IL162699A0 - Combinations of peroxisome proliferator-activated receptor-alpha agonists and cyclooxygenase-2- selective inhibitors - Google Patents

Combinations of peroxisome proliferator-activated receptor-alpha agonists and cyclooxygenase-2- selective inhibitors

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Publication number
IL162699A0
IL162699A0 IL16269903A IL16269903A IL162699A0 IL 162699 A0 IL162699 A0 IL 162699A0 IL 16269903 A IL16269903 A IL 16269903A IL 16269903 A IL16269903 A IL 16269903A IL 162699 A0 IL162699 A0 IL 162699A0
Authority
IL
Israel
Prior art keywords
cyclooxygenase
combinations
activated receptor
selective inhibitors
peroxisome proliferator
Prior art date
Application number
IL16269903A
Other languages
English (en)
Original Assignee
Pharmacia Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pharmacia Corp filed Critical Pharmacia Corp
Publication of IL162699A0 publication Critical patent/IL162699A0/xx

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    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42Oxazoles
    • A61K31/4211,3-Oxazoles, e.g. pemoline, trimethadione
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    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
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    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/192Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid 
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    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/20Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
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    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/20Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
    • A61K31/202Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids having three or more double bonds, e.g. linolenic
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    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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IL16269903A 2002-01-14 2003-01-14 Combinations of peroxisome proliferator-activated receptor-alpha agonists and cyclooxygenase-2- selective inhibitors IL162699A0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US34829702P 2002-01-14 2002-01-14
US10/341,217 US20030212138A1 (en) 2002-01-14 2003-01-13 Combinations of peroxisome proliferator-activated receptor-alpha agonists and cyclooxygenase-2 selective inhibitors and therapeutic uses therefor
PCT/US2003/000956 WO2003059294A2 (en) 2002-01-14 2003-01-14 Combinations of peroxisome proliferator-activated receptor-alpha agonists and cyclooxygenase-2 selective inhibitors and therapeutic uses therefor

Publications (1)

Publication Number Publication Date
IL162699A0 true IL162699A0 (en) 2005-11-20

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IL16269903A IL162699A0 (en) 2002-01-14 2003-01-14 Combinations of peroxisome proliferator-activated receptor-alpha agonists and cyclooxygenase-2- selective inhibitors

Country Status (10)

Country Link
US (1) US20030212138A1 (xx)
EP (1) EP1569640A4 (xx)
JP (1) JP2005525313A (xx)
KR (1) KR20040095207A (xx)
AU (1) AU2003207535A1 (xx)
CA (1) CA2472168A1 (xx)
IL (1) IL162699A0 (xx)
MX (1) MXPA04006796A (xx)
PL (1) PL374962A1 (xx)
WO (1) WO2003059294A2 (xx)

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WO2006118821A2 (en) * 2005-05-02 2006-11-09 The Regents Of The University Of Colorado Systems and methods for treating human inflammatory and proliferative diseases, with a combination of compounds, or a bifunctional compound,that provides fatty acid metabolism and glycolysis inhibition
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FR2999936B1 (fr) * 2012-12-21 2015-01-16 Urgo Lab Utilisation d'acide acetylsalicylique pour la prevention et/ou le traitement des plaies du diabetique
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JP2005525313A (ja) 2005-08-25
WO2003059294A3 (en) 2005-07-14
EP1569640A4 (en) 2006-06-21
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US20030212138A1 (en) 2003-11-13
PL374962A1 (en) 2005-11-14

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