IL163769A0 - Quinoline derivatives - Google Patents

Quinoline derivatives

Info

Publication number
IL163769A0
IL163769A0 IL16376903A IL16376903A IL163769A0 IL 163769 A0 IL163769 A0 IL 163769A0 IL 16376903 A IL16376903 A IL 16376903A IL 16376903 A IL16376903 A IL 16376903A IL 163769 A0 IL163769 A0 IL 163769A0
Authority
IL
Israel
Prior art keywords
quinoline derivatives
quinoline
derivatives
Prior art date
Application number
IL16376903A
Other languages
English (en)
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of IL163769A0 publication Critical patent/IL163769A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/10Ophthalmic agents for accommodation disorders, e.g. myopia
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Ophthalmology & Optometry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
IL16376903A 2002-03-07 2003-03-06 Quinoline derivatives IL163769A0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP02005115 2002-03-07
EP02005117 2002-03-07
PCT/EP2003/002321 WO2003074511A1 (en) 2002-03-07 2003-03-06 Quinoline derivatives

Publications (1)

Publication Number Publication Date
IL163769A0 true IL163769A0 (en) 2005-12-18

Family

ID=27790094

Family Applications (1)

Application Number Title Priority Date Filing Date
IL16376903A IL163769A0 (en) 2002-03-07 2003-03-06 Quinoline derivatives

Country Status (28)

Country Link
US (2) US7399768B2 (enExample)
EP (1) EP1480970B1 (enExample)
JP (2) JP2005519117A (enExample)
KR (1) KR101027977B1 (enExample)
CN (2) CN1939915A (enExample)
AR (1) AR038730A1 (enExample)
AU (1) AU2003219023B2 (enExample)
BR (1) BR0308201A (enExample)
CA (2) CA2477720C (enExample)
CO (1) CO5611196A2 (enExample)
CY (1) CY1106409T1 (enExample)
DE (1) DE60311233T2 (enExample)
DK (1) DK1480970T3 (enExample)
EC (1) ECSP045271A (enExample)
EG (1) EG24415A (enExample)
ES (1) ES2279100T3 (enExample)
IL (1) IL163769A0 (enExample)
MX (1) MXPA04008666A (enExample)
MY (1) MY134325A (enExample)
NO (1) NO20044117L (enExample)
NZ (1) NZ534732A (enExample)
PE (1) PE20030927A1 (enExample)
PL (2) PL215012B1 (enExample)
PT (1) PT1480970E (enExample)
RU (1) RU2345991C2 (enExample)
SI (1) SI1480970T1 (enExample)
TW (1) TW200406401A (enExample)
WO (1) WO2003074511A1 (enExample)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
ATE438640T1 (de) * 2002-03-07 2009-08-15 Novartis Pharma Gmbh Chinolinderivate und ihre anwendung bei glaukom und kurzsichtigkeit
AR113908A1 (es) 2017-11-24 2020-06-24 H Lundbeck As Profármacos de catecolamina para uso en el tratamiento de la enfermedad de parkinson
US11168056B2 (en) 2019-05-20 2021-11-09 H. Lundbeck A/S Process for the manufacturing of (6aR,10aR)-7-propyl-6,6a,7,8,9,10,10a,11-octahydro-[1,3]dioxolo[4′,5′:5,6]benzo[1,2-G]quinoline and (4aR,10aR)-1-propyl-1,2,3,4,4a,5,10,10a-octahydro-benzo[G]quinoline-6,7-diol
US11111263B2 (en) 2019-05-20 2021-09-07 H. Lundbeck A/S Process for the manufacture of (2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-(((4aR,10aR)-7-hydroxy-1-propyl-1,2,3,4,4a,5,10,10a-octahydrobenzo[g]quinolin-6-yl)oxy)tetrahydro-2H-pyran-2-carboxylic acid
US11130775B2 (en) 2019-05-20 2021-09-28 H. Lundbeck A/S Solid forms of (2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-(((4aR,10aR)-7-hydroxy-1-propyl-1,2,3,4,4A,5,10,10A-octahydrobenzo[g]quinolin-6-yl)oxy)tetrahydro-2H-pyran-2-carboxylic acid
US11104697B2 (en) 2019-05-20 2021-08-31 H. Lundbeck A/S Process for the manufacture of (2S,3S,4S,5R,6S)-3,4,5-trihydroxy-6-(((4AR,10AR)-7-hydroxy-1- propyl-1,2,3,4,4A,5,10,10A-octahydrobenzo[g]quinolin-6-yl)oxy)tetrahydro-2H-pyran-2-carboxylic acid
JP7696829B2 (ja) 2019-05-21 2025-06-23 ハー・ルンドベック・アクチエゼルスカベット パーキンソン病の治療に使用するためのカテコールアミンカルバメートプロドラッグ
US12384765B2 (en) 2019-05-21 2025-08-12 H. Lundbeck A/S Catecholamine prodrugs for use in the treatment of Parkinson's Disease
WO2020234275A1 (en) 2019-05-21 2020-11-26 H. Lundbeck A/S New catecholamine prodrugs for use in the treatment of parkinson's diseases
WO2020234276A1 (en) 2019-05-21 2020-11-26 H. Lundbeck A/S New catecholamine prodrugs for use in the treatment of parkinson's disease

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL100555A (en) * 1991-02-07 2000-08-31 Hoechst Marion Roussel Inc N-substituted quinoline derivatives their preparation their use for the preparation of medicaments and the pharmaceutical compositions containing them
GB9326010D0 (en) * 1993-12-21 1994-02-23 Sandoz Ltd Improvements in or relating to organic compounds
TW378209B (en) * 1996-07-08 2000-01-01 Novartis Ag Benzo[g]quinoline derivatives, their preparation and the pharmaceutical composition containing them
PE20030240A1 (es) * 2001-07-09 2003-04-16 Novartis Ag DERIVADOS DE BENZO [g] QUINOLINA

Also Published As

Publication number Publication date
PL370915A1 (en) 2005-06-13
AR038730A1 (es) 2005-01-26
KR20040089615A (ko) 2004-10-21
CA2477720A1 (en) 2003-09-12
CN1293070C (zh) 2007-01-03
MXPA04008666A (es) 2004-12-06
SI1480970T1 (sl) 2007-06-30
PL215012B1 (pl) 2013-10-31
RU2345991C2 (ru) 2009-02-10
DE60311233T2 (de) 2007-11-15
EG24415A (en) 2009-05-25
JP2005519117A (ja) 2005-06-30
PL394208A1 (pl) 2011-08-16
ECSP045271A (es) 2004-10-26
JP2010095550A (ja) 2010-04-30
US20050234085A1 (en) 2005-10-20
ES2279100T3 (es) 2007-08-16
EP1480970A1 (en) 2004-12-01
CN1639148A (zh) 2005-07-13
CO5611196A2 (es) 2006-02-28
PL210336B1 (pl) 2012-01-31
BR0308201A (pt) 2005-01-04
AU2003219023A1 (en) 2003-09-16
HK1071364A1 (en) 2005-07-15
KR101027977B1 (ko) 2011-04-13
CA2477720C (en) 2010-09-21
US7399768B2 (en) 2008-07-15
CN1939915A (zh) 2007-04-04
TW200406401A (en) 2004-05-01
CA2706618A1 (en) 2003-09-12
NZ534732A (en) 2006-05-26
RU2004129767A (ru) 2005-06-27
PT1480970E (pt) 2007-03-30
WO2003074511A1 (en) 2003-09-12
NO20044117L (no) 2004-09-28
PE20030927A1 (es) 2003-12-26
MY134325A (en) 2007-12-31
DE60311233D1 (de) 2007-03-08
CY1106409T1 (el) 2011-10-12
AU2003219023B2 (en) 2006-11-30
DK1480970T3 (da) 2007-03-05
EP1480970B1 (en) 2007-01-17
US20080255176A1 (en) 2008-10-16

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