ID29241A - Turunan-turunan kinolin teranelasi-1,2 - Google Patents

Turunan-turunan kinolin teranelasi-1,2

Info

Publication number
ID29241A
ID29241A IDW00200101373A ID20011373A ID29241A ID 29241 A ID29241 A ID 29241A ID W00200101373 A IDW00200101373 A ID W00200101373A ID 20011373 A ID20011373 A ID 20011373A ID 29241 A ID29241 A ID 29241A
Authority
ID
Indonesia
Prior art keywords
teranelasi
kinolin
districts
teranelasi kinolin
kinolin districts
Prior art date
Application number
IDW00200101373A
Other languages
English (en)
Indonesian (id)
Inventor
Rene Patrick Angibaud
Marc Gaston Venet
Xavier Marc Bourdrez
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of ID29241A publication Critical patent/ID29241A/id

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/4738Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/4745Quinolines; Isoquinolines ortho- or peri-condensed with heterocyclic ring systems condensed with ring systems having nitrogen as a ring hetero atom, e.g. phenantrolines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/498Pyrazines or piperazines ortho- and peri-condensed with carbocyclic ring systems, e.g. quinoxaline, phenazine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D403/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
    • C07D403/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/06Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Quinoline Compounds (AREA)
  • Processing And Handling Of Plastics And Other Materials For Molding In General (AREA)
  • Information Retrieval, Db Structures And Fs Structures Therefor (AREA)
IDW00200101373A 1998-12-23 1999-12-17 Turunan-turunan kinolin teranelasi-1,2 ID29241A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP98204444 1998-12-23

Publications (1)

Publication Number Publication Date
ID29241A true ID29241A (id) 2001-08-16

Family

ID=8234557

Family Applications (1)

Application Number Title Priority Date Filing Date
IDW00200101373A ID29241A (id) 1998-12-23 1999-12-17 Turunan-turunan kinolin teranelasi-1,2

Country Status (32)

Country Link
US (2) US6458800B1 (cs)
EP (1) EP1140935B1 (cs)
JP (1) JP4725940B2 (cs)
KR (2) KR100712226B1 (cs)
CN (1) CN1178938C (cs)
AR (1) AR021995A1 (cs)
AT (1) ATE240327T1 (cs)
AU (1) AU765437B2 (cs)
BG (1) BG65124B1 (cs)
BR (1) BR9916827A (cs)
CA (1) CA2355717C (cs)
CZ (1) CZ302374B6 (cs)
DE (1) DE69907964T2 (cs)
DK (1) DK1140935T3 (cs)
EA (1) EA004542B1 (cs)
EE (1) EE04962B1 (cs)
ES (1) ES2200591T3 (cs)
HK (1) HK1038746B (cs)
HR (1) HRP20010454B1 (cs)
HU (1) HU229404B1 (cs)
ID (1) ID29241A (cs)
IL (2) IL143859A0 (cs)
NO (1) NO318922B1 (cs)
PL (1) PL199080B1 (cs)
PT (1) PT1140935E (cs)
SI (1) SI1140935T1 (cs)
SK (1) SK286072B6 (cs)
TR (1) TR200101961T2 (cs)
TW (1) TW531533B (cs)
UA (1) UA71592C2 (cs)
WO (1) WO2000039082A2 (cs)
ZA (1) ZA200105136B (cs)

Families Citing this family (67)

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CA2396865C (en) * 2000-02-04 2009-04-14 Janssen Pharmaceutica N.V. Farnesyl protein transferase inhibitors for treating breast cancer
US6838467B2 (en) 2000-02-24 2005-01-04 Janssen Pharmaceutica N. V. Dosing regimen
EP1261348A2 (en) * 2000-02-29 2002-12-04 Janssen Pharmaceutica N.V. Combinations of a farnesyl protein transferase inhibitor with nitrogen mustard or nitrosourea alkylating agents
WO2001064246A2 (en) * 2000-02-29 2001-09-07 Janssen Pharmaceutica N.V. Farnesyl protein transferase inhibitor combinations with an her2 antibody
CA2397475A1 (en) * 2000-02-29 2001-09-07 Janssen Pharmaceutica N.V. Farnesyl protein transferase inhibitor combinations with vinca alkaloids
WO2001064226A2 (en) * 2000-02-29 2001-09-07 Janssen Pharmaceutica N.V. Farnesyl protein transferase inhibitor combinations with platinum compounds
AU2001244166A1 (en) * 2000-02-29 2001-09-12 Janssen Pharmaceutica N.V. Farnesyl protein transferase inhibitor combinations with further anti-cancer agents
CA2397694A1 (en) * 2000-02-29 2001-09-07 Janssen Pharmaceutica Inc. Farnesyl protein transferase inhibitor combinations
AU2001246478A1 (en) * 2000-02-29 2001-09-12 Janssen Pharmaceutica N.V. Farnesyl protein transferase inhibitor combinations with taxane compounds
EP1267872A2 (en) * 2000-02-29 2003-01-02 Janssen Pharmaceutica N.V. Farnesyl protein transferase inhibitor combinations with anti-tumor anthracycline derivatives
CA2397256A1 (en) * 2000-02-29 2001-09-07 Mary Ellen Margaret Rybak Farnesyl protein transferase inhibitor combinations with anti-tumor podophyllotoxin derivatives
AU2001256166A1 (en) * 2000-02-29 2001-09-12 Janssen Pharmaceutica N.V. Farnesyl protein transferase inhibitor combinations with anti-tumor nucleoside derivatives
JP2003525234A (ja) * 2000-02-29 2003-08-26 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ カンプトテシン化合物とのファルネシルタンパク質トランスフェラーゼ阻害剤の組み合わせ剤
JO2361B1 (en) 2000-06-22 2006-12-12 جانسين فارماسيوتيكا ان. في Enaniumer 1,2-anylated quinoline inhibitor for the transporter - farnesyl
EP1322644A1 (en) * 2000-09-25 2003-07-02 Janssen Pharmaceutica N.V. Farnesyl transferase inhibiting 6-heterocyclylmethyl quinolinone derivatives
EP1322636A1 (en) 2000-09-25 2003-07-02 Janssen Pharmaceutica N.V. Farnesyl transferase inhibiting 6- (substituted phenyl)methyl]-quinoline and quinazoline derivatives
AU2001293826A1 (en) * 2000-09-25 2002-04-02 Janssen Pharmaceutica N.V. Farnesyl transferase inhibiting quinoline and quinazoline derivatives as farnesyl transferase inhibitors
JP4974438B2 (ja) * 2000-09-25 2012-07-11 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ ファルネシルトランスフェラーゼを阻害する6−ヘテロシクリルメチルキノリンおよびキナゾリン誘導体
EA007464B1 (ru) * 2000-10-02 2006-10-27 Янссен Фармацевтика Н.В. Антагонисты метаботропных рецепторов глутамата
DE60139080D1 (de) * 2000-11-21 2009-08-06 Janssen Pharmaceutica Nv Farnesyltransferase hemmende benzoheterocyclische derivate
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DE60117847T2 (de) 2000-12-27 2006-11-16 Janssen Pharmaceutica N.V. Farnesyltransferase hemmende, in der 4-stellung substituierte chinolin- und chinazolinderivate
ATE415161T1 (de) * 2001-02-15 2008-12-15 Janssen Pharmaceutica Nv Farnesyl-protein-transferase hemmer in kombination mit antiöstrogenen
US20040157773A1 (en) * 2001-04-25 2004-08-12 End David William Farnesyl protein transferase inhibitors for treating cachexia
US6740757B2 (en) * 2001-08-29 2004-05-25 Pfizer Inc Enantiomers of 6-[(4-chloro-phenyl)-hydroxy-(3-methyl-3h-imidazol-4-yl)-methyl]-4-[3-(3-hydroxy-3-methyl-but-1-ynyl)-phenyl]-1-methyl-1h-quinolin-2-one and salts thereof, useful in the treatment of cancer
CA2468015A1 (en) * 2001-11-27 2003-06-05 Merck & Co., Inc. 2-aminoquinoline compounds
AU2002358677B2 (en) 2001-12-19 2008-02-07 Janssen Pharmaceutica N.V. 1,8-annelated quinoline derivatives substituted with carbon-linked triazoles as farnesyl transferase inhibitors
EP1490065B1 (en) 2002-03-22 2007-06-13 Janssen Pharmaceutica N.V. Benzylimidazolyl substituted 2-quinolinone and quinazolinone derivatives for use as farnesyl transferase inhibitors
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JP4384505B2 (ja) * 2002-04-15 2009-12-16 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ ファルネシルトランスフェラーゼを阻害する炭素連結イミダゾールもしくはトリアゾール置換三環状キナゾリン誘導体
US20030125268A1 (en) * 2002-08-28 2003-07-03 Rybak Mary Ellen Margaret Farnesyl protein transferase inhibitor combinations with anti-tumor anthracycline derivatives
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Also Published As

Publication number Publication date
BR9916827A (pt) 2001-10-16
PL349504A1 (en) 2002-07-29
ES2200591T3 (es) 2004-03-01
IL143859A0 (en) 2002-04-21
KR20010087396A (ko) 2001-09-15
EE200100318A (et) 2002-10-15
HUP0104582A3 (en) 2002-12-28
DE69907964D1 (de) 2003-06-18
AU765437B2 (en) 2003-09-18
CZ20012142A3 (cs) 2002-01-16
SI1140935T1 (en) 2003-10-31
BG105631A (en) 2002-02-28
US20030119843A1 (en) 2003-06-26
UA71592C2 (uk) 2004-12-15
CN1331693A (zh) 2002-01-16
DE69907964T2 (de) 2004-02-19
IL143859A (en) 2008-04-13
EP1140935A2 (en) 2001-10-10
HU229404B1 (en) 2013-12-30
NO20013088L (no) 2001-06-21
NO318922B1 (no) 2005-05-23
EP1140935B1 (en) 2003-05-14
SK286072B6 (sk) 2008-02-05
AR021995A1 (es) 2002-09-04
HUP0104582A2 (hu) 2002-04-29
EA200100708A1 (ru) 2001-12-24
ZA200105136B (en) 2002-06-21
CA2355717A1 (en) 2000-07-06
KR100712226B1 (ko) 2007-04-27
AU2795300A (en) 2000-07-31
PL199080B1 (pl) 2008-08-29
WO2000039082A2 (en) 2000-07-06
CZ302374B6 (cs) 2011-04-20
TR200101961T2 (tr) 2001-12-21
HK1038746A1 (en) 2002-03-28
CA2355717C (en) 2011-02-08
KR100818541B1 (ko) 2008-04-02
BG65124B1 (bg) 2007-03-30
EE04962B1 (et) 2008-02-15
WO2000039082A3 (en) 2000-10-26
JP4725940B2 (ja) 2011-07-13
KR20060117380A (ko) 2006-11-16
JP2002533435A (ja) 2002-10-08
HK1038746B (en) 2003-09-05
US6914066B2 (en) 2005-07-05
EA004542B1 (ru) 2004-06-24
DK1140935T3 (da) 2003-09-01
NO20013088D0 (no) 2001-06-21
ATE240327T1 (de) 2003-05-15
US6458800B1 (en) 2002-10-01
PT1140935E (pt) 2003-10-31
SK8732001A3 (en) 2002-02-05
HRP20010454A2 (en) 2002-06-30
CN1178938C (zh) 2004-12-08
HRP20010454B1 (en) 2004-06-30
TW531533B (en) 2003-05-11

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