IL41170A - 2-Carbalkoxy-amino-benzimidazole) 6 (5-Phenyl sites with activity against worms and a process for their preparation - Google Patents
2-Carbalkoxy-amino-benzimidazole) 6 (5-Phenyl sites with activity against worms and a process for their preparationInfo
- Publication number
- IL41170A IL41170A IL41170A IL4117072A IL41170A IL 41170 A IL41170 A IL 41170A IL 41170 A IL41170 A IL 41170A IL 4117072 A IL4117072 A IL 4117072A IL 41170 A IL41170 A IL 41170A
- Authority
- IL
- Israel
- Prior art keywords
- amino
- formula
- benzimidazole
- methyl
- diphenyl ether
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/30—Nitrogen atoms not forming part of a nitro radical
- C07D235/32—Benzimidazole-2-carbamic acids, unsubstituted or substituted; Esters thereof; Thio-analogues thereof
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Fodder In General (AREA)
- Plural Heterocyclic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE2164690A DE2164690C3 (de) | 1971-12-27 | 1971-12-27 | Anthelmintisch wirksame 5-Phenoxy- und 5-Phenylthiobenzimidazolyl-(2)-carbamin-säuremethylester und Verfahren zu ihrer Herstellung |
Publications (2)
Publication Number | Publication Date |
---|---|
IL41170A0 IL41170A0 (en) | 1973-02-28 |
IL41170A true IL41170A (en) | 1977-01-31 |
Family
ID=5829297
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL41170A IL41170A (en) | 1971-12-27 | 1972-12-25 | 2-Carbalkoxy-amino-benzimidazole) 6 (5-Phenyl sites with activity against worms and a process for their preparation |
Country Status (30)
Country | Link |
---|---|
US (1) | US3954791A (fi) |
JP (1) | JPS5033067B2 (fi) |
KR (1) | KR780000116B1 (fi) |
AT (1) | AT320638B (fi) |
AU (1) | AU465226B2 (fi) |
BE (1) | BE793358A (fi) |
BG (2) | BG20591A3 (fi) |
CA (1) | CA1017750A (fi) |
CH (2) | CH583710A5 (fi) |
CS (2) | CS173650B2 (fi) |
DD (2) | DD109219A5 (fi) |
DE (1) | DE2164690C3 (fi) |
DK (1) | DK130293B (fi) |
EG (1) | EG11122A (fi) |
ES (1) | ES409860A1 (fi) |
FI (1) | FI54299C (fi) |
FR (1) | FR2166048B1 (fi) |
GB (1) | GB1360180A (fi) |
HU (1) | HU165060B (fi) |
IL (1) | IL41170A (fi) |
IT (1) | IT1043888B (fi) |
KE (1) | KE2613A (fi) |
MY (1) | MY7600092A (fi) |
NL (1) | NL153187B (fi) |
NO (1) | NO137092C (fi) |
PL (1) | PL85192B1 (fi) |
RO (1) | RO71503A (fi) |
SE (1) | SE395890B (fi) |
SU (2) | SU492086A3 (fi) |
ZA (1) | ZA729076B (fi) |
Families Citing this family (30)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3965113A (en) * | 1972-12-29 | 1976-06-22 | Syntex (U.S.A.) Inc. | 5(6)-Benzene ring substituted benzimidazole-2-carbamate derivatives having anthelmintic activity |
HU169503B (fi) * | 1974-02-05 | 1976-12-28 | ||
RO64921A (fr) * | 1974-05-28 | 1979-07-15 | Syntex Inc | Procede pour la preparation des derives des benzimidazole-2-carbamates |
DE2432631A1 (de) * | 1974-07-06 | 1976-01-22 | Hoechst Ag | 5-phenylsulfinyl-2-benzimidazol-carbaminsaeureester und verfahren zu ihrer herstellung |
DE2441201C2 (de) * | 1974-08-28 | 1986-08-07 | Hoechst Ag, 6230 Frankfurt | Anthelminthisch wirksame 2-Carbalkoxyamino-5(6)-phenyl-sulfonyloxy-benzimidazole und Verfahren zu ihrer Herstellung |
DE2441202C2 (de) * | 1974-08-28 | 1986-05-28 | Hoechst Ag, 6230 Frankfurt | 2-Carbalkoxyamino-benzimidazolyl-5(6)-sulfonsäure-phenylester, Verfahren zu ihrer Herstellung und diese enthaltende anthelmintische Mittel |
US4076828A (en) * | 1977-02-17 | 1978-02-28 | E. R. Squibb & Sons, Inc. | Method of treating helminthiasis by parenteral administration of sulfoxide derivatives of benzimidazoles |
US4076825A (en) * | 1977-06-22 | 1978-02-28 | E. R. Squibb & Sons, Inc. | Method of treating helminthiasis by parenteral or topical administration of sulfoxide derivatives of benzimidazoles |
US4076827A (en) * | 1977-04-28 | 1978-02-28 | E. R. Squibb & Sons, Inc. | Method of treating helminthiasis by parenteral administration of sulfoxide derivatives of benzimidazoles |
IT1076022B (it) * | 1977-04-20 | 1985-04-22 | Montedison Spa | Benzimidazolcarbammati antielmintici |
SE443977B (sv) * | 1977-05-10 | 1986-03-17 | Chinoin Gyogyszer Es Vegyeszet | Forfarande for framstellning av 5(6)-tio-bensimidazolderivat |
US4136174A (en) * | 1978-01-18 | 1979-01-23 | E. R. Squibb & Sons, Inc. | Benzimidazolecarbamates and method |
US4156006A (en) * | 1978-01-09 | 1979-05-22 | E. R. Squibb & Sons, Inc. | Vinyl sulfide derivatives of benzimidazoles |
US4154846A (en) * | 1978-06-16 | 1979-05-15 | E. R. Squibb & Sons, Inc. | Substituted thio-, sulfinyl-, and sulfonyl-alkyl benzimidazole carbamates |
EP0028455A1 (en) * | 1979-10-12 | 1981-05-13 | Imperial Chemical Industries Plc | 5-Phenylselenobenzimidazole derivatives, their preparation and anthelmintic or fasciolicidal compositions containing them |
US4299837A (en) | 1979-12-05 | 1981-11-10 | Montedison S.P.A. | Anthelmintic benzimidazole-carbamates |
US4662935A (en) * | 1980-01-14 | 1987-05-05 | Rohm And Haas Company | Herbicidal 4-trifluoromethyl-4-nitrodiphenyl ethers |
EP0060810B1 (de) * | 1981-03-18 | 1984-10-17 | Ciba-Geigy Ag | Anthelmintika |
IE56125B1 (en) * | 1982-10-28 | 1991-04-24 | Ici Plc | Indole derivatives |
WO1990010630A1 (en) * | 1989-03-15 | 1990-09-20 | Janssen Pharmaceutica N.V. | [5(6)-(benzisoxa-, benzisothia- or indazol-3-yl)-1h-benzimidazol-2-yl] carbamates |
NZ232785A (en) * | 1989-03-15 | 1991-03-26 | Janssen Pharmaceutica Nv | 5-(1,2 benzisoxazol-, benzimidazol and benzisothiazol-3- yl)-1h-benzimadazol-2-yl carbamic acid ester derivatives preparatory processes, intermediates and anthelmintic compositions |
US5538989A (en) * | 1993-11-10 | 1996-07-23 | Hoechst-Roussel Agri-Vet Company | Fenbendazole formulations |
US5861142A (en) * | 1996-03-25 | 1999-01-19 | Schick; Mary Pichler | Method for promoting hair, nail, and skin keratinization |
GB9900752D0 (en) | 1999-01-15 | 1999-03-03 | Angiogene Pharm Ltd | Benzimidazole vascular damaging agents |
US7396819B2 (en) | 2003-08-08 | 2008-07-08 | Virbac Corporation | Anthelmintic formulations |
US7582612B2 (en) * | 2004-03-12 | 2009-09-01 | Hartz Mountain Corporation | Multi-action anthelmintic formulations |
US7893271B2 (en) * | 2005-07-28 | 2011-02-22 | Intervet International B.V. | Benzimidazole carbamates and (thio) carbamates, and the synthesis and use thereof |
EP2032046B1 (en) * | 2006-06-12 | 2015-11-04 | Smith & Nephew, Inc. | Systems and devices for tibial resection |
CA2660647C (en) | 2006-06-14 | 2015-07-28 | Intervet International B.V. | A suspension comprising benzimidazole carbamate and a polysorbate |
CN108884054B (zh) | 2015-11-30 | 2022-08-02 | 儿童医学中心公司 | 用于治疗增殖性疾病的化合物 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3480642A (en) * | 1967-03-22 | 1969-11-25 | Smithkline Corp | Process for producing 2-carbalkoxyaminobenzimidazoles |
DK131821C (da) * | 1967-03-22 | 1976-03-08 | Smith Kline French Lab | Analogifremgangsmade til fremstilling af en 2-karbalkoksyaminobenzimidazol |
FR2063815A5 (en) * | 1969-10-31 | 1971-07-09 | Aries Robert | Antifungal and anthelmintic benzimidazole carbamates |
-
0
- BE BE793358D patent/BE793358A/xx not_active IP Right Cessation
-
1971
- 1971-12-27 DE DE2164690A patent/DE2164690C3/de not_active Expired
-
1972
- 1972-12-19 RO RO7273205A patent/RO71503A/ro unknown
- 1972-12-20 ES ES409860A patent/ES409860A1/es not_active Expired
- 1972-12-20 CH CH827476A patent/CH583710A5/xx not_active IP Right Cessation
- 1972-12-20 HU HUHO1535A patent/HU165060B/hu unknown
- 1972-12-20 CS CS5893A patent/CS173650B2/cs unknown
- 1972-12-20 CS CS8805A patent/CS173615B2/cs unknown
- 1972-12-20 CH CH1856672A patent/CH580080A5/xx not_active IP Right Cessation
- 1972-12-21 DD DD167796A patent/DD109219A5/xx unknown
- 1972-12-21 DD DD178527*A patent/DD110760A5/xx unknown
- 1972-12-21 FI FI3637/72A patent/FI54299C/fi active
- 1972-12-22 AU AU50486/72A patent/AU465226B2/en not_active Expired
- 1972-12-22 CA CA159,777A patent/CA1017750A/en not_active Expired
- 1972-12-22 NO NO4753/72A patent/NO137092C/no unknown
- 1972-12-22 AT AT1099672A patent/AT320638B/de not_active IP Right Cessation
- 1972-12-22 IT IT33528/72A patent/IT1043888B/it active Protection Beyond IP Right Term
- 1972-12-22 DK DK642872AA patent/DK130293B/da unknown
- 1972-12-22 NL NL727217532A patent/NL153187B/xx not_active IP Right Cessation
- 1972-12-23 PL PL1972159809A patent/PL85192B1/pl unknown
- 1972-12-23 BG BG025960A patent/BG20591A3/xx unknown
- 1972-12-23 BG BG22217A patent/BG22080A3/xx unknown
- 1972-12-25 IL IL41170A patent/IL41170A/en unknown
- 1972-12-26 US US05/318,271 patent/US3954791A/en not_active Expired - Lifetime
- 1972-12-26 EG EG541/72A patent/EG11122A/xx active
- 1972-12-26 KR KR7201961A patent/KR780000116B1/ko active
- 1972-12-27 ZA ZA729076A patent/ZA729076B/xx unknown
- 1972-12-27 SU SU1865601A patent/SU492086A3/ru active
- 1972-12-27 JP JP734324A patent/JPS5033067B2/ja not_active Expired
- 1972-12-27 GB GB5966672A patent/GB1360180A/en not_active Expired
- 1972-12-27 SE SE7216998A patent/SE395890B/xx unknown
- 1972-12-27 FR FR7246316A patent/FR2166048B1/fr not_active Expired
-
1973
- 1973-11-11 SU SU1967977A patent/SU493967A3/ru active
-
1976
- 1976-03-22 KE KE2613*UA patent/KE2613A/xx unknown
- 1976-12-30 MY MY92/76A patent/MY7600092A/xx unknown
Also Published As
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