IL152889A0 - Imidazopyridine and imidazopyrimidine derivatives and pharmaceutical compositions containing the same - Google Patents
Imidazopyridine and imidazopyrimidine derivatives and pharmaceutical compositions containing the sameInfo
- Publication number
- IL152889A0 IL152889A0 IL15288901A IL15288901A IL152889A0 IL 152889 A0 IL152889 A0 IL 152889A0 IL 15288901 A IL15288901 A IL 15288901A IL 15288901 A IL15288901 A IL 15288901A IL 152889 A0 IL152889 A0 IL 152889A0
- Authority
- IL
- Israel
- Prior art keywords
- imidazopyridine
- same
- pharmaceutical compositions
- compositions containing
- imidazopyrimidine derivatives
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D473/00—Heterocyclic compounds containing purine ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Virology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US21144700P | 2000-06-13 | 2000-06-13 | |
US26336301P | 2001-01-22 | 2001-01-22 | |
PCT/US2001/014775 WO2001095910A1 (fr) | 2000-06-13 | 2001-05-08 | Agents antiviraux d'imidazopyridine et d'imidazopyrimidine |
Publications (1)
Publication Number | Publication Date |
---|---|
IL152889A0 true IL152889A0 (en) | 2003-06-24 |
Family
ID=26906145
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
IL15288901A IL152889A0 (en) | 2000-06-13 | 2001-05-08 | Imidazopyridine and imidazopyrimidine derivatives and pharmaceutical compositions containing the same |
Country Status (20)
Country | Link |
---|---|
US (1) | US6489338B2 (fr) |
EP (1) | EP1311268A4 (fr) |
JP (1) | JP2004503501A (fr) |
KR (1) | KR20030008151A (fr) |
CN (1) | CN1436079A (fr) |
AR (1) | AR029128A1 (fr) |
AU (2) | AU7290601A (fr) |
BR (1) | BR0111569A (fr) |
CA (1) | CA2412327A1 (fr) |
CZ (1) | CZ20024078A3 (fr) |
HU (1) | HUP0400766A2 (fr) |
IL (1) | IL152889A0 (fr) |
MX (1) | MXPA02012204A (fr) |
NO (1) | NO20025977L (fr) |
NZ (1) | NZ523566A (fr) |
PE (1) | PE20011348A1 (fr) |
PL (1) | PL360290A1 (fr) |
RU (1) | RU2003100828A (fr) |
UY (1) | UY26758A1 (fr) |
WO (1) | WO2001095910A1 (fr) |
Families Citing this family (39)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6774134B2 (en) * | 2000-12-20 | 2004-08-10 | Bristol-Myers Squibb Company | Heterocyclic substituted 2-methyl-benzimidazole antiviral agents |
EP1461036A4 (fr) | 2001-12-10 | 2005-11-16 | Bristol Myers Squibb Co | Sel de bis hydrochloride monohydrate d'un inhibiteur de fusion du virus respiratoire syncytial (rsv) |
US6919331B2 (en) * | 2001-12-10 | 2005-07-19 | Bristol-Myers Squibb Company | Substituted 2-methyl-benzimidazole respiratory syncytial virus antiviral agents |
AU2003294249A1 (en) * | 2002-11-08 | 2004-06-03 | Trimeris, Inc. | Hetero-substituted benzimidazole compounds and antiviral uses thereof |
US20050070460A1 (en) * | 2003-08-05 | 2005-03-31 | 3M Innovative Properties Company | Infection prophylaxis using immune response modifier compounds |
CA2541618C (fr) | 2003-10-30 | 2011-12-13 | Boehringer Ingelheim (Canada) Ltd. | Inhibiteurs polymerase rsv |
KR20060127909A (ko) | 2003-12-24 | 2006-12-13 | 비오타 사이언티픽 매니지먼트 피티와이 엘티디 | 호흡기 다핵체 바이러스 감염 치료용 다환 물질 |
GB0406279D0 (en) * | 2004-03-19 | 2004-04-21 | Arrow Therapeutics Ltd | Therapeutic compounds |
GB0406282D0 (en) * | 2004-03-19 | 2004-04-21 | Arrow Therapeutics Ltd | Therapeutic compounds |
KR101238430B1 (ko) | 2004-07-27 | 2013-02-28 | 길리애드 사이언시즈, 인코포레이티드 | 이미다조[4,5-d]피리미딘, 그들의 용도 및 제조방법 |
AU2006260970B2 (en) | 2005-06-20 | 2012-07-05 | Janssen Sciences Ireland Uc | Heterocyclylaminoalkyl substituted benzimidazoles |
AU2006260971B2 (en) | 2005-06-20 | 2011-09-15 | Janssen Sciences Ireland Uc | 2-substituted benzimidazoles |
CA2612263C (fr) | 2005-06-20 | 2015-04-14 | Tibotec Pharmaceuticals Ltd. | 1-(2-amino-3-(alkyl substitue)-3h-benzimidazolylmethyl)-(3-subtitue)-1,3-dihydrobenzoimidazol-2-ones ayant une activite sur le virus syncyntial respiratoire |
TWI423972B (zh) | 2006-09-28 | 2014-01-21 | Biota Scient Management | 治療呼吸系融合細胞病毒感染之多環劑 |
WO2009084544A1 (fr) * | 2007-12-27 | 2009-07-09 | Idemitsu Kosan Co., Ltd. | Dérivé hétérocyclique contenant de l'azote et dispositif organique électroluminescent l'utilisant |
WO2010103306A1 (fr) | 2009-03-10 | 2010-09-16 | Astrazeneca Uk Limited | Dérivés de benzimidazole et leur utilisation comme agents antiviraux |
TWI508968B (zh) | 2010-02-08 | 2015-11-21 | Biota Scient Management | 用於治療呼吸道融合性病毒感染的化合物 |
WO2011115150A1 (fr) * | 2010-03-18 | 2011-09-22 | 興和株式会社 | Procédé pour la production d'un composé de benzothiazine |
US8796303B2 (en) | 2010-11-26 | 2014-08-05 | Biota Scientific Management Pty Ltd. | Imidazo[2,1-G][1,7]naphthyridines for treating respiratory syncytial virus infections |
TWI515187B (zh) * | 2010-12-16 | 2016-01-01 | 健生科學愛爾蘭無限公司 | 作為呼吸道融合病毒抗病毒劑之吲哚類 |
TWI501967B (zh) | 2010-12-16 | 2015-10-01 | Janssen R&D Ireland | 作為呼吸道融合病毒抗病毒劑之氮雜吲哚類 |
TWI541241B (zh) * | 2010-12-16 | 2016-07-11 | 健生科學愛爾蘭無限公司 | 作為呼吸道融合病毒抗病毒劑之咪唑并吡啶類 |
TWI530495B (zh) * | 2010-12-16 | 2016-04-21 | 健生科學愛爾蘭無限公司 | 苯并咪唑呼吸道融合病毒抑制劑 |
TWI527814B (zh) * | 2010-12-16 | 2016-04-01 | 健生科學愛爾蘭無限公司 | 作為呼吸道融合病毒抗病毒劑之氮雜苯并咪唑類 |
CN102690262B (zh) * | 2011-03-23 | 2014-05-28 | 上海市第一人民医院 | 靶向人La蛋白的先导化合物及其在制备抗乙型肝炎病毒的药物中的用途 |
US9550737B2 (en) * | 2012-06-11 | 2017-01-24 | Ucb Biopharma Sprl | TNF -α modulating benzimidazoles |
LT2864323T (lt) * | 2012-06-15 | 2017-07-25 | Janssen Sciences Ireland Uc | 1,3-dihidro-2h-benzimidazol-2-ono dariniai, turintys heterociklų pakaitų, kaip antivirusiniai agentai prieš respiratorinį sincitinį virusą |
KR20150033645A (ko) * | 2012-06-15 | 2015-04-01 | 얀센 알 앤드 디 아일랜드 | 호흡기 합포체 바이러스의 항바이러스제로서의 벤즈이미다졸로 치환된 1,3-디하이드로-2h-벤즈이미다졸-2-온 유도체 |
CN104507916A (zh) * | 2012-06-15 | 2015-04-08 | 爱尔兰詹森研发公司 | 作为呼吸道合胞病毒抗病毒剂的被苯并咪唑取代的4-取代的1,3-二氢-2h-苯并咪唑-2-酮衍生物 |
KR20150032283A (ko) * | 2012-06-15 | 2015-03-25 | 얀센 알 앤드 디 아일랜드 | 호흡기 합포체 바이러스의 항바이러스제로서의 헤테로사이클로 치환된 1,3-디하이드로-2h-벤즈이미다졸-2-온 유도체 |
CN104903313B (zh) * | 2012-10-16 | 2017-12-29 | 爱尔兰詹森科学公司 | Rsv抗病毒化合物 |
JP2016145155A (ja) * | 2013-04-30 | 2016-08-12 | 日本農薬株式会社 | フタルアミド誘導体及び該誘導体を含有する農園芸用殺虫剤並びにその使用方法 |
JP2016535043A (ja) * | 2013-10-29 | 2016-11-10 | メディヴィル・アクチエボラーグ | キナゾリンベースの呼吸器合胞体ウイルス阻害剤 |
WO2015065336A1 (fr) * | 2013-10-29 | 2015-05-07 | Medivir Ab | Inhibiteurs du virus respiratoire syncytial |
EP3414234B1 (fr) * | 2015-10-14 | 2022-06-29 | Zibo Biopolar Changsheng Pharmaceutical Co. Ltd. | Inhibiteurs de la tyrosine kinase de bruton |
WO2019046364A1 (fr) * | 2017-08-29 | 2019-03-07 | Emory University | Inhibiteurs de la réplication du virus respiratoire syncytial (vrs) et leurs utilisations |
WO2021083996A1 (fr) | 2019-10-30 | 2021-05-06 | Janssen Sciences Ireland Unlimited Company | Synthèse de 3-nitro-n-(2,2,2-trifluoroéthyl)-4-pyridinamine |
WO2022184606A1 (fr) * | 2021-03-01 | 2022-09-09 | Janssen Sciences Ireland Unlimited Company | Synthèse de rilématovir |
WO2023143520A1 (fr) * | 2022-01-28 | 2023-08-03 | Insilico Medicine Ip Limited | Inhibiteurs d'ectonucléotide pyrophosphatase-phosphodiestérase 1 (enpp1) et leurs utilisations |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US4324794A (en) | 1980-08-26 | 1982-04-13 | Research Triangle Institute | Inhibition of respiratory syncytial virus-induced cell fusion by amidino compounds |
DK154078C (da) | 1981-02-06 | 1989-05-22 | Ucb Sa | Analogifremgangsmaade til fremstilling af 2-(2-(4-(diphenyl-methyl)-1-piperazinyl)ethoxy)-acetamider eller syreadditionssalte heraf |
US5256668A (en) | 1993-03-17 | 1993-10-26 | American Home Products Corporation | Aminopyrimidine derivatives as antiviral agents for respiratory syncytial virus |
BR9700939A (pt) | 1996-02-13 | 1998-09-01 | American Cyanamid Co | Compostos aniônicos contendo traiazina úteis como agentes antivirais |
JP2002501894A (ja) | 1998-01-29 | 2002-01-22 | バイロファーマ・インコーポレイテッド | ニューモウイルス感染および関連疾患の治療または予防のための化合物、組成物および方法 |
WO2000004900A1 (fr) | 1998-07-20 | 2000-02-03 | Bristol-Myers Squibb Company | Antiviraux a base de benzimidazoles substitues |
JP2003503403A (ja) | 1999-06-28 | 2003-01-28 | ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ | 呼吸合胞体ウイルス複製阻害剤 |
-
2001
- 2001-04-23 US US09/840,279 patent/US6489338B2/en not_active Expired - Fee Related
- 2001-05-08 NZ NZ523566A patent/NZ523566A/en unknown
- 2001-05-08 CA CA002412327A patent/CA2412327A1/fr not_active Abandoned
- 2001-05-08 EP EP01952114A patent/EP1311268A4/fr not_active Withdrawn
- 2001-05-08 WO PCT/US2001/014775 patent/WO2001095910A1/fr not_active Application Discontinuation
- 2001-05-08 KR KR1020027016924A patent/KR20030008151A/ko not_active Application Discontinuation
- 2001-05-08 PL PL36029001A patent/PL360290A1/xx not_active Application Discontinuation
- 2001-05-08 HU HU0400766A patent/HUP0400766A2/hu unknown
- 2001-05-08 AU AU7290601A patent/AU7290601A/xx active Pending
- 2001-05-08 MX MXPA02012204A patent/MXPA02012204A/es unknown
- 2001-05-08 CN CN01811136A patent/CN1436079A/zh active Pending
- 2001-05-08 RU RU2003100828/15A patent/RU2003100828A/ru not_active Application Discontinuation
- 2001-05-08 IL IL15288901A patent/IL152889A0/xx unknown
- 2001-05-08 CZ CZ20024078A patent/CZ20024078A3/cs unknown
- 2001-05-08 BR BR0111569-3A patent/BR0111569A/pt not_active Withdrawn
- 2001-05-08 AU AU2001272906A patent/AU2001272906B2/en not_active Ceased
- 2001-05-08 JP JP2002510088A patent/JP2004503501A/ja not_active Withdrawn
- 2001-06-11 UY UY26758A patent/UY26758A1/es not_active Application Discontinuation
- 2001-06-12 AR ARP010102772A patent/AR029128A1/es unknown
- 2001-06-13 PE PE2001000559A patent/PE20011348A1/es not_active Application Discontinuation
-
2002
- 2002-12-12 NO NO20025977A patent/NO20025977L/no not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
AU2001272906B2 (en) | 2004-08-26 |
HUP0400766A2 (hu) | 2004-07-28 |
JP2004503501A (ja) | 2004-02-05 |
RU2003100828A (ru) | 2004-06-27 |
NZ523566A (en) | 2004-08-27 |
EP1311268A1 (fr) | 2003-05-21 |
US20020016309A1 (en) | 2002-02-07 |
PL360290A1 (en) | 2004-09-06 |
CZ20024078A3 (cs) | 2003-08-13 |
KR20030008151A (ko) | 2003-01-24 |
UY26758A1 (es) | 2002-01-31 |
AU7290601A (en) | 2001-12-24 |
AR029128A1 (es) | 2003-06-04 |
NO20025977D0 (no) | 2002-12-12 |
CA2412327A1 (fr) | 2001-12-20 |
CN1436079A (zh) | 2003-08-13 |
BR0111569A (pt) | 2003-04-29 |
US6489338B2 (en) | 2002-12-03 |
WO2001095910A1 (fr) | 2001-12-20 |
NO20025977L (no) | 2003-01-29 |
EP1311268A4 (fr) | 2004-06-30 |
PE20011348A1 (es) | 2002-02-07 |
MXPA02012204A (es) | 2003-10-15 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
IL152889A0 (en) | Imidazopyridine and imidazopyrimidine derivatives and pharmaceutical compositions containing the same | |
IL150734A0 (en) | Azaindole derivatives and pharmaceutical compositions containing the same | |
IL156354A0 (en) | Pyridoindole derivatives and pharmaceutical compositions containing the same | |
IL152451A0 (en) | 2-chloro-2-nitrophenylcarboxamide derivatives and pharmaceutical compositions containing the same | |
HUP0301178A3 (en) | Glucopyranosyloxybenzylbenzene derivatives and pharmaceutical compositions containing the same | |
IL151952A0 (en) | Aminopyridine derivatives and pharmaceutical compositions containing the same | |
IL153123A0 (en) | N-ureidoheterocycloalkyl-piperidine derivatives and pharmaceutical compositions containing the same | |
IL144977A0 (en) | Pyrrolotriazine derivatives and pharmaceutical compositions containing the same | |
HUP0203895A3 (en) | Substituted azaindoles and pharmaceutical compositions containing them and their use | |
HUP0100179A3 (en) | Imidazopyrimidine and imidazopyridine derivatives and pharmaceutical compositions thereof | |
IL156558A0 (en) | Novel quinuclidine derivatives and medicinal compositions containing the same | |
EG24066A (en) | Novel quinuclidine derivatives and medicinal compositions containing the same | |
IL166232A0 (en) | Azaindole derivatives and pharmaceutical compositions containing the same | |
IL152490A0 (en) | Pyridine derivatives and pharmaceutical compositions containing the same | |
HUP0400784A3 (en) | Bicyclic heterocondensated pyrrolcarboxamide derivatives, their use and pharmaceutical compositions containing them | |
IL161616A0 (en) | Indazolypyrrolotriazine derivatives and pharmaceutical compositions containing the same | |
IL150224A0 (en) | Lipopeptides and pharmaceutical compositions containing the same | |
IL150223A0 (en) | Lipopeptides and pharmaceutical compositions containing the same | |
IL158044A0 (en) | Cyclopropylindole derivatives and pharmaceutical compositions containing the same | |
IL158300A0 (en) | Bisarylimidazol derivatives and pharmaceutical compositions containing the same | |
IL156812A0 (en) | Phthalazinone-piperidino derivatives and pharmaceutical compositions containing the same | |
IL152094A0 (en) | Ecteinascidin derivatives and pharmaceutical compositions containing the same | |
IL155067A0 (en) | (dihydro) isoquinoline derivatives and pharmaceutical compositions containing the same | |
IL147214A0 (en) | 1-methylcarbapenem derivatives and pharmaceutical compositions containing the same | |
IL150905A0 (en) | Andrographolide derivatives and pharmaceutical compositions containing the same |