IL162699A0 - Combinations of peroxisome proliferator-activated receptor-alpha agonists and cyclooxygenase-2- selective inhibitors - Google Patents
Combinations of peroxisome proliferator-activated receptor-alpha agonists and cyclooxygenase-2- selective inhibitorsInfo
- Publication number
- IL162699A0 IL162699A0 IL16269903A IL16269903A IL162699A0 IL 162699 A0 IL162699 A0 IL 162699A0 IL 16269903 A IL16269903 A IL 16269903A IL 16269903 A IL16269903 A IL 16269903A IL 162699 A0 IL162699 A0 IL 162699A0
- Authority
- IL
- Israel
- Prior art keywords
- cyclooxygenase
- combinations
- activated receptor
- selective inhibitors
- peroxisome proliferator
- Prior art date
Links
- 229940127520 Peroxisome Proliferator-activated Receptor alpha Agonists Drugs 0.000 title 1
- 229940124639 Selective inhibitor Drugs 0.000 title 1
Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
- A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/42—Oxazoles
- A61K31/421—1,3-Oxazoles, e.g. pemoline, trimethadione
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- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
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- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/192—Carboxylic acids, e.g. valproic acid having aromatic groups, e.g. sulindac, 2-aryl-propionic acids, ethacrynic acid
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- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/20—Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
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- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/20—Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids
- A61K31/202—Carboxylic acids, e.g. valproic acid having a carboxyl group bound to a chain of seven or more carbon atoms, e.g. stearic, palmitic, arachidic acids having three or more double bonds, e.g. linolenic
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
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- A61K31/425—Thiazoles
- A61K31/426—1,3-Thiazoles
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- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
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- A61K31/568—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone
- A61K31/5685—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol substituted in positions 10 and 13 by a chain having at least one carbon atom, e.g. androstanes, e.g. testosterone having an oxo group in position 17, e.g. androsterone
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Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US34829702P | 2002-01-14 | 2002-01-14 | |
US10/341,217 US20030212138A1 (en) | 2002-01-14 | 2003-01-13 | Combinations of peroxisome proliferator-activated receptor-alpha agonists and cyclooxygenase-2 selective inhibitors and therapeutic uses therefor |
PCT/US2003/000956 WO2003059294A2 (fr) | 2002-01-14 | 2003-01-14 | Combinaisons d'agonistes du recepteur alpha activateur de la proliferation des peroxisomes et d'inhibiteurs selectifs de la cyclooxygenase-2 et leurs utilisations therapeutiques |
Publications (1)
Publication Number | Publication Date |
---|---|
IL162699A0 true IL162699A0 (en) | 2005-11-20 |
Family
ID=26992419
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL16269903A IL162699A0 (en) | 2002-01-14 | 2003-01-14 | Combinations of peroxisome proliferator-activated receptor-alpha agonists and cyclooxygenase-2- selective inhibitors |
Country Status (10)
Country | Link |
---|---|
US (1) | US20030212138A1 (fr) |
EP (1) | EP1569640A4 (fr) |
JP (1) | JP2005525313A (fr) |
KR (1) | KR20040095207A (fr) |
AU (1) | AU2003207535A1 (fr) |
CA (1) | CA2472168A1 (fr) |
IL (1) | IL162699A0 (fr) |
MX (1) | MXPA04006796A (fr) |
PL (1) | PL374962A1 (fr) |
WO (1) | WO2003059294A2 (fr) |
Families Citing this family (27)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20040152752A1 (en) * | 2002-05-30 | 2004-08-05 | Chong Kong Teck | Treatment for human papillomavirus |
EP2295529B2 (fr) | 2002-07-11 | 2022-05-18 | Basf As | Procédé de diminution des polluants environnementaux dans une huile ou une graisse et produit d'alimentation pour poissons |
SE0202188D0 (sv) * | 2002-07-11 | 2002-07-11 | Pronova Biocare As | A process for decreasing environmental pollutants in an oil or a fat, a volatile fat or oil environmental pollutants decreasing working fluid, a health supplement, and an animal feed product |
AU2003300264A1 (en) * | 2002-12-20 | 2004-07-22 | Pharmacia Corporation | Compositions of cyclooxygenase-2 selective inhibitors and selective serotonin reuptake inhibitors for the treatment or prevention of a vaso-occlusive event |
US7601756B2 (en) | 2003-06-06 | 2009-10-13 | Snowden Pharmaceuticals, Llc | Method of treatment for irritable bowel syndrome |
CA2534816A1 (fr) * | 2003-06-12 | 2004-12-23 | Evan Newell | Systemes et procedes de traitement de maladies inflammatoires et proliferatives humaines et de lesions au moyen d'inhibiteurs du metabolisme des acides gras et/ou d'inhibiteurs glycolytiques |
US7264813B2 (en) * | 2003-09-24 | 2007-09-04 | Nikken Sohonsha Corporation | Therapeutic uses of Dunaliella powder |
US7510710B2 (en) * | 2004-01-08 | 2009-03-31 | The Regents Of The University Of Colorado | Compositions of UCP inhibitors, Fas antibody, a fatty acid metabolism inhibitor and/or a glucose metabolism inhibitor |
WO2005115370A2 (fr) * | 2004-04-23 | 2005-12-08 | The Regents Of The University Of California | Composes et procedes de traitement de la douleur non inflammatoire au moyen d'agonistes de pparalpha |
DE102004022253A1 (de) * | 2004-05-04 | 2005-12-08 | Phenion Gmbh & Co. Kg | Verwendung von Pirinixinsäure und deren Salzen zur Behandlung von chronisch entzündlichen Krankheiten |
JP2005350451A (ja) * | 2004-05-11 | 2005-12-22 | Santen Pharmaceut Co Ltd | 角結膜障害治療剤 |
CA2571683A1 (fr) * | 2004-06-30 | 2006-01-12 | Combinatorx, Incorporated | Procedes et reactifs pour le traitement de troubles metaboliques |
US20060009506A1 (en) * | 2004-07-09 | 2006-01-12 | Odyssey Thera, Inc. | Drugs for the treatment of neoplastic disorders |
ITMI20041825A1 (it) * | 2004-09-24 | 2004-12-24 | Medestea Res & Production Srl | Agonisti dei ricettori attivanti la proliferazione dei perossisomi, utili nella prevenzione o nel trattamento della gastrite |
CN101098690A (zh) * | 2004-12-06 | 2008-01-02 | 瑞莱恩特医药品有限公司 | 用于血脂治疗的ω-3脂肪酸和脂血异常剂 |
WO2006116217A2 (fr) * | 2005-04-28 | 2006-11-02 | The Regents Of The University Of Colorado | Systemes et procedes servant a traiter des maladies inflammatoires et proliferatives humaines, au moyen d'un compose qui inhibe le metabolisme des acides gras et la glycolyse |
WO2006118821A2 (fr) * | 2005-05-02 | 2006-11-09 | The Regents Of The University Of Colorado | Systemes et procedes de traitement de maladies inflammatoires et proliferatives humaines au moyen d'une combinaison de composes, ou d'un compose bifonctionnel inhibant le metabolisme des acides gras et la glycolyse |
WO2007106912A2 (fr) * | 2006-03-16 | 2007-09-20 | University Of Pittsburgh Of The Commonwealth System Of Higher Education | Agonistes du récepteur-alpha activé de la prolifération des peroxysomes pour la conservation d'organe |
US20100015085A1 (en) * | 2006-05-01 | 2010-01-21 | Johns Hopkins University | Phase 2 inducers and related signaling pathways protect cartilage against inflammation/infection, apoptosis and stress |
FR2999936B1 (fr) * | 2012-12-21 | 2015-01-16 | Urgo Lab | Utilisation d'acide acetylsalicylique pour la prevention et/ou le traitement des plaies du diabetique |
CN105636935B (zh) * | 2013-10-01 | 2018-04-03 | 欧拉泰克治疗有限责任公司 | 3‑苄磺酰基丙腈的药学用途 |
US9999610B2 (en) | 2013-10-01 | 2018-06-19 | Olatec Therapeutics Llc | Pharmaceutical use of 3-benzylsulfonylpropionitrile |
KR101724585B1 (ko) * | 2014-09-15 | 2017-04-10 | 경북대학교 산학협력단 | Pdk 억제제를 유효성분으로 함유하는 만성 염증성 통증 치료용 조성물 |
CA2989052C (fr) | 2015-06-15 | 2020-11-24 | Rush Unversity Medical Center | Ligands ppar-alpha derives du cerveau |
EP3468604B1 (fr) * | 2016-06-08 | 2021-01-20 | Support-Venture GmbH | Combinaisons pharmaceutiques pour le traitement du cancer |
KR101826697B1 (ko) * | 2016-08-25 | 2018-02-07 | 경북대학교 산학협력단 | Pdk 억제제를 유효성분으로 함유하는 만성 염증성 통증 치료용 조성물 |
CN115417825A (zh) * | 2022-08-15 | 2022-12-02 | 山东大学 | 一种五元或六元稠环并嘧啶类环丙基萘衍生物及其制备方法与应用 |
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-
2003
- 2003-01-13 US US10/341,217 patent/US20030212138A1/en not_active Abandoned
- 2003-01-14 CA CA002472168A patent/CA2472168A1/fr not_active Abandoned
- 2003-01-14 WO PCT/US2003/000956 patent/WO2003059294A2/fr not_active Application Discontinuation
- 2003-01-14 MX MXPA04006796A patent/MXPA04006796A/es unknown
- 2003-01-14 KR KR10-2004-7010888A patent/KR20040095207A/ko not_active Application Discontinuation
- 2003-01-14 IL IL16269903A patent/IL162699A0/xx unknown
- 2003-01-14 EP EP03705746A patent/EP1569640A4/fr not_active Withdrawn
- 2003-01-14 AU AU2003207535A patent/AU2003207535A1/en not_active Withdrawn
- 2003-01-14 PL PL03374962A patent/PL374962A1/xx not_active Application Discontinuation
- 2003-01-14 JP JP2003559459A patent/JP2005525313A/ja not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
MXPA04006796A (es) | 2004-12-06 |
KR20040095207A (ko) | 2004-11-12 |
AU2003207535A2 (en) | 2003-07-30 |
EP1569640A2 (fr) | 2005-09-07 |
WO2003059294A2 (fr) | 2003-07-24 |
CA2472168A1 (fr) | 2003-07-24 |
JP2005525313A (ja) | 2005-08-25 |
WO2003059294A3 (fr) | 2005-07-14 |
EP1569640A4 (fr) | 2006-06-21 |
AU2003207535A1 (en) | 2003-07-30 |
US20030212138A1 (en) | 2003-11-13 |
PL374962A1 (en) | 2005-11-14 |
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