IL217954A - Derivatives of 5-fluoro-2-oxopyrimidine-1 (2 h) - carboxylate - Google Patents

Derivatives of 5-fluoro-2-oxopyrimidine-1 (2 h) - carboxylate

Info

Publication number
IL217954A
IL217954A IL217954A IL21795412A IL217954A IL 217954 A IL217954 A IL 217954A IL 217954 A IL217954 A IL 217954A IL 21795412 A IL21795412 A IL 21795412A IL 217954 A IL217954 A IL 217954A
Authority
IL
Israel
Prior art keywords
oxopyrimidine
fluoro
carboxylate derivatives
carboxylate
derivatives
Prior art date
Application number
IL217954A
Other languages
English (en)
Hebrew (he)
Other versions
IL217954A0 (en
Inventor
Bryan Kristy
A Boebel Timothy
Lorsbach Beth
p martin Timothy
john owen W
Pobanz Mark
Thornburgh Scott
D Webster Jeffery
Yao Chenglin
Original Assignee
Dow Agrosciences Llc
Bryan Kristy
A Boebel Timothy
Lorsbach Beth
p martin Timothy
john owen W
Pobanz Mark
Thornburgh Scott
D Webster Jeffery
Yao Chenglin
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535293&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL217954(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Dow Agrosciences Llc, Bryan Kristy, A Boebel Timothy, Lorsbach Beth, p martin Timothy, john owen W, Pobanz Mark, Thornburgh Scott, D Webster Jeffery, Yao Chenglin filed Critical Dow Agrosciences Llc
Publication of IL217954A0 publication Critical patent/IL217954A0/en
Publication of IL217954A publication Critical patent/IL217954A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/16—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof the nitrogen atom being part of a heterocyclic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/20—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D239/22—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms directly attached to ring carbon atoms

Landscapes

  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Environmental Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL217954A 2009-08-07 2012-02-05 Derivatives of 5-fluoro-2-oxopyrimidine-1 (2 h) - carboxylate IL217954A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US23223209P 2009-08-07 2009-08-07
PCT/US2010/044585 WO2011017544A1 (en) 2009-08-07 2010-08-05 5-fluoro-2-oxopyrimidine- 1(2h)-carboxylate derivatives

Publications (2)

Publication Number Publication Date
IL217954A0 IL217954A0 (en) 2012-03-29
IL217954A true IL217954A (en) 2016-02-29

Family

ID=43535293

Family Applications (1)

Application Number Title Priority Date Filing Date
IL217954A IL217954A (en) 2009-08-07 2012-02-05 Derivatives of 5-fluoro-2-oxopyrimidine-1 (2 h) - carboxylate

Country Status (28)

Country Link
US (1) US8318758B2 (enExample)
EP (1) EP2462133B1 (enExample)
JP (1) JP5818791B2 (enExample)
KR (1) KR101792286B1 (enExample)
CN (1) CN102548979B (enExample)
AU (1) AU2010279408B2 (enExample)
BR (1) BR112012002807B1 (enExample)
CA (1) CA2769251C (enExample)
CL (1) CL2012000314A1 (enExample)
CO (1) CO6491089A2 (enExample)
CR (1) CR20120033A (enExample)
DK (1) DK2462133T3 (enExample)
EA (1) EA022930B1 (enExample)
EC (1) ECSP12011651A (enExample)
ES (1) ES2506169T3 (enExample)
HN (1) HN2012000261A (enExample)
IL (1) IL217954A (enExample)
IN (1) IN2012DN00695A (enExample)
MX (1) MX2012001623A (enExample)
NI (1) NI201200019A (enExample)
NZ (1) NZ597638A (enExample)
PE (1) PE20120689A1 (enExample)
PL (1) PL2462133T3 (enExample)
PT (1) PT2462133E (enExample)
RS (1) RS53658B1 (enExample)
UA (1) UA106086C2 (enExample)
WO (1) WO2011017544A1 (enExample)
ZA (1) ZA201305992B (enExample)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2010279411B2 (en) * 2009-08-07 2014-10-23 Adama Makhteshim Ltd. N1-sulfonyl-5-fluoropyrimidinone derivatives
HUE047711T2 (hu) 2012-12-28 2020-05-28 Adama Makhteshim Ltd N-(szubsztituált)-5-fluor-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2H)-karboxilát származékok
UA117123C2 (uk) * 2012-12-28 2018-06-25 Адама Махтешім Лтд. Похідні 1-(заміщений бензоїл)-5-фтор-4-іміно-3-метил-3,4-дигідропіримідин-2(1h)-ону
RU2015131149A (ru) 2012-12-28 2017-02-03 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи N-(замещенные)-5-фтор-4-имино-3-метил-2-оксо-3,4-дигидропиримидин-1(2н)-карбоксамидные производные
CA2894553C (en) 2012-12-31 2021-03-02 Dow Agrosciences Llc 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
EP3097096A4 (en) 2013-12-31 2017-10-11 Adama Makhteshim Ltd. 5-fluoro-4-imino-3-(alkyl/substituted alkyl)-1- (arylsulfonyl)-3,4-dihydropyrimidin-2(1h)-one and processes for their preparation
EA030030B1 (ru) 2013-12-31 2018-06-29 Адама Мактешим Лтд. Синергетические фунгицидные смеси и синергетические фунгицидные композиции для борьбы с грибами
WO2016040193A1 (en) 2014-09-08 2016-03-17 Samumed, Llc 3-(1h-imidazo[4,5-c]pyridin-2-yl)-1h-pyrazolo[3,4-b]pyridine and therapeutic uses thereof
WO2017079759A1 (en) 2015-11-06 2017-05-11 Samumed, Llc 2-(1h-indazol-3-yl)-3h-imidazo[4,5-c]pyridines and their anti-inflammatory uses thereof
MY199242A (en) 2016-06-01 2023-10-22 Samumed Llc Process for preparing n-(5-(3-(7-(3-fluorophenyl)-3h-imidazo[4,5-c]pyridin-2-yl)-1h-indazol-5-yl)pyridin-3-yl)-3-methylbutanamide
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
CR20210270A (es) 2018-11-05 2021-07-20 Adama Makhteshim Ltd Mezclas y composiciones que comprenden 5-fluoro-4-imino-3-metil-1-tosil-3,4-dihidropirimidin-2-ona, y métodos de uso de los mismos
TWI808347B (zh) 2019-09-23 2023-07-11 以色列商亞當馬赫特希姆有限公司 用於製備5-氟-4-亞胺基-3-甲基-1-甲苯磺醯基-3,4-二氫嘧啶-2(1h)-酮及該化合物的衍生物之方法
MX2022011088A (es) 2020-03-09 2022-09-29 Adama Makhteshim Ltd Procedimiento para preparar 5-fluoro-4-imino-3-metil-1-(tolueno-4- sulfonil)-3,4-dihidro-1h-pirimidin-2-ona.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
IL125589A0 (en) 1996-03-11 1999-03-12 Novartis Ag Pyrimidin-4-one derivatives as pesticides
WO2004037159A2 (en) * 2002-10-23 2004-05-06 Obetherapy Biotechnology Compounds, compositions and methods for modulating fat metabolism
DK2151439T3 (en) * 2007-04-27 2014-03-10 Daiichi Sankyo Co Ltd Nitrogenated AROMATIC 6-membered RINGDERIVAT, AND THIS pharmaceutical composition comprising
WO2010047866A2 (en) 2008-08-01 2010-04-29 Dow Agrosciences Llc Use of 5-fluorocytosine as a fungicide

Also Published As

Publication number Publication date
ES2506169T3 (es) 2014-10-13
WO2011017544A1 (en) 2011-02-10
ECSP12011651A (es) 2012-03-30
JP5818791B2 (ja) 2015-11-18
DK2462133T3 (en) 2015-01-05
BR112012002807A8 (pt) 2017-07-11
US8318758B2 (en) 2012-11-27
JP2013501726A (ja) 2013-01-17
IN2012DN00695A (enExample) 2015-06-19
EA201270255A1 (ru) 2012-07-30
NZ597638A (en) 2014-06-27
CO6491089A2 (es) 2012-07-31
CL2012000314A1 (es) 2012-10-05
BR112012002807A2 (pt) 2015-10-13
CA2769251A1 (en) 2011-02-10
PT2462133E (pt) 2014-12-26
EA022930B1 (ru) 2016-03-31
AU2010279408B2 (en) 2015-09-10
CN102548979B (zh) 2015-05-13
HN2012000261A (es) 2015-01-05
EP2462133A1 (en) 2012-06-13
MX2012001623A (es) 2012-04-11
PL2462133T3 (pl) 2015-03-31
ZA201305992B (en) 2014-10-29
CA2769251C (en) 2018-05-15
HK1172892A1 (en) 2013-05-03
RS53658B1 (sr) 2015-04-30
US20110034491A1 (en) 2011-02-10
PE20120689A1 (es) 2012-06-06
CR20120033A (es) 2012-03-22
BR112012002807B1 (pt) 2018-07-10
EP2462133A4 (en) 2013-01-16
CN102548979A (zh) 2012-07-04
EP2462133B1 (en) 2014-09-24
KR101792286B1 (ko) 2017-10-31
UA106086C2 (uk) 2014-07-25
AU2010279408A1 (en) 2012-02-09
IL217954A0 (en) 2012-03-29
NI201200019A (es) 2012-05-22
KR20120043069A (ko) 2012-05-03

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