IL57533A - 17alpha-acetylene derivatives of androst-4-ene,process for preparing them and pharmaceutical compositions containing them - Google Patents

17alpha-acetylene derivatives of androst-4-ene,process for preparing them and pharmaceutical compositions containing them

Info

Publication number
IL57533A
IL57533A IL57533A IL5753379A IL57533A IL 57533 A IL57533 A IL 57533A IL 57533 A IL57533 A IL 57533A IL 5753379 A IL5753379 A IL 5753379A IL 57533 A IL57533 A IL 57533A
Authority
IL
Israel
Prior art keywords
17alpha
androst
ene
preparing
pharmaceutical compositions
Prior art date
Application number
IL57533A
Other languages
English (en)
Other versions
IL57533A0 (en
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Priority to IL6869379A priority Critical patent/IL68693A/xx
Publication of IL57533A0 publication Critical patent/IL57533A0/xx
Priority to IL68693A priority patent/IL68693A0/xx
Publication of IL57533A publication Critical patent/IL57533A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003—Androstane derivatives
    • C07J1/0033—Androstane derivatives substituted in position 17 alfa and 17 beta
    • C07J1/004—Androstane derivatives substituted in position 17 alfa and 17 beta the substituent in position 17 alfa being an unsaturated hydrocarbon group
    • C07J1/0048—Alkynyl derivatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003—Androstane derivatives
    • C07J1/0011—Androstane derivatives substituted in position 17 by a keto group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J1/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, not substituted in position 17 beta by a carbon atom, e.g. estrane, androstane
    • C07J1/0003—Androstane derivatives
    • C07J1/0033—Androstane derivatives substituted in position 17 alfa and 17 beta

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Rheumatology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
IL57533A 1978-07-13 1979-06-11 17alpha-acetylene derivatives of androst-4-ene,process for preparing them and pharmaceutical compositions containing them IL57533A (en)

Priority Applications (2)

Application Number Priority Date Filing Date Title
IL6869379A IL68693A (en) 1978-07-13 1979-06-11 3-ethoxy-11beta-hydroxy-6-methylandrosta-3,5-dien-17-one and its preparation
IL68693A IL68693A0 (en) 1978-07-13 1983-05-13 3-ethoxy-11beta-hydroxy-6-methyl-androsta-3,5-dien-17-one and its preparation

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
FR7820971A FR2430952A1 (fr) 1978-07-13 1978-07-13 Nouveaux derives acetyleniques de l'androst 4-ene, leur procede de preparation et leur application comme medicament

Publications (2)

Publication Number Publication Date
IL57533A0 IL57533A0 (en) 1979-10-31
IL57533A true IL57533A (en) 1984-01-31

Family

ID=9210731

Family Applications (1)

Application Number Title Priority Date Filing Date
IL57533A IL57533A (en) 1978-07-13 1979-06-11 17alpha-acetylene derivatives of androst-4-ene,process for preparing them and pharmaceutical compositions containing them

Country Status (24)

Country Link
US (1) US4233297A (es)
JP (2) JPS5515474A (es)
AT (1) AT370109B (es)
AU (1) AU534841B2 (es)
BE (1) BE877658A (es)
CA (1) CA1140110A (es)
CH (2) CH641475A5 (es)
DE (2) DE2954699C2 (es)
DK (1) DK160560C (es)
ES (1) ES8101081A1 (es)
FR (1) FR2430952A1 (es)
GB (2) GB2025422B (es)
GR (1) GR81403B (es)
HU (1) HU180519B (es)
IL (1) IL57533A (es)
IT (1) IT1164697B (es)
LU (1) LU81497A1 (es)
MA (1) MA18516A1 (es)
NL (1) NL7905481A (es)
OA (1) OA06258A (es)
PH (1) PH17055A (es)
PT (1) PT69906A (es)
SE (1) SE440781B (es)
ZA (1) ZA793100B (es)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2547587B1 (fr) * 1983-06-14 1985-10-25 Roussel Uclaf Steroides radioactifs, leur procede de preparation, leur application a la mise en evidence des recepteurs de glucocorticoides et au dosage du nombre de sites de fixation
FR2644788B1 (fr) * 1989-03-22 1995-02-03 Roussel Uclaf Nouveaux steroides 3-ceto comportant une chaine en 17 amino-substituee, leur procede de preparation et les intermediaires de ce procede, leur application comme medicaments et les compositions pharmaceutiques les contenant
JPH02141007U (es) * 1989-04-26 1990-11-27
EP0485392B1 (en) * 1989-07-07 1998-09-09 Endorecherche Inc. Androgen derivatives for use in the inhibition of sex steroid activity
AU680818B2 (en) * 1992-05-21 1997-08-14 Endorecherche Inc. Improved antiandrogens
JP2741286B2 (ja) * 1993-05-17 1998-04-15 アンドルシェルシュ・インコーポレイテッド 改良された抗アンドロゲン
CN103145785B (zh) * 2013-03-19 2016-03-02 浙江仙居仙乐药业有限公司 一种醋酸环丙孕酮脱氢物的合成方法

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2740798A (en) * 1953-05-25 1956-04-03 Searle & Co 11 beta-hydroxy-17-ethynyl testosterone and esters thereof
US3010957A (en) * 1958-11-26 1961-11-28 Schering Corp Ethinyl androstadienes
FR1349113A (fr) * 1959-01-28 1964-01-17 Upjohn Co Procédé de fabrication de 6-fluoro-11 oxygéné-17-bêta-hydroxy-17 alpha-alkynyl inférieur-4-androstène-3-ones et leurs dérivés acylés
US3793308A (en) * 1972-11-08 1974-02-19 Upjohn Co 4-spiro(cyclopropyl)androstenes and process for their production
SE7801152L (sv) * 1977-02-22 1978-08-23 Roussel Uclaf Sett att framstella 17alfa-acetylen-derivat av androst-4-en

Also Published As

Publication number Publication date
PH17055A (en) 1984-05-17
DE2954699C2 (es) 1992-04-16
AU4889479A (en) 1980-01-17
MA18516A1 (fr) 1980-04-01
GR81403B (es) 1984-12-11
FR2430952B1 (es) 1980-12-05
IT1164697B (it) 1987-04-15
OA06258A (fr) 1981-06-30
AU534841B2 (en) 1984-02-16
SE7904431L (sv) 1980-01-14
DE2928374A1 (de) 1980-01-31
HU180519B (en) 1983-03-28
DK160560C (da) 1991-09-09
BE877658A (fr) 1980-01-14
AT370109B (de) 1983-03-10
LU81497A1 (fr) 1980-02-14
SE440781B (sv) 1985-08-19
IT7949743A0 (it) 1979-07-12
CH641475A5 (fr) 1984-02-29
GB2108503A (en) 1983-05-18
DK292679A (da) 1980-01-14
DE2928374C2 (es) 1991-12-12
ES482387A0 (es) 1980-12-01
ATA488979A (de) 1982-07-15
US4233297A (en) 1980-11-11
ZA793100B (en) 1980-06-25
ES8101081A1 (es) 1980-12-01
IL57533A0 (en) 1979-10-31
FR2430952A1 (fr) 1980-02-08
JPS6345295A (ja) 1988-02-26
JPS6252758B2 (es) 1987-11-06
CA1140110A (fr) 1983-01-25
CH642977A5 (fr) 1984-05-15
GB2025422A (en) 1980-01-23
GB2108503B (en) 1983-09-14
GB2025422B (en) 1983-05-05
JPS6362515B2 (es) 1988-12-02
PT69906A (fr) 1979-08-01
DK160560B (da) 1991-03-25
JPS5515474A (en) 1980-02-02
NL7905481A (nl) 1980-01-15

Similar Documents

Publication Publication Date Title
DE2960553D1 (en) Derivatives of carbazolyl-4-oxypropanolamine, methods for their preparation and medicines containing them
DE2960222D1 (en) Phenoxyalkylcarboxylic-acid derivatives, process for their preparation and medicaments containing them
DE2960178D1 (en) New substituted phenylpiperazine derivatives, pharmaceutical compositions containing them and process for their preparation
DE2965279D1 (en) Indanyl derivatives, process for their preparation and pharmaceutical compositions containing these compounds
PT69821A (en) Process for the preparation of new 5-phenylpyrazole derivatives the salts thereof and the pharmaceutical compositions containing same
DE2961571D1 (en) Penicillins, their salts, process for their preparation and pharmaceutical compositions containing them
DE2963573D1 (en) Isoquinoline derivatives, process for their preparation and pharmaceutical compositions containing them
DE2964209D1 (en) Spiro-furanohydantoin derivatives, process for their preparation and pharmaceutical compositions containing them
DE2961983D1 (en) Pyrrolidine-2-methanol derivatives, process for their preparation and medicaments containing them
DE2962112D1 (en) Alkanolamine derivatives, process for their preparation and pharmaceutical compositions containing them
IL54069A (en) 14,15-dihydro-20,21-dinoreburnamenin-14-ol derivatives,process for preparing them and pharmaceutical compositions containing them
IL57533A (en) 17alpha-acetylene derivatives of androst-4-ene,process for preparing them and pharmaceutical compositions containing them
ZA793682B (en) New piperidylbenzimidazolinone derivatives,processes for their preparation and pharmaceutical compositions containing them
GB2038802B (en) Aryltrifluoroethanols process for their preparation and pharmaceutical compositions containing them
DE2964198D1 (en) Indanamine derivatives, process for their preparation and medicaments containing them
HUT36099A (en) Pharmaceutical compositions containing process for preparing 4-aroyl-imidazol-2-one derivatives
DE2860212D1 (en) 4-phenyl-8-amino-tetrahydroisoquinolines, pharmaceutical compositions containing them and process for preparation of these compositions
DE2967215D1 (en) Isoquinoline derivatives, process for their preparation, intermediates and pharmaceutical compositions containing them
DE2966639D1 (en) Benzodiazepine derivatives, process for their preparation and pharmaceutical compositions containing them
DE2962303D1 (en) Derivatives of ergopeptide alkaloids, process for their preparation and pharmaceutical compositions containing them
EP0012641A3 (en) 2-substituted-19-nor-pregn-4-ene-3,20-dione derivatives, process for their preparation, pharmaceutical compositions containing them, and intermediates
IL61602A0 (en) New derivatives of 1-aminopropan-2-ol,process for preparing them and pharmaceutical compositions containing them
IL54070A0 (en) 17 -acetylene derivatives of androst-4-ene, process for preparing them and pharmaceutical compositions
DE2960205D1 (en) 4-hydroxy-2-benzimidazolin-thion derivatives, process for their preparation and medicaments containing them
HK58085A (en) Novel azathianaphthalene derivatives,process for their manufacture,pharmaceutical preparations containing them and their use

Legal Events

Date Code Title Description
KB Patent renewed