IL274234B2 - Compositions and methods for the treatment of eye disorders - Google Patents

Compositions and methods for the treatment of eye disorders

Info

Publication number
IL274234B2
IL274234B2 IL274234A IL27423420A IL274234B2 IL 274234 B2 IL274234 B2 IL 274234B2 IL 274234 A IL274234 A IL 274234A IL 27423420 A IL27423420 A IL 27423420A IL 274234 B2 IL274234 B2 IL 274234B2
Authority
IL
Israel
Prior art keywords
pharmaceutical composition
compound
composition
pilocarpine
treating
Prior art date
Application number
IL274234A
Other languages
English (en)
Hebrew (he)
Other versions
IL274234A (en
IL274234B (en
Inventor
Mahesh Kandula
Original Assignee
Cellix Bio Private Ltd
Mahesh Kandula
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Cellix Bio Private Ltd, Mahesh Kandula filed Critical Cellix Bio Private Ltd
Publication of IL274234A publication Critical patent/IL274234A/en
Publication of IL274234B publication Critical patent/IL274234B/en
Publication of IL274234B2 publication Critical patent/IL274234B2/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/38—Heterocyclic compounds having sulfur as a ring hetero atom
    • A61K31/385—Heterocyclic compounds having sulfur as a ring hetero atom having two or more sulfur atoms in the same ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4178—1,3-Diazoles not condensed 1,3-diazoles and containing further heterocyclic rings, e.g. pilocarpine, nitrofurantoin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0048—Eye, e.g. artificial tears
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00—Drugs for disorders of the senses
    • A61P27/02—Ophthalmic agents
    • A61P27/06—Antiglaucoma agents or miotics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00—Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Steroid Compounds (AREA)
IL274234A 2017-11-17 2020-04-26 Compositions and methods for the treatment of eye disorders IL274234B2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IN201741041231 2017-11-17
PCT/IB2018/057342 WO2019097318A1 (en) 2017-11-17 2018-09-22 Compositions and methods for the treatment of eye disorders

Publications (3)

Publication Number Publication Date
IL274234A IL274234A (en) 2020-06-30
IL274234B IL274234B (en) 2022-10-01
IL274234B2 true IL274234B2 (en) 2023-02-01

Family

ID=66540065

Family Applications (1)

Application Number Title Priority Date Filing Date
IL274234A IL274234B2 (en) 2017-11-17 2020-04-26 Compositions and methods for the treatment of eye disorders

Country Status (14)

Country Link
US (1) US10933052B2 (https=)
EP (1) EP3651747A4 (https=)
JP (1) JP7006990B2 (https=)
KR (1) KR102349776B1 (https=)
CN (1) CN111372576A (https=)
AU (1) AU2018367909B2 (https=)
BR (1) BR112020009361A2 (https=)
CA (1) CA3081553C (https=)
IL (1) IL274234B2 (https=)
MX (1) MX389626B (https=)
RU (1) RU2761436C1 (https=)
SG (1) SG11202004019SA (https=)
WO (1) WO2019097318A1 (https=)
ZA (1) ZA202002066B (https=)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3522873B1 (en) * 2016-10-04 2022-03-16 Cellix Bio Private Limited Compositions and methods for the treatment of xerostomia
IL274233B2 (en) * 2017-11-17 2024-04-01 Cellix Bio Private Ltd Compounds, compositions and methods for treatment of eye disorders and skin diseases
BR112020015436A2 (pt) * 2018-02-05 2020-12-22 Cellix Bio Private Limited Composição farmacêutica, mistura física e uso de uma composição
MX2022006803A (es) * 2019-12-04 2022-09-19 Restore Vision Llc Formulaciones oftalmicas para el tratamiento de la presbicia.
US11400039B2 (en) * 2020-01-16 2022-08-02 James W. Hill Changing eye color by gene transduction
IL298476A (en) * 2020-05-26 2023-01-01 Cellix Bio Private Ltd Pharmaceutical formulations of pilocarpine r-(+)-lipoate
WO2023052974A1 (en) * 2021-09-29 2023-04-06 Avaca Pharma Private Limited Ocular compositions and methods for the treatment of ophthalmic diseases and disorders
WO2024108202A2 (en) * 2022-11-19 2024-05-23 Iview Therapeutics, Inc. Compounds, compositions and methods for treatment of age-related ocular disorders
WO2025230326A1 (ko) * 2024-04-30 2025-11-06 주식회사태준제약 필로카르핀을 포함하는 점안 조성물

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Also Published As

Publication number Publication date
KR102349776B1 (ko) 2022-01-10
MX2020004666A (es) 2022-01-26
CA3081553A1 (en) 2019-05-23
IL274234A (en) 2020-06-30
RU2761436C1 (ru) 2021-12-08
JP7006990B2 (ja) 2022-02-10
MX389626B (es) 2025-03-20
WO2019097318A1 (en) 2019-05-23
ZA202002066B (en) 2021-07-28
IL274234B (en) 2022-10-01
EP3651747A1 (en) 2020-05-20
SG11202004019SA (en) 2020-05-28
CA3081553C (en) 2022-11-15
NZ763688A (en) 2021-10-29
AU2018367909B2 (en) 2022-03-10
EP3651747A4 (en) 2020-07-22
CN111372576A (zh) 2020-07-03
KR20200089292A (ko) 2020-07-24
AU2018367909A1 (en) 2020-05-07
BR112020009361A2 (pt) 2020-10-13
JP2021503449A (ja) 2021-02-12
US10933052B2 (en) 2021-03-02
US20200179343A1 (en) 2020-06-11

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