IL49205A - 5-chloro-4-(2-imidazolin-2-ylamino)-2,1,3-benzothiadiazole its production and pharmaceutical compositions containing it - Google Patents

5-chloro-4-(2-imidazolin-2-ylamino)-2,1,3-benzothiadiazole its production and pharmaceutical compositions containing it

Info

Publication number
IL49205A
IL49205A IL49205A IL4920573A IL49205A IL 49205 A IL49205 A IL 49205A IL 49205 A IL49205 A IL 49205A IL 4920573 A IL4920573 A IL 4920573A IL 49205 A IL49205 A IL 49205A
Authority
IL
Israel
Prior art keywords
compound
formula
chloro
halogen
production
Prior art date
Application number
IL49205A
Other languages
English (en)
Other versions
IL49205A0 (en
Original Assignee
Wander Ag Dr A
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wander Ag Dr A filed Critical Wander Ag Dr A
Publication of IL49205A0 publication Critical patent/IL49205A0/xx
Publication of IL49205A publication Critical patent/IL49205A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/14—Thiadiazoles; Hydrogenated thiadiazoles condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
IL49205A 1972-05-09 1973-05-08 5-chloro-4-(2-imidazolin-2-ylamino)-2,1,3-benzothiadiazole its production and pharmaceutical compositions containing it IL49205A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH686572A CH570401A5 (nl) 1972-05-09 1972-05-09

Publications (2)

Publication Number Publication Date
IL49205A0 IL49205A0 (en) 1976-05-31
IL49205A true IL49205A (en) 1977-05-31

Family

ID=4316243

Family Applications (2)

Application Number Title Priority Date Filing Date
IL49205A IL49205A (en) 1972-05-09 1973-05-08 5-chloro-4-(2-imidazolin-2-ylamino)-2,1,3-benzothiadiazole its production and pharmaceutical compositions containing it
IL42231A IL42231A (en) 1972-05-09 1973-05-09 4-(2-imidazolin-2-ylamino)-2,1,3-benzothiadiazole derivatives their production and pharmaceutical compositions containing them

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL42231A IL42231A (en) 1972-05-09 1973-05-09 4-(2-imidazolin-2-ylamino)-2,1,3-benzothiadiazole derivatives their production and pharmaceutical compositions containing them

Country Status (26)

Country Link
US (1) US3843668A (nl)
JP (3) JPS5533718B2 (nl)
AT (1) AT336006B (nl)
BE (1) BE799332A (nl)
CH (1) CH570401A5 (nl)
CS (2) CS202052B2 (nl)
CY (1) CY989A (nl)
DD (1) DD106180A5 (nl)
DE (1) DE2322880C2 (nl)
DK (1) DK135454B (nl)
ES (3) ES414470A1 (nl)
FI (1) FI60010C (nl)
FR (1) FR2183930B1 (nl)
GB (2) GB1429926A (nl)
HK (1) HK11179A (nl)
HU (1) HU166329B (nl)
IE (1) IE38012B1 (nl)
IL (2) IL49205A (nl)
MY (1) MY7900117A (nl)
NL (1) NL161445C (nl)
NO (1) NO138566C (nl)
PL (1) PL89214B1 (nl)
SE (1) SE386445B (nl)
SU (1) SU493966A3 (nl)
YU (4) YU36174B (nl)
ZA (1) ZA733143B (nl)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5930899B2 (ja) * 1973-02-01 1984-07-30 隆弘 上野 内燃機関の制動方法及びその装置
GB1559811A (en) * 1975-07-28 1980-01-30 Sandoz Ltd Pharmaceutically active benzothiadiazole derivatives
CH613966A5 (en) * 1975-08-22 1979-10-31 Sandoz Ag Process for the preparation of novel 5-(2-imidazolin-2-ylamino)-2,1,3-benzothiadiazoles
US4217356A (en) * 1975-08-22 1980-08-12 Sandoz Ltd. 2-Imidazolinylamino-2,1,3-benzothiadiazoles
CH632268A5 (de) * 1977-01-14 1982-09-30 Sandoz Ag Verfahren zur herstellung von neuen heterocyclylaminoderivaten.
FR2499991A1 (fr) * 1981-02-19 1982-08-20 Sandoz Sa Nouveaux 2,1,3-benzothiadiazoles et 2,1,3-benzoxadiazoles, leur preparation et leur application comme medicaments
FR2502951B1 (fr) * 1981-04-06 1985-12-06 Sandoz Sa Compositions pharmaceutiques topiques sous forme d'une micro-emulsion
JPS5826094U (ja) * 1981-08-13 1983-02-19 ヤマハ株式会社 電子楽器の制御装置
JPS61268828A (ja) * 1985-05-22 1986-11-28 Kubota Ltd 圧縮空気取出装置付き容積形内燃機関
JPH0622121Y2 (ja) * 1988-01-18 1994-06-08 川崎重工業株式会社 空気圧縮機兼用多気筒エンジン
JP2668816B2 (ja) * 1993-09-09 1997-10-27 株式会社パーマケム・アジア ベンゾチアジアゾール誘導体の製法
US6455557B1 (en) 2001-11-28 2002-09-24 Elan Pharmaceuticals, Inc. Method of reducing somnolence in patients treated with tizanidine
US20040220240A1 (en) * 2001-11-28 2004-11-04 Pellegrini Cara A. Method of increasing the extent of absorption of tizanidine
IL163666A0 (en) 2002-02-22 2005-12-18 New River Pharmaceuticals Inc Active agent delivery systems and methods for protecting and administering active agents
GB0224198D0 (en) * 2002-10-17 2002-11-27 Novartis Ag Organic compounds
EP2218442A1 (en) 2005-11-09 2010-08-18 CombinatoRx, Inc. Methods, compositions, and kits for the treatment of ophthalmic disorders
WO2008008394A1 (en) * 2006-07-12 2008-01-17 Transform Pharmaceuticals, Inc. Tizanidine succinate salt forms and methods of making and using the same
US8524749B2 (en) * 2007-02-09 2013-09-03 Alza Corporation Controlled release compositions of tizanidine
CZ301889B6 (cs) 2008-12-18 2010-07-21 Farmak, A. S. Zpusob prípravy tizanidinu hydrochloridu
ES2637387T3 (es) 2011-10-24 2017-10-13 Braeburn Pharmaceuticals, Inc. Composiciones de tizanidina implantables y procedimientos de tratamiento asociados
CN106946874A (zh) * 2017-04-07 2017-07-14 四川智强医药科技开发有限公司 替扎尼定的脱色方法

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1211341A (fr) * 1955-12-19 1960-03-15 A Wander Dr Procédé pour la préparation de 2-amino-imidazolines
BE754832A (fr) * 1969-08-14 1971-02-15 Beecham Group Ltd Iminazolines

Also Published As

Publication number Publication date
IE38013L (en) 1973-11-09
GB1429683A (en) 1976-03-24
DK135454C (nl) 1977-10-17
AT336006B (de) 1977-04-12
FI60010B (fi) 1981-07-31
FI60010C (fi) 1981-11-10
CY989A (en) 1979-08-02
JPS562071B2 (nl) 1981-01-17
YU119673A (en) 1981-06-30
NL7306228A (nl) 1973-11-13
DE2322880C2 (de) 1982-09-23
FR2183930B1 (nl) 1976-03-05
ES440599A1 (es) 1977-05-16
MY7900117A (en) 1979-12-31
NL161445C (nl) 1980-02-15
GB1429926A (en) 1976-03-31
HK11179A (en) 1979-03-16
CH570401A5 (nl) 1975-12-15
DD106180A5 (nl) 1974-06-05
YU36025B (en) 1981-11-13
DE2322880A1 (de) 1973-11-22
CS208788B2 (en) 1981-09-15
DK135454B (da) 1977-05-02
NO138566C (no) 1978-09-27
NO138566B (no) 1978-06-19
IL42231A0 (en) 1973-07-30
ES414470A1 (es) 1976-05-01
YU36174B (en) 1982-02-25
PL89214B1 (nl) 1976-11-30
JPS4954370A (nl) 1974-05-27
IL42231A (en) 1977-06-30
YU36024B (en) 1981-11-13
CS202052B2 (en) 1980-12-31
JPS5533718B2 (nl) 1980-09-02
YU36026B (en) 1981-11-13
IL49205A0 (en) 1976-05-31
ES440598A1 (es) 1977-05-16
YU50679A (en) 1981-04-30
IE38012B1 (en) 1977-12-07
NL161445B (nl) 1979-09-17
ZA733143B (en) 1975-01-29
US3843668A (en) 1974-10-22
YU50479A (en) 1981-04-30
JPS5350168A (en) 1978-05-08
SE386445B (sv) 1976-08-09
JPS5543081A (en) 1980-03-26
FR2183930A1 (nl) 1973-12-21
YU50579A (en) 1981-04-30
JPS5442983B2 (nl) 1979-12-17
BE799332A (fr) 1973-11-09
AU5540873A (en) 1974-11-14
ATA403273A (de) 1976-08-15
SU493966A3 (ru) 1975-11-28
HU166329B (nl) 1975-02-28

Similar Documents

Publication Publication Date Title
IL49205A (en) 5-chloro-4-(2-imidazolin-2-ylamino)-2,1,3-benzothiadiazole its production and pharmaceutical compositions containing it
CA1152515A (en) Imidazole derivatives, their production and use
US3505350A (en) Certain substituted 2-mercaptoimidazole derivatives
US3282938A (en) 3-tertiary aminoloweralkyl-4-lower alkyl or phenyl-7-lower carbalkoxy lower alkyl or carboxy lower alkyl coumarins
IE53274B1 (en) Chemical compounds derived from cyclobutene
US4518712A (en) Piperazine derivative and analgesic composition containing the same
US2746960A (en) New chemotherapeutic nitrofurans
US3681360A (en) Antiviral substituted acridanones
US4163785A (en) Benzothiazepine compounds and compositions
US3740401A (en) 2-(n-cycloalkyl-phenylamino)-2-imidazolines-(2) and salts thereof
CA1154015A (en) Tetrahydroquinoline derivatives, a process for their preparation, their use, and pharmaceutical formulations containing them
US2786059A (en) Derivatives of 2-nu-methyl-1, 2, 3, 4-tetrahydro-gamma-carbolines
US3655685A (en) 2-(imidazolid inylidence-(2)-amino)-5-nitro-thiazoles and salts thereof
JPS6136754B2 (nl)
US3423424A (en) 3-phenyl-4-dialkylaminoalkyl-pyrazol-5-ol compounds
SE438857B (sv) Sett att framstella kromonderivat
CA1159828A (en) Process for preparing new 1,2,4-oxadiazine derivatives
US3350407A (en) Sulfur containing pyrazole derivatives
US3449354A (en) 2-((2-trifluoromethylphenoxy)methyl)-2-imidazoline
US4128550A (en) 1-Methyl-4-piperidyl 5-phenyl-2-furoates
US3812135A (en) Pyrroloindole and pyridoindole derivatives
US3100772A (en) Method for preparing phenothiazine derivatives
US3347862A (en) Piperazine 2, 6-diiodo-4-nitrophenyl phosphate
CS208746B2 (en) Method of making the 3,6-disubstituted-1,2,4-triazin 5-ons
US2807616A (en) Oxazolopyrimidines and method of preparing same