) CA2413802A1 (ja)
CZ (1) CZ20024150A3 (ja)
EA (1) EA006483B1 (ja)
GE (1) GEP20053688B (ja)
HK (1) HK1052646A1 (ja)
HU (1) HUP0300798A3 (ja)
IL (1) IL152869A0 (ja)
IN (1) IN2003KO00001A (ja)
MX (1) MXPA02011913A (ja)
NO (1) NO20026195L (ja)
NZ (1) NZ523807A (ja)
PL (1) PL360027A1 (ja)
SK (1) SK18412002A3 (ja)
WO (1) WO2002002563A2 (ja)
ZA (1) ZA200300793B (ja)

Families Citing this family (48)

* Cited by examiner, † Cited by third party
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US6255309B1 (en) 1999-03-19 2001-07-03 American Cyanomid Co. Fungicidal trifluoromethylalkylamino-triazolopyrimidines
AU2002221831A1 (en) * 2000-11-13 2002-05-21 Basf Aktiengesellschaft 7-(r)-amino-triazolopyrimidines, the production thereof and use of the same for combating phytopathogenic fungi
WO2002083677A1 (en) * 2001-04-11 2002-10-24 Basf Aktiengesellschaft 6-(2-chloro-6-fluoro-phenyl)-triazolopyrimidines
ATE287405T1 (de) * 2001-04-11 2005-02-15 Wyeth Corp 5-halogen-6-phenyl-7-fluoroalkylamino- triazolopyrimidine als fungizide
DE10121101A1 (de) * 2001-04-27 2002-10-31 Bayer Ag Triazolopyrimidine
DE10121162A1 (de) * 2001-04-30 2002-10-31 Bayer Ag Triazolopyrimidine
DE10124208A1 (de) † 2001-05-18 2002-11-21 Bayer Ag Verwendung von Triazolopyrimidin-Derivaten als Mikrobizide
JP2005504744A (ja) * 2001-07-18 2005-02-17 ビーエーエスエフ アクチェンゲゼルシャフト 殺菌薬としての置換された６−（２−トリル）−トリアゾロピリミジン
DE50309022D1 (de) 2002-03-21 2008-03-06 Basf Ag Fungizide triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
JPWO2004011467A1 (ja) * 2002-07-29 2005-12-15 北興化学工業株式会社 トリアゾロピリミジン誘導体および農園芸用殺菌剤
UA80304C2 (en) * 2002-11-07 2007-09-10 Basf Ag Substituted 6-(2-halogenphenyl)triazolopyrimidines
CN1768060A (zh) * 2003-03-31 2006-05-03 巴斯福股份公司 7－(链烯基氨基)三唑并嘧啶、其生产方法及其在防治有害真菌中的用途以及包含所述三唑并嘧啶的物质
WO2004108136A1 (en) * 2003-06-04 2004-12-16 Vernalis (Cambridge) Limited Triazolo `1 , 5-a!pyrimidines and their use in medicine
DE10325133A1 (de) * 2003-06-04 2004-12-23 Bayer Cropscience Ag Triazolopyrimidine
DE10328171A1 (de) * 2003-06-24 2005-01-13 Bayer Cropscience Ag Triazolopyrimidine
DE10328173A1 (de) * 2003-06-24 2005-01-13 Bayer Cropscience Ag Triazolopyrimidine
DE10328481A1 (de) * 2003-06-25 2005-01-13 Bayer Ag Triazolopyrimidine
US7419982B2 (en) 2003-09-24 2008-09-02 Wyeth Holdings Corporation Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts
WO2005030218A1 (en) * 2003-09-24 2005-04-07 Wyeth Holdings Corporation 6-aryl-7-halo-imidazo[1,2-a]pyrimidines as anticancer agent
JP2007506744A (ja) 2003-09-24 2007-03-22 ワイス・ホールディングズ・コーポレイション 抗癌剤としての６−［（置換）フェニル］トリアゾロピリミジン類
EP1674454A4 (en) * 2003-10-17 2006-12-27 Nippon Kayaku Kk SUBSTITUTED 2-AMINO-1,2,4-TRIAZOLO 1,5-A-PYRIMIDINE DERIVATIVE AND THE USE THEREOF
JP4606015B2 (ja) * 2003-11-25 2011-01-05 日本化薬株式会社 ［１，２，４］トリアゾロ［１，５−ａ］ピリミジン誘導体の新規医薬用途
MY179926A (en) 2003-12-08 2020-11-19 Wyeth Corp Process for the preparation of tubulin inhibitors
BRPI0417637A (pt) * 2003-12-17 2007-03-27 Basf Ag compostos, processo para preparar os mesmos, agente, semente, e, processo para combater fungos nocivos fitopatogênicos
CN1890243A (zh) * 2003-12-17 2007-01-03 巴斯福股份公司 6－(2,4,6－三卤代苯基)三唑并嘧啶、其制备方法及其在防治病原性真菌中的用途以及包含所述物质的组合物
BRPI0508717A (pt) * 2004-03-30 2007-08-07 Basf Ag compostos, processo para preparar os mesmos, agente, semente, e, processo para combater fungos nocivos fitopatogênicos
JP2007538028A (ja) * 2004-05-17 2007-12-27 ビーエーエスエフ　アクチェンゲゼルシャフト トリアゾロピリミジン化合物および病原菌を制御するためのそれらの使用
CN1964629A (zh) * 2004-06-09 2007-05-16 巴斯福股份公司 三唑并嘧啶化合物及其在防治有害真菌中的用途
JP2008503538A (ja) * 2004-06-25 2008-02-07 ビーエーエスエフ　アクチェンゲゼルシャフト トリアゾロピリミジン化合物およびそれらの病原性菌類を防除するための使用
AU2006251989B2 (en) * 2005-05-20 2010-05-27 Alantos-Pharmaceuticals, Inc. Pyrimidine or triazine fused bicyclic metalloprotease inhibitors
US20070155738A1 (en) * 2005-05-20 2007-07-05 Alantos Pharmaceuticals, Inc. Heterobicyclic metalloprotease inhibitors
WO2007011759A2 (en) * 2005-07-15 2007-01-25 Kalypsys, Inc. Inhibitors of mitotic kinesin
CN101370813A (zh) * 2005-12-16 2009-02-18 惠氏公司 用作抗癌药物的6-[(取代的)苯基]三唑并嘧啶类的二聚体和加合物
TW200800026A (en) * 2006-02-28 2008-01-01 Basf Ag Substituted 6-phenyl-7-amino-[1,2,4]-triazolo[1,5-a] pyrimidines and their use for controlling harmful fungi
WO2007116011A2 (de) * 2006-04-10 2007-10-18 Basf Se Substituierte triazolopyrimidine, verfahren zu ihrer herstellung und ihre verwendung zur bekämpfung von schadpilzen sowie sie enthaltende mittel
JP5231829B2 (ja) 2007-02-15 2013-07-10 石原産業株式会社 ピリジル−トリアゾロピリミジン誘導体又はその塩、それらを含有する有害生物防除剤並びにそれらの製造方法
ES2396177T3 (es) 2007-08-14 2013-02-19 Bayer Intellectual Property Gmbh Pirimidinas bicíclicas fusionadas
WO2012047856A2 (en) 2010-10-04 2012-04-12 Institute For Hepatitis And Virus Research Novel inhibitors of secretion of hepatitis b virus antigens
CN104395298A (zh) 2012-06-22 2015-03-04 住友化学株式会社 稠合杂环化合物
CN103360398B (zh) * 2013-07-22 2015-03-25 山东大学 一种三唑并嘧啶类hiv-1逆转录酶抑制剂及其制备方法与应用
GB201504565D0 (en) 2015-03-18 2015-05-06 Takeda Pharmaceutical Novel compounds
KR101995533B1 (ko) * 2017-03-21 2019-07-02 한국화학연구원 [1,2,4]트리아졸로[4,3-a]퀴노잘린 아미노 페닐 유도체 또는 이의 약학적으로 허용가능한 염, 이의 제조방법 및 이를 유효성분으로 포함하는 BET 단백질 관련 질환의 예방 또는 치료용 약학적 조성물
WO2020159942A1 (en) * 2019-01-29 2020-08-06 Tosk, Inc. Pyrazolopyrimidine modulators of ras gtpase
AU2021255495A1 (en) * 2020-04-14 2022-12-15 The Regents Of The University Of California Substituted {1,2,4,} triazolo{1,5-a} pyrimidine compounds and use in stabilizing microtubules
IL297327A (en) * 2020-05-01 2022-12-01 Gilead Sciences Inc 4,2-deoxypyrimidine compounds that inhibit cd73
US20230279006A1 (en) * 2020-07-08 2023-09-07 Klotho Therapeutics, Inc. Novel compounds and methods for increasing klotho gene expression
WO2023077030A1 (en) 2021-10-29 2023-05-04 Gilead Sciences, Inc. Cd73 compounds
WO2023143194A1 (zh) * 2022-01-25 2023-08-03 瑞石生物医药有限公司 一种ccr4小分子拮抗剂及其用途

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FR2784380B1 (fr) * 1998-09-25 2002-09-06 American Cyanamid Co Triazolopyrimidines 7-oxy- et 7-thio-substituees fongicides
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DE10121102A1 (de) * 2001-04-27 2002-11-07 Bayer Ag Triazolopyrimidine
DE10121101A1 (de) * 2001-04-27 2002-10-31 Bayer Ag Triazolopyrimidine
DE10121162A1 (de) * 2001-04-30 2002-10-31 Bayer Ag Triazolopyrimidine
US7037902B2 (en) * 2002-07-03 2006-05-02 Receptron, Inc. Affinity small molecules for the EPO receptor
US7419982B2 (en) * 2003-09-24 2008-09-02 Wyeth Holdings Corporation Crystalline forms of 5-chloro-6-{2,6-difluoro-4-[3-(methylamino)propoxy]phenyl}-N-[(1S)-2,2,2-trifluoro-1-methylethyl][1,2,4]triazolo[1,5-a]pyrimidin-7-amine salts
JP2007506744A (ja) * 2003-09-24 2007-03-22 ワイス・ホールディングズ・コーポレイション 抗癌剤としての６−［（置換）フェニル］トリアゾロピリミジン類

Also Published As

Publication number Publication date
SK18412002A3 (sk) 2003-06-03
EP1307200A2 (en) 2003-05-07
HUP0300798A2 (hu) 2003-07-28
HUP0300798A3 (en) 2006-02-28
IL152869A0 (en) 2003-06-24
CZ20024150A3 (cs) 2003-09-17
NO20026195L (no) 2003-02-27
US7329663B2 (en) 2008-02-12
HK1052646A1 (zh) 2003-09-26
WO2002002563A3 (en) 2003-01-03
EA006483B1 (ru) 2005-12-29
JP2004502691A (ja) 2004-01-29
KR20030013475A (ko) 2003-02-14
NO20026195D0 (no) 2002-12-23
AU2001273062B2 (en) 2005-11-24
PL360027A1 (en) 2004-09-06
CA2413802A1 (en) 2002-01-10
CN1592624A (zh) 2005-03-09
AU7306201A (en) 2002-01-14
US20020068744A1 (en) 2002-06-06
BG107277A (bg) 2004-01-30
MXPA02011913A (es) 2003-04-22
AR034553A1 (es) 2004-03-03
WO2002002563A2 (en) 2002-01-10
EA200300091A1 (ru) 2003-08-28
GEP20053688B (en) 2005-12-12
NZ523807A (en) 2004-09-24
ZA200300793B (en) 2004-07-20
BR0112038A (pt) 2003-04-01

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