IL202822A0 - A regioselective metal catalyzed synthesis of annelated benzimidazoles and azabenzimidazoles - Google Patents

A regioselective metal catalyzed synthesis of annelated benzimidazoles and azabenzimidazoles

Info

Publication number
IL202822A0
IL202822A0 IL202822A IL20282209A IL202822A0 IL 202822 A0 IL202822 A0 IL 202822A0 IL 202822 A IL202822 A IL 202822A IL 20282209 A IL20282209 A IL 20282209A IL 202822 A0 IL202822 A0 IL 202822A0
Authority
IL
Israel
Prior art keywords
azabenzimidazoles
benzimidazoles
annelated
regioselective
metal catalyzed
Prior art date
Application number
IL202822A
Other languages
English (en)
Original Assignee
Sanofi Aventis
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi Aventis filed Critical Sanofi Aventis
Publication of IL202822A0 publication Critical patent/IL202822A0/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
    • C07D491/14—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Measuring Oxygen Concentration In Cells (AREA)
  • Plural Heterocyclic Compounds (AREA)
IL202822A 2007-06-26 2009-12-17 A regioselective metal catalyzed synthesis of annelated benzimidazoles and azabenzimidazoles IL202822A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP07290801 2007-06-26
PCT/EP2008/004638 WO2009000412A1 (en) 2007-06-26 2008-06-11 A regioselective metal catalyzed synthesis of annelated benzimidazoles and azabenzimidazoles

Publications (1)

Publication Number Publication Date
IL202822A0 true IL202822A0 (en) 2010-06-30

Family

ID=39720505

Family Applications (1)

Application Number Title Priority Date Filing Date
IL202822A IL202822A0 (en) 2007-06-26 2009-12-17 A regioselective metal catalyzed synthesis of annelated benzimidazoles and azabenzimidazoles

Country Status (11)

Country Link
US (1) US20100216988A1 (enExample)
EP (1) EP2173747B1 (enExample)
JP (1) JP5492769B2 (enExample)
KR (1) KR20100033484A (enExample)
CN (1) CN101687865A (enExample)
AT (1) ATE538120T1 (enExample)
AU (1) AU2008267443A1 (enExample)
BR (1) BRPI0813273A2 (enExample)
CA (1) CA2693142A1 (enExample)
IL (1) IL202822A0 (enExample)
WO (1) WO2009000412A1 (enExample)

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Also Published As

Publication number Publication date
BRPI0813273A2 (pt) 2014-12-30
JP5492769B2 (ja) 2014-05-14
CA2693142A1 (en) 2008-12-31
WO2009000412A1 (en) 2008-12-31
KR20100033484A (ko) 2010-03-30
EP2173747A1 (en) 2010-04-14
EP2173747B1 (en) 2011-12-21
ATE538120T1 (de) 2012-01-15
US20100216988A1 (en) 2010-08-26
AU2008267443A1 (en) 2008-12-31
JP2010531312A (ja) 2010-09-24
CN101687865A (zh) 2010-03-31

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