IL80729A0 - Thiazole derivatives,processes for the preparation thereof and pharmaceutical composition comprising the same - Google Patents

Thiazole derivatives,processes for the preparation thereof and pharmaceutical composition comprising the same

Info

Publication number
IL80729A0
IL80729A0 IL80729A IL8072986A IL80729A0 IL 80729 A0 IL80729 A0 IL 80729A0 IL 80729 A IL80729 A IL 80729A IL 8072986 A IL8072986 A IL 8072986A IL 80729 A0 IL80729 A0 IL 80729A0
Authority
IL
Israel
Prior art keywords
processes
preparation
same
pharmaceutical composition
thiazole derivatives
Prior art date
Application number
IL80729A
Other languages
English (en)
Original Assignee
Fujisawa Pharmaceutical Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fujisawa Pharmaceutical Co filed Critical Fujisawa Pharmaceutical Co
Publication of IL80729A0 publication Critical patent/IL80729A0/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/16—Otologicals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL80729A 1985-12-05 1986-11-23 Thiazole derivatives,processes for the preparation thereof and pharmaceutical composition comprising the same IL80729A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP27446585 1985-12-05
JP23687986 1986-10-03

Publications (1)

Publication Number Publication Date
IL80729A0 true IL80729A0 (en) 1987-02-27

Family

ID=26532916

Family Applications (1)

Application Number Title Priority Date Filing Date
IL80729A IL80729A0 (en) 1985-12-05 1986-11-23 Thiazole derivatives,processes for the preparation thereof and pharmaceutical composition comprising the same

Country Status (20)

Country Link
US (1) US4742057A (fi)
EP (1) EP0224919B1 (fi)
JP (1) JPS63225374A (fi)
KR (1) KR890003356B1 (fi)
CN (1) CN1017707B (fi)
AR (1) AR242574A1 (fi)
AT (1) ATE66224T1 (fi)
AU (1) AU601911B2 (fi)
CA (1) CA1311754C (fi)
DE (1) DE3680877D1 (fi)
DK (1) DK575386A (fi)
ES (1) ES2040206T3 (fi)
FI (1) FI87212C (fi)
GR (1) GR3002606T3 (fi)
HU (1) HU207315B (fi)
IE (1) IE59624B1 (fi)
IL (1) IL80729A0 (fi)
NO (1) NO165397C (fi)
PH (1) PH23004A (fi)
SU (2) SU1597102A3 (fi)

Families Citing this family (24)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IE58370B1 (en) * 1985-04-10 1993-09-08 Lundbeck & Co As H Indole derivatives
GB8726763D0 (en) * 1987-11-16 1987-12-23 Fujisawa Pharmaceutical Co Thiazole compounds
DK733788A (da) * 1988-01-14 1989-07-15 Fujisawa Pharmaceutical Co Indolylpiperidinderivater og fremgangsmaade til fremstilling deraf
GB8908085D0 (en) * 1989-04-11 1989-05-24 Lundbeck & Co As H New therapeutic use
US5238945A (en) * 1989-04-11 1993-08-24 H. Lundbeck A/S Method of treating psychoses
US5643784A (en) * 1990-12-04 1997-07-01 H, Lundbeck A/S Indan derivatives
NZ243065A (en) * 1991-06-13 1995-07-26 Lundbeck & Co As H Piperidine derivatives and pharmaceutical compositions
JP2600644B2 (ja) * 1991-08-16 1997-04-16 藤沢薬品工業株式会社 チアゾリルベンゾフラン誘導体
DK78692D0 (da) * 1992-06-12 1992-06-12 Lundbeck & Co As H Dimere piperidin- og piperazinderivater
US5457099A (en) * 1992-07-02 1995-10-10 Sawai Pharmaceutical Co., Ltd. Carbostyril derivatives and antiallergic agent
JP3719612B2 (ja) * 1993-06-14 2005-11-24 塩野義製薬株式会社 ヘテロ環を含有する尿素誘導体
US5521196A (en) * 1994-10-05 1996-05-28 Eli Lilly And Company 5-HT1F agonists for the treatment of migraine
US5521197A (en) * 1994-12-01 1996-05-28 Eli Lilly And Company 3-<1-alkylenearyl>-4-<1,2,3,6-tetrahydropyridinyl>-and 3-<1-alkylenearyl>-4-piperidinyl-1h-indoles: new 5-HT1F agonists
CN1184425A (zh) * 1995-03-20 1998-06-10 伊莱利利公司 5－取代－3－(1,2,3,6－四氢吡啶－4－基)－和3－(哌啶－4－基)－1h－吲哚:新型5－ht1f激动剂
CZ168896A3 (en) * 1995-06-27 1997-01-15 Egyt Gyogyszervegyeszeti Gyar Oxaindene derivatives and process for preparing thereof
ES2165274B1 (es) * 1999-06-04 2003-04-01 Almirall Prodesfarma Sa Nuevos derivados de indolilpiperidina como agentes antihistaminicos y antialergicos.
ES2172436B1 (es) * 2000-10-31 2004-01-16 Almirall Prodesfarma Sa Derivados de indolilpiperidina como agentes antihistaminicos y antialergicos.
ES2201907B1 (es) 2002-05-29 2005-06-01 Almirall Prodesfarma, S.A. Nuevos derivados de indolilpiperidina como potentes agentes antihistaminicos y antialergicos.
GB0328909D0 (en) * 2003-12-12 2004-01-14 Syngenta Participations Ag Chemical compounds
US20080015214A1 (en) * 2005-10-24 2008-01-17 Bignan Gilles C 3-piperidin-4-yl-indole orl-1 receptor modulators
DK3027603T3 (en) * 2013-08-02 2018-09-17 Pfizer HETEROBICYCLOARYL-RORC2 INHIBITORS AND METHODS FOR USING IT
US20150315179A1 (en) * 2014-05-02 2015-11-05 Torrey Pines Institute For Molecular Studies Compounds and methods of treating neurological disorders
JP2018510131A (ja) 2015-01-30 2018-04-12 ファイザー・インク Ｒｏｒｃ２のスルホンアミド置換インドールモジュレーターおよびその使用方法
EP3250570A1 (en) 2015-01-30 2017-12-06 Pfizer Inc Methoxy-substituted pyrrolopyridine modulators of rorc2 and methods of use thereof

Family Cites Families (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3361759A (en) * 1963-10-07 1968-01-02 Upjohn Co 3-(2-pyrrolidinyl)-indoles and method of preparation
FR2193584B1 (fi) * 1972-07-28 1975-08-08 Roussel Uclaf
US3873559A (en) * 1973-03-30 1975-03-25 Squibb & Sons Inc Heterocyclic carboxamido thiazolinyl indoles
DE2322470A1 (de) * 1973-05-04 1974-11-21 Boehringer Sohn Ingelheim Neue indolyl-piperidino-(bzw. 1,2,5,6tetrahydro-pyridyl-)butyrophenone und verfahren zu ihrer herstellung
IL48508A (en) * 1974-12-09 1979-10-31 Roussel Uclaf Pharmaceutical compositions comprising piperidylindole derivatives
FR2349331A1 (fr) * 1976-04-30 1977-11-25 Roussel Uclaf Nouveaux derives de 2,3 dihydro a/4-(3-indolyl) 1-piperidinyl/methyl 1,4-benzodioxin-2-methanol, un procede pour leur preparation et leur application comme medicaments
FR2362628A1 (fr) * 1976-08-26 1978-03-24 Roussel Uclaf Nouveaux derives du piperidyl-indole et leurs sels, procede de preparation et application a titre de medicaments
FR2421899A1 (fr) * 1978-01-16 1979-11-02 Roussel Uclaf Nouveaux derives du tetrahydropyridinyl-indole et leurs sels, le procede de preparation et l'application a titre de medicaments de ces nouveaux produits
FR2426465B1 (fi) * 1978-01-16 1983-04-29 Roussel Uclaf
FR2460947A1 (fr) * 1979-07-13 1981-01-30 Roussel Uclaf Nouveau derives n-substitues du tetrahydropyridinyl-indole, leurs sels, procede de preparation, application a titre de medicaments et compositions les renfermant
US4359468A (en) * 1981-02-25 1982-11-16 Boehringer Ingelheim Ltd. Antiallergic N-[4-(indolyl)-piperidino-alkyl]-benzimidazolones
FR2533924A1 (fr) * 1982-10-05 1984-04-06 Roussel Uclaf Nouveaux derives du 4-(1h-indol-3-yl)a-methyl piperidine-1-ethanol, leurs sels, le procede de preparation, l'application a titre de medicaments et les compositions les renfermant
US4548939A (en) * 1984-10-01 1985-10-22 Janssen Pharmaceutica N. V. 1H-Indol-3-yl containing 1,3-dimethyl-1H-purine-2,6-diones
IE58370B1 (en) * 1985-04-10 1993-09-08 Lundbeck & Co As H Indole derivatives

Also Published As

Publication number Publication date
FI864879A0 (fi) 1986-12-01
CN86108205A (zh) 1987-06-17
NO864879D0 (no) 1986-12-04
KR890003356B1 (ko) 1989-09-19
AU601911B2 (en) 1990-09-20
DK575386D0 (da) 1986-11-28
ES2040206T3 (es) 1993-10-16
EP0224919A3 (en) 1988-03-30
IE59624B1 (en) 1994-03-09
NO165397B (no) 1990-10-29
KR870006039A (ko) 1987-07-08
US4742057A (en) 1988-05-03
HU207315B (en) 1993-03-29
FI864879A (fi) 1987-06-06
FI87212C (fi) 1992-12-10
CN1017707B (zh) 1992-08-05
DK575386A (da) 1987-06-06
IE863103L (en) 1987-06-05
ATE66224T1 (de) 1991-08-15
SU1753948A3 (ru) 1992-08-07
AR242574A1 (es) 1993-04-30
PH23004A (en) 1989-02-24
HUT46320A (en) 1988-10-28
DE3680877D1 (de) 1991-09-19
FI87212B (fi) 1992-08-31
CA1311754C (en) 1992-12-22
JPS63225374A (ja) 1988-09-20
SU1597102A3 (ru) 1990-09-30
GR3002606T3 (en) 1993-01-25
AU6581086A (en) 1987-06-11
NO864879L (no) 1987-06-09
EP0224919B1 (en) 1991-08-14
NO165397C (no) 1991-02-06
EP0224919A2 (en) 1987-06-10

Similar Documents

Publication Publication Date Title
IL77762A (en) 11beta-phenyl gonane derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same
IL80729A0 (en) Thiazole derivatives,processes for the preparation thereof and pharmaceutical composition comprising the same
HK18194A (en) Substituted benzamide derivatives,processes for the preparation thereof,and pharmaceutical compositions containing the same
EP0201741A3 (en) Dipeptide derivatives, processes for preparing them, pharmaceutical composition and use
EP0157346A3 (en) Quinolizinone compound, processes for preparation thereof and pharmaceutical composition comprising the same
IL80160A (en) Beta-lactam derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same
IL92939A0 (en) Thiazole derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same
IL84913A0 (en) Alkanesulfonanilide derivatives,processes for preparation thereof and pharmaceutical composition comprising the same
IL88903A0 (en) Indolylpiperidine derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same
IL95548A0 (en) Thiazole derivatives,processes for the preparation thereof and pharmaceutical composition containing the same
EP0168005A3 (en) Semicarbazide derivatives, processes for preparation thereof and pharmaceutical composition comprising the same
GB8917687D0 (en) Aminopiperazine derivatives,processes for preparation thereof and pharmaceutical composition comprising the same
AU8146587A (en) New benzothiadiazine compounds, processes for the preparation thereof and pharmaceutical composition comprising the same
IL78576A0 (en) 5-pyrimidinecarboxamide,processes for the preparation thereof and pharmaceutical compositions containing same
IL87563A0 (en) Isoxazole-beta-carboline derivatives,processes for the preparation thereof and pharmaceutical compositions containing the same
GB2179347B (en) Methylenedioxyphenanthrene and -stilbene derivatives, processes for the preparation thereof and pharmaceutical compositions containing them
IL84210A0 (en) Thiadiazole derivative,processes for preparation thereof and pharmaceutical compositions comprising the same
ZA879706B (en) New alkanesulfonanilide derivatives,processes for preparation thereof and pharmaceutical composition comprising the same
IL76837A0 (en) Benzimidazole derivatives,processes for the preparation thereof and pharmaceutical compositions containing them
ZA873022B (en) Substituted benzamide derivatives,processes for the preparation thereof,and pharmaceutical compositions containing the same
ZA868751B (en) New thiazole compounds,processes for the preparation thereof and pharmaceutical composition comprising the same
ZA853658B (en) Semicarbazide derivatives,processes for preparation thereof and pharmaceutical composition comprising the same
ZA883534B (en) New alkanesulfonanilide derivatives,processes for preparation thereof and pharmaceutical composition comprising the same
ZA906638B (en) New thiazole derivatives,processes for the preparation thereof and pharmaceutical composition comprising the same
ZA847850B (en) Thiazine derivatives,processes for preparation thereof and pharmaceutical composition comprising the same

Legal Events

Date Code Title Description
RH Patent void