IL164781A0 - Process for preparing highly functionalized y-butyrolactams and y-amino acids - Google Patents
Process for preparing highly functionalized y-butyrolactams and y-amino acidsInfo
- Publication number
- IL164781A0 IL164781A0 IL16478104A IL16478104A IL164781A0 IL 164781 A0 IL164781 A0 IL 164781A0 IL 16478104 A IL16478104 A IL 16478104A IL 16478104 A IL16478104 A IL 16478104A IL 164781 A0 IL164781 A0 IL 164781A0
- Authority
- IL
- Israel
- Prior art keywords
- butyrolactams
- amino acids
- preparing highly
- highly functionalized
- functionalized
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/04—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
- C07C229/06—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton
- C07C229/08—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to hydrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/22—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton from lactams, cyclic ketones or cyclic oximes, e.g. by reactions involving Beckmann rearrangement
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C229/00—Compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C229/02—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton
- C07C229/04—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated
- C07C229/06—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton
- C07C229/18—Compounds containing amino and carboxyl groups bound to the same carbon skeleton having amino and carboxyl groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being acyclic and saturated having only one amino and one carboxyl group bound to the carbon skeleton the nitrogen atom of the amino group being further bound to carbon atoms of six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
- C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/36—Oxygen or sulfur atoms
- C07D207/38—2-Pyrrolones
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Peptides Or Proteins (AREA)
- Pyrrole Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US37699102P | 2002-04-30 | 2002-04-30 | |
PCT/IB2003/001646 WO2003093220A1 (en) | 2002-04-30 | 2003-04-17 | Process for preparing highly functionalized y-butyrolactams and y-amino acids |
Publications (1)
Publication Number | Publication Date |
---|---|
IL164781A0 true IL164781A0 (en) | 2005-12-18 |
Family
ID=29401429
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL16478104A IL164781A0 (en) | 2002-04-30 | 2004-10-21 | Process for preparing highly functionalized y-butyrolactams and y-amino acids |
Country Status (15)
Country | Link |
---|---|
US (2) | US20030225149A1 (pt) |
EP (1) | EP1499583A1 (pt) |
JP (1) | JP2005523932A (pt) |
KR (1) | KR20040106415A (pt) |
CN (1) | CN1649827A (pt) |
AR (1) | AR039467A1 (pt) |
AU (1) | AU2003219425A1 (pt) |
BR (1) | BR0309743A (pt) |
CA (1) | CA2483830A1 (pt) |
IL (1) | IL164781A0 (pt) |
MX (1) | MXPA04010771A (pt) |
PL (1) | PL373296A1 (pt) |
RU (1) | RU2004131840A (pt) |
TW (1) | TW200400929A (pt) |
WO (1) | WO2003093220A1 (pt) |
Families Citing this family (29)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL126999A (en) | 1996-07-24 | 2002-03-10 | Warner Lambert Co | Pharmaceutical preparations containing isobutylgaba and its history for use in the treatment of pain |
ATE455093T1 (de) * | 2004-06-21 | 2010-01-15 | Warner Lambert Co | Herstellung von pregabalin und verwandten verbindungen |
PL1773902T3 (pl) | 2004-08-04 | 2018-05-30 | Foam Supplies, Inc. | Odchylenie reaktywności i rozkład katalizatora w piance poliuretanowej |
WO2006108151A1 (en) * | 2005-04-06 | 2006-10-12 | Teva Pharmaceutical Industries Ltd. | Crystalline forms of pregabalin |
US7488846B2 (en) * | 2005-04-11 | 2009-02-10 | Teva Pharmaceuical Industries Ltd. | Pregabalin free of lactam and a process for preparation thereof |
EP1768950A2 (en) * | 2005-04-11 | 2007-04-04 | Teva Pharmaceutical Industries Ltd. | Process for making (s)-pregabalin |
ATE486841T1 (de) * | 2005-05-10 | 2010-11-15 | Teva Pharma | Verfahren zur herstellung von pregabalin und salzen daraus |
KR20070118305A (ko) * | 2005-05-10 | 2007-12-14 | 테바 파마슈티컬 인더스트리즈 리미티드 | 3-카르바모일메틸-5-메틸 헥산산의 광학 분할 |
MX2007000525A (es) * | 2005-05-10 | 2007-03-28 | Teva Pharma | Pregabalina libre de acido isobutilglutarico y un proceso para la preparacion de ella. |
CZ297970B6 (cs) * | 2005-08-10 | 2007-05-09 | Zentiva, A. S | Zpusob výroby (S)-3-(aminomethyl)-5-methyl-hexanové kyseliny (pregabalinu) |
KR20080034205A (ko) * | 2005-09-19 | 2008-04-18 | 테바 파마슈티컬 인더스트리즈 리미티드 | (s)-프레가발린의 신규한 합성을 위한 주요 중간체인 키랄3-카르바모일메틸-5-메틸 헥산산 |
CA2646474A1 (en) * | 2006-04-24 | 2007-11-08 | Teva Pharmaceutical Industries Ltd. | Processes for the synthesis of 3-isobutylglutaric acid |
WO2007139933A2 (en) * | 2006-05-24 | 2007-12-06 | Teva Pharmaceutical Industries Ltd. | Processes for the preparation of r-(+)-3-(carbamoyl methyl)-5-methylhexanoic acid and salts thereof |
KR20080036060A (ko) * | 2006-05-31 | 2008-04-24 | 테바 파마슈티컬 인더스트리즈 리미티드 | 프레가발린의 중간체의 제조에 효소 분할을 이용하는 방법 |
EP1912931A2 (en) * | 2006-05-31 | 2008-04-23 | Teva Pharmaceutical Industries Ltd. | Preparation of (s)-pregabalin-nitrile |
TW200846308A (en) * | 2007-03-22 | 2008-12-01 | Teva Pharma | Synthesis of (s)-(+)-3-(aminomethyl)-5-methyl hexanoic acid |
WO2008127646A2 (en) * | 2007-04-11 | 2008-10-23 | Dsm Ip Assets B.V. | Transaminase-based processes for preparation of pregabalin |
ES2551552T3 (es) * | 2007-06-05 | 2015-11-19 | Akzo Nobel Coatings International B.V. | Composición de revestimiento curable por radiación derivada de aceites vegetales epoxidados |
KR20090101462A (ko) * | 2007-10-03 | 2009-09-28 | 테바 파마슈티컬 인더스트리즈 리미티드 | 프레가발린-4-엘리미네이트, 프레가발린 5-엘리미네이트, 기준 마커 및 표준물로서의 이들의 용도, 및 이들을 낮은 수준으로 함유하는 프레가발린의 제조 방법 |
JP2011507941A (ja) * | 2007-12-26 | 2011-03-10 | ジェネリクス・(ユーケー)・リミテッド | プレガバリンの製造方法 |
JP2010043063A (ja) | 2008-05-09 | 2010-02-25 | Agency For Science Technology & Research | 川崎病の診断及び治療 |
WO2009158343A1 (en) * | 2008-06-23 | 2009-12-30 | Teva Pharmaceutical Industries, Ltd. | Stereoselective enzymatic synthesis of (s) or (r)-iso-butyl-glutaric ester |
WO2010100122A1 (en) | 2009-03-05 | 2010-09-10 | Akzo Nobel Coatings International B.V. | Hydroxyl functional oil polyols and coating compositions prepared from hydroxyl functional oil polyols |
WO2011086565A1 (en) * | 2010-01-15 | 2011-07-21 | Lupin Limited | Method for preparation of enantiomerically enriched and/or racemic gamma-amino acids |
MX2013007459A (es) | 2010-12-28 | 2013-07-29 | Akzo Nobel Coatings Int Bv | Composiciones de recubrimiento curable por radiacion para metal. |
GB201121317D0 (en) | 2011-12-09 | 2012-01-25 | Syngenta Ltd | Herbicidal compounds |
BR112014014107B1 (pt) | 2011-12-21 | 2020-12-08 | Akzo Nobel Coatings International B.V | método de preparação de uma composição de revestimento e substrato revestido |
EP2794704B1 (en) | 2011-12-21 | 2017-04-05 | Akzo Nobel Coatings International B.V. | Water-based coating compositions |
WO2014155291A1 (en) * | 2013-03-27 | 2014-10-02 | Pfizer Ireland Pharmaceuticals | Process and intermediates for the preparation of pregabalin |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3935210A (en) | 1971-07-29 | 1976-01-27 | Sandoz, Inc. | Preparation of 1-aryl-4,5-dihalo-pyridazone-6 |
SK283281B6 (sk) * | 1992-05-20 | 2003-05-02 | Northwestern University | Deriváty gamaaminomaslovej kyseliny, spôsoby a medziprodukty na ich výrobu, ich použitie a farmaceutické prostriedky |
DZ2770A1 (fr) | 1998-04-17 | 2003-12-01 | Lilly Co Eli | Procédé de préparation de 1h-indol-3 glyoxamides substituées en position 4. |
US6306910B1 (en) | 1998-07-09 | 2001-10-23 | Warner-Lambert Company | Use of Gaba-analogues for treating insomnia |
TR200103587T2 (tr) * | 1999-06-10 | 2002-04-22 | Warner Lambert Company | Mono-ve çift ikame edilmiş 3-propil gama aminobutirik asitler. |
-
2003
- 2003-02-13 US US10/365,430 patent/US20030225149A1/en not_active Abandoned
- 2003-04-17 CA CA002483830A patent/CA2483830A1/en not_active Abandoned
- 2003-04-17 WO PCT/IB2003/001646 patent/WO2003093220A1/en not_active Application Discontinuation
- 2003-04-17 RU RU2004131840/04A patent/RU2004131840A/ru not_active Application Discontinuation
- 2003-04-17 KR KR10-2004-7017412A patent/KR20040106415A/ko not_active Application Discontinuation
- 2003-04-17 EP EP03715236A patent/EP1499583A1/en not_active Withdrawn
- 2003-04-17 CN CNA038096412A patent/CN1649827A/zh active Pending
- 2003-04-17 PL PL03373296A patent/PL373296A1/xx not_active Application Discontinuation
- 2003-04-17 AU AU2003219425A patent/AU2003219425A1/en not_active Abandoned
- 2003-04-17 BR BR0309743-9A patent/BR0309743A/pt not_active IP Right Cessation
- 2003-04-17 MX MXPA04010771A patent/MXPA04010771A/es not_active Application Discontinuation
- 2003-04-17 JP JP2004501360A patent/JP2005523932A/ja not_active Withdrawn
- 2003-04-23 US US10/421,350 patent/US6924377B2/en not_active Expired - Fee Related
- 2003-04-28 AR ARP030101461A patent/AR039467A1/es unknown
- 2003-04-29 TW TW092110024A patent/TW200400929A/zh unknown
-
2004
- 2004-10-21 IL IL16478104A patent/IL164781A0/xx unknown
Also Published As
Publication number | Publication date |
---|---|
AR039467A1 (es) | 2005-02-23 |
BR0309743A (pt) | 2005-02-09 |
RU2004131840A (ru) | 2005-05-27 |
JP2005523932A (ja) | 2005-08-11 |
US6924377B2 (en) | 2005-08-02 |
MXPA04010771A (es) | 2005-03-07 |
AU2003219425A1 (en) | 2003-11-17 |
US20030236415A1 (en) | 2003-12-25 |
WO2003093220A1 (en) | 2003-11-13 |
PL373296A1 (en) | 2005-08-22 |
EP1499583A1 (en) | 2005-01-26 |
KR20040106415A (ko) | 2004-12-17 |
CA2483830A1 (en) | 2003-11-13 |
US20030225149A1 (en) | 2003-12-04 |
TW200400929A (en) | 2004-01-16 |
CN1649827A (zh) | 2005-08-03 |
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