IL98599A - מלחים יציבים של " 4-דהאוקסי-" 4-אפי- מתילאמינו אברמקטין ותכשירים קוטלי חרקים המכילים אותם - Google Patents

מלחים יציבים של " 4-דהאוקסי-" 4-אפי- מתילאמינו אברמקטין ותכשירים קוטלי חרקים המכילים אותם

Info

Publication number
IL98599A
IL98599A IL9859991A IL9859991A IL98599A IL 98599 A IL98599 A IL 98599A IL 9859991 A IL9859991 A IL 9859991A IL 9859991 A IL9859991 A IL 9859991A IL 98599 A IL98599 A IL 98599A
Authority
IL
Israel
Prior art keywords
deoxy
epi
acid
avermectin
blb
Prior art date
Application number
IL9859991A
Other languages
English (en)
Other versions
IL98599A0 (en
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of IL98599A0 publication Critical patent/IL98599A0/xx
Publication of IL98599A publication Critical patent/IL98599A/he

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
IL9859991A 1990-06-28 1991-06-24 מלחים יציבים של " 4-דהאוקסי-" 4-אפי- מתילאמינו אברמקטין ותכשירים קוטלי חרקים המכילים אותם IL98599A (he)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US54522990A 1990-06-28 1990-06-28

Publications (2)

Publication Number Publication Date
IL98599A0 IL98599A0 (en) 1992-07-15
IL98599A true IL98599A (he) 1995-06-29

Family

ID=24175383

Family Applications (1)

Application Number Title Priority Date Filing Date
IL9859991A IL98599A (he) 1990-06-28 1991-06-24 מלחים יציבים של " 4-דהאוקסי-" 4-אפי- מתילאמינו אברמקטין ותכשירים קוטלי חרקים המכילים אותם

Country Status (21)

Country Link
US (1) US5288710A (he)
EP (1) EP0465121B1 (he)
JP (1) JPH0822870B2 (he)
KR (1) KR100224292B1 (he)
AT (1) ATE134377T1 (he)
AU (1) AU641777B2 (he)
CA (1) CA2045864C (he)
CY (1) CY1949A (he)
DE (1) DE69117223T2 (he)
DK (1) DK0465121T3 (he)
ES (1) ES2084110T3 (he)
FI (1) FI97890C (he)
GR (1) GR3019067T3 (he)
HK (1) HK157096A (he)
IE (1) IE71175B1 (he)
IL (1) IL98599A (he)
LV (1) LV5740B4 (he)
NO (2) NO2001007I2 (he)
NZ (1) NZ238705A (he)
PT (1) PT98117B (he)
ZA (1) ZA914961B (he)

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JP4701538B2 (ja) 2001-05-21 2011-06-15 住友化学株式会社 農業害虫防除剤組成物
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DE10203688A1 (de) * 2002-01-31 2003-08-07 Bayer Cropscience Ag Synergistische insektizide Mischungen
DE10207242A1 (de) * 2002-02-21 2003-09-04 Bayer Cropscience Ag Synergistische insektizide Mischungen
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TW200407330A (en) 2002-05-07 2004-05-16 Syngenta Participations Ag 4"-Deoxy-4"-(S)-amido avermectin derivatives
GB0302310D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin- and avermectin monosaccharide derivatives substituted in the 4"- or 4' - positionhaving pesticidal properties
GB0302308D0 (en) 2003-01-31 2003-03-05 Syngenta Participations Ag Avermectin and avermectin monosaccharide derivatives substituted in the 4"- or 4'-position having pesticidal properties
GB0320176D0 (en) 2003-08-28 2003-10-01 Syngenta Participations Ag Avermectins and avermectin monosaccharides substitued in the 4'-and 4"-positionhaving pesticidal properties
ATE406348T1 (de) 2004-09-23 2008-09-15 Schering Plough Ltd Bekämpfung von parasiten in tieren durch verwendung neuer trifluormethansulfonanilidoximetherderivate
WO2006055565A2 (en) * 2004-11-19 2006-05-26 Schering-Plough Ltd. Control of parasites in animals by the use of parasiticidal 2-phenyl-3-(1h-pyrrol-2-yl) acrylonitrile derivatives
PE20070108A1 (es) * 2005-06-09 2007-02-09 Schering Plough Ltd Control de parasitos en animales con derivados de n-[(feniloxi)fenil]-1,1,1-trifluorometansulfonamida y de n-[(fenilsulfanil)fenil]-1,1,1-trifluorometansulfonamida
US8119667B2 (en) * 2005-12-29 2012-02-21 Schering-Plough Animal Health Corporation Carbonates of fenicol antibiotics
EP1849363A1 (en) * 2006-03-09 2007-10-31 Cheminova A/S Synergistic combination of glutamate- and GABA-gated chloride agonist pesticide and at least one of Vitamin E or Niacin
US20070238700A1 (en) * 2006-04-10 2007-10-11 Winzenberg Kevin N N-phenyl-1,1,1-trifluoromethanesulfonamide hydrazone derivative compounds and their usage in controlling parasites
TWI422328B (zh) 2006-06-19 2014-01-11 Univ California 結合有殺線蟲之種子塗覆物的生物控制劑
FR2906469B1 (fr) * 2006-09-28 2008-11-28 Galderma Sa Utilisation de composes de la famille des avermectines pour le traitement de desordres dermatologiques chez l'homme
CA2672586A1 (en) * 2006-12-13 2008-06-26 Schering-Plough Ltd. Water-soluble prodrugs of florfenicol and its analogs
US8044230B2 (en) * 2006-12-13 2011-10-25 Intervet Inc. Water-soluble prodrugs of chloramphenicol, thiamphenicol, and analogs thereof
DE102007002872A1 (de) 2007-01-15 2008-07-17 Alpha-Biocare Gmbh Verwendung von Avermectin-Derivaten zur Behandlung gegen Parasiten von Fischen
TWI430995B (zh) 2007-06-26 2014-03-21 Du Pont 萘異唑啉無脊椎有害動物控制劑
CN101743000A (zh) 2007-06-27 2010-06-16 杜邦公司 动物虫害控制方法
TWI556741B (zh) 2007-08-17 2016-11-11 英特威特國際股份有限公司 異唑啉組成物及其作為抗寄生蟲藥上的應用
TWI401023B (zh) 2008-02-06 2013-07-11 Du Pont 中離子農藥
CA2732017A1 (en) * 2008-07-30 2010-02-04 Intervet International B.V. Process for preparing oxazoline-protected aminodiol compounds useful as intermediates to florfenicol
CA2755753A1 (en) 2009-03-17 2010-09-23 Intervet International B.V. Macrocyclic lactone drug delivery system
WO2011017334A2 (en) 2009-08-05 2011-02-10 E. I. Du Pont De Nemours And Company Mesoionic pesticides
UA107804C2 (en) 2009-08-05 2015-02-25 Du Pont Mixtures of pesticides mezoionnyh
EP2462125A2 (en) 2009-08-05 2012-06-13 E. I. du Pont de Nemours and Company Mesoionic pesticides
UA110924C2 (uk) 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Мезоіонні пестициди
MD4363C1 (ro) 2010-05-27 2016-03-31 E.I. Du Pont De Nemours And Company Forma cristalină a 4-[5-[3-cloro-5-(trifluorometil)fenil]-4,5-dihidro-5-(trifluorometil)-3-izoxazolil]-N-[2-oxo-2-[(2,2,2-trifluoroetil)amino]etil]-1-naftalencarboxamidei şi utilizările sale
AR081970A1 (es) 2010-06-24 2012-10-31 Intervet Int Bv Formulacion inyectable de una lactona macrociclica y levamisol, formulacion y uso veterinario
EP2629772B1 (en) 2010-10-20 2016-05-18 Galderma S.A. Ivermectin for use in the treatment of hemorrhoids
WO2012087630A1 (en) 2010-12-20 2012-06-28 E.I. Du Pont De Nemours And Company Pyridine and pyrimidine compounds for controlling invertebrate
PT2658542T (pt) 2010-12-27 2022-03-10 Intervet Int Bv Formulação de isoxazolina localizada tópica
EP2658541B1 (en) 2010-12-27 2022-01-26 Intervet International B.V. Topical localized isoxazoline formulation comprising glycofurol
WO2013015993A1 (en) 2011-07-28 2013-01-31 Syngenta Participations Ag Methods and compositions for controlling nematode pests
WO2013158422A1 (en) 2012-04-17 2013-10-24 E. I. Du Pont De Nemours And Company Heterocyclic compounds for controlling invertebrate pests
US9409920B1 (en) * 2015-06-08 2016-08-09 Rotam Agrochem International Company Limited Method for purifying emamectin benzoate and compositions comprising the same
US9643991B2 (en) * 2015-06-08 2017-05-09 Rotam Agrochem International Company Limited Process for preparing a novel crystalline form of emamectin benzoate and use the same
CN107344954B (zh) * 2017-08-07 2020-08-11 河北蓝泰化工科技有限公司 增效型甲氨基阿维菌素b1或b2的盐及制备方法和应用
CN108840893A (zh) * 2018-07-01 2018-11-20 李万强 一种甲氨基阿维菌素苯甲酸盐的新晶型及其制备方法
CN108864230B (zh) * 2018-07-26 2021-05-14 河北威远生物化工有限公司 一种有机磷基团取代的阿维菌素衍生物及其制备方法和应用

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Also Published As

Publication number Publication date
NZ238705A (en) 1993-07-27
KR920000781A (ko) 1992-01-29
ZA914961B (en) 1992-07-29
NO912535D0 (no) 1991-06-27
JPH0822870B2 (ja) 1996-03-06
NO912535L (no) 1991-12-30
IE912251A1 (en) 1992-01-01
DE69117223T2 (de) 1996-09-12
AU641777B2 (en) 1993-09-30
NO178339C (no) 1996-03-06
KR100224292B1 (ko) 1999-10-15
FI97890B (fi) 1996-11-29
FI913137A (fi) 1991-12-29
FI913137A0 (fi) 1991-06-27
ATE134377T1 (de) 1996-03-15
LV5740A4 (lv) 1996-08-20
ES2084110T3 (es) 1996-05-01
LV5740B4 (lv) 1997-12-20
NO2001007I2 (no) 2007-02-26
CY1949A (en) 1991-06-27
PT98117B (pt) 1998-12-31
EP0465121A1 (en) 1992-01-08
GR3019067T3 (en) 1996-05-31
DE69117223D1 (de) 1996-03-28
US5288710A (en) 1994-02-22
AU7939291A (en) 1992-01-02
IE71175B1 (en) 1997-01-29
CA2045864A1 (en) 1991-12-29
NO178339B (no) 1995-11-27
FI97890C (fi) 1997-03-10
PT98117A (pt) 1993-10-29
CA2045864C (en) 2001-11-27
DK0465121T3 (da) 1996-03-18
HK157096A (en) 1996-08-23
IL98599A0 (en) 1992-07-15
EP0465121B1 (en) 1996-02-21
JPH05306294A (ja) 1993-11-19

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