ATE275151T1 - 3,6-ketal-makrolidantibiotika - Google Patents
3,6-ketal-makrolidantibiotikaInfo
- Publication number
- ATE275151T1 ATE275151T1 AT99301325T AT99301325T ATE275151T1 AT E275151 T1 ATE275151 T1 AT E275151T1 AT 99301325 T AT99301325 T AT 99301325T AT 99301325 T AT99301325 T AT 99301325T AT E275151 T1 ATE275151 T1 AT E275151T1
- Authority
- AT
- Austria
- Prior art keywords
- macrolida
- ketal
- antibiotic
- macrolida antibiotic
- ketal macrolida
- Prior art date
Links
- 230000003115 biocidal effect Effects 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Tropical Medicine & Parasitology (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US7663098P | 1998-03-03 | 1998-03-03 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE275151T1 true ATE275151T1 (de) | 2004-09-15 |
Family
ID=22133253
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT99301325T ATE275151T1 (de) | 1998-03-03 | 1999-02-23 | 3,6-ketal-makrolidantibiotika |
Country Status (17)
| Country | Link |
|---|---|
| US (1) | US6043226A (de) |
| EP (1) | EP0941998B1 (de) |
| JP (1) | JP3666788B2 (de) |
| CN (1) | CN1244532A (de) |
| AR (1) | AR016715A1 (de) |
| AT (1) | ATE275151T1 (de) |
| AU (1) | AU741435B2 (de) |
| BR (1) | BR9900856A (de) |
| CA (1) | CA2263203C (de) |
| DE (1) | DE69919769T2 (de) |
| DK (1) | DK0941998T3 (de) |
| ES (1) | ES2226282T3 (de) |
| HU (1) | HUP9900492A3 (de) |
| NO (1) | NO312366B1 (de) |
| NZ (1) | NZ334442A (de) |
| PT (1) | PT941998E (de) |
| ZA (1) | ZA991664B (de) |
Families Citing this family (30)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AP9801420A0 (en) * | 1998-01-02 | 1998-12-31 | Pfizer Prod Inc | Novel macrolides. |
| AP1060A (en) * | 1998-01-02 | 2002-04-23 | Pfizer Prod Inc | Novel erythromycin derivatives. |
| ID28286A (id) * | 1998-11-03 | 2001-05-10 | Pfizer Prod Inc | Antibiotik-antibiotik makrolida baru |
| US6514944B2 (en) | 1999-04-16 | 2003-02-04 | Kosan Biosciences, Inc. | Macrolide antiinfective agents |
| US6590083B1 (en) * | 1999-04-16 | 2003-07-08 | Ortho-Mcneil Pharmaceutical, Inc. | Ketolide antibacterials |
| AU775637B2 (en) | 1999-04-16 | 2004-08-12 | Kosan Biosciences, Inc. | Macrolide antiinfective agents |
| US6939861B2 (en) | 1999-04-16 | 2005-09-06 | Kosan Biosciences, Inc. | Amido macrolides |
| US6451768B1 (en) * | 1999-04-16 | 2002-09-17 | Kosan Biosciences, Inc. | Macrolide antiinfective agents |
| BR0010938A (pt) * | 1999-05-24 | 2002-03-19 | Pfizer Prod Inc | Derivados da 13-metil eritromicina |
| EP1146051A3 (de) * | 2000-04-10 | 2001-10-31 | Pfizer Products Inc. | Erythromycin A-Derivate |
| AU2001214707A1 (en) * | 2000-11-07 | 2002-05-21 | Morphotek Inc. | Methods for isolating novel antimicrobial agents from hypermutable mammalian cells |
| US8063021B2 (en) * | 2002-01-17 | 2011-11-22 | Kosan Biosciences Incorporated | Ketolide anti-infective compounds |
| ITMI20021726A1 (it) | 2002-08-01 | 2004-02-02 | Zambon Spa | Macrolidi ad attivita' antiinfiammatoria. |
| ITMI20022292A1 (it) * | 2002-10-29 | 2004-04-30 | Zambon Spa | 9a-azalidi ad attivita' antiinfiammatoria. |
| WO2004073492A2 (en) * | 2003-02-14 | 2004-09-02 | Massachusetts Eye And Ear Infirmary | Chlamydia pneumoniae associated chronic intraocular disorders and treatment thereof |
| PL1836211T3 (pl) * | 2004-12-21 | 2010-07-30 | Pfizer Prod Inc | Makrolidy |
| US7517859B2 (en) * | 2005-05-04 | 2009-04-14 | Enanta Pharmaceuticals, Inc. | Spirocyclic bicyclolides |
| CN104004039A (zh) * | 2007-09-17 | 2014-08-27 | 英安塔制药有限公司 | 6,11-桥联的联芳大环内酯类 |
| JP2020517749A (ja) * | 2017-04-20 | 2020-06-18 | ライジング タイド ファウンデーション | 抗がん剤としてホスホニウムイオンを含むアジスロマイシン誘導体 |
| WO2018193126A1 (en) * | 2017-04-20 | 2018-10-25 | Novintum Biotechnology Gmbh | Azithromycin derivatives containing a phosphonium ion as antibacterial agents |
| CA3079368A1 (en) | 2017-04-20 | 2018-10-25 | Rising Tide Foundation | Azithromycin derivatives containing a phosphonium ion as anticancer agents |
| WO2018193111A1 (en) * | 2017-04-20 | 2018-10-25 | Novintum Biotechnology Gmbh | Azithromycin derivatives containing a phosphonium ion as anticancer agents |
| GB201706299D0 (en) * | 2017-04-20 | 2017-06-07 | Novintum Biotechnology Gmbh | Compounds |
| WO2018193116A1 (en) * | 2017-04-20 | 2018-10-25 | Novintum Biotechnology Gmbh | Azithromycin derivatives containing a phosphonium ion as anticancer agents |
| WO2018195434A1 (en) | 2017-04-21 | 2018-10-25 | Lisanti Michael P | Vitamin c and doxycycline: a synthetic lethal combination therapy for eradicating cancer stem cells (cscs) |
| US11229657B2 (en) | 2017-04-21 | 2022-01-25 | Lunella Biotech, Inc. | Targeting hypoxic cancer stem cells (CSCs) with doxycycline: implications for improving anti-angiogenic therapy |
| KR20200010343A (ko) | 2017-05-19 | 2020-01-30 | 루넬라 바이오테크 인코포레이티드 | 안티미토신: 암 줄기 세포를 근절하기 위한 미토콘드리아 생물발생의 표적화 억제제 |
| WO2018213764A1 (en) | 2017-05-19 | 2018-11-22 | Lunella Biotech, Inc. | Companion diagnostics for mitochondrial inhibitors |
| MX2019014806A (es) | 2017-06-26 | 2020-02-10 | Lunella Biotech Inc | Mitocetoscinas: agentes terapeuticos basados en mitocondrias que fijan como objetivo el metabolismo de cetonas en celulas cancerosas. |
| GB201817083D0 (en) * | 2018-10-19 | 2018-12-05 | Novintum Biotechnology Gmbh | Compounds |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8721165D0 (en) * | 1987-09-09 | 1987-10-14 | Beecham Group Plc | Chemical compounds |
| EP0344106A3 (de) * | 1988-05-24 | 1990-01-31 | Ciba-Geigy Ag | Blaue Dispersionsfarbstoffe und Mischungen blauer Dispersionsfarbstoffe |
| US5302705A (en) * | 1989-10-07 | 1994-04-12 | Taisho Pharmaceutical Co., Ltd. | 6-O-methylerythromycin a oxime derivatives |
| WO1994017088A1 (fr) * | 1993-01-26 | 1994-08-04 | Taisho Pharmaceutical Co., Ltd. | Derive de 5-o-desosaminylerythronolide |
| WO1997042204A1 (en) * | 1996-05-07 | 1997-11-13 | Abbott Laboratories | 6-o-substituted erythromycins and method for making them |
-
1999
- 1999-02-23 DE DE69919769T patent/DE69919769T2/de not_active Expired - Fee Related
- 1999-02-23 PT PT99301325T patent/PT941998E/pt unknown
- 1999-02-23 ES ES99301325T patent/ES2226282T3/es not_active Expired - Lifetime
- 1999-02-23 AT AT99301325T patent/ATE275151T1/de not_active IP Right Cessation
- 1999-02-23 DK DK99301325T patent/DK0941998T3/da active
- 1999-02-23 EP EP99301325A patent/EP0941998B1/de not_active Expired - Lifetime
- 1999-02-25 US US09/257,709 patent/US6043226A/en not_active Expired - Fee Related
- 1999-03-01 AR ARP990100858A patent/AR016715A1/es unknown
- 1999-03-01 CA CA002263203A patent/CA2263203C/en not_active Expired - Fee Related
- 1999-03-02 NZ NZ334442A patent/NZ334442A/xx unknown
- 1999-03-02 NO NO19991012A patent/NO312366B1/no not_active IP Right Cessation
- 1999-03-02 ZA ZA9901664A patent/ZA991664B/xx unknown
- 1999-03-02 HU HU9900492A patent/HUP9900492A3/hu unknown
- 1999-03-02 JP JP05371599A patent/JP3666788B2/ja not_active Expired - Fee Related
- 1999-03-03 BR BR9900856-4A patent/BR9900856A/pt not_active IP Right Cessation
- 1999-03-03 AU AU18562/99A patent/AU741435B2/en not_active Ceased
- 1999-03-03 CN CN99105681A patent/CN1244532A/zh active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| HUP9900492A2 (hu) | 1999-09-28 |
| CA2263203A1 (en) | 1999-09-03 |
| JPH11315093A (ja) | 1999-11-16 |
| US6043226A (en) | 2000-03-28 |
| CA2263203C (en) | 2002-09-03 |
| CN1244532A (zh) | 2000-02-16 |
| DK0941998T3 (da) | 2004-09-20 |
| AU1856299A (en) | 1999-09-16 |
| NZ334442A (en) | 2000-03-27 |
| ES2226282T3 (es) | 2005-03-16 |
| EP0941998B1 (de) | 2004-09-01 |
| NO991012L (no) | 1999-09-06 |
| ZA991664B (en) | 2000-10-12 |
| PT941998E (pt) | 2004-12-31 |
| AU741435B2 (en) | 2001-11-29 |
| DE69919769T2 (de) | 2005-01-27 |
| EP0941998A3 (de) | 1999-10-06 |
| NO991012D0 (no) | 1999-03-02 |
| BR9900856A (pt) | 2000-04-25 |
| JP3666788B2 (ja) | 2005-06-29 |
| NO312366B1 (no) | 2002-04-29 |
| HUP9900492A3 (en) | 2001-08-28 |
| AR016715A1 (es) | 2001-07-25 |
| HU9900492D0 (en) | 1999-04-28 |
| DE69919769D1 (de) | 2004-10-07 |
| EP0941998A2 (de) | 1999-09-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| UEP | Publication of translation of european patent specification |
Ref document number: 0941998 Country of ref document: EP |
|
| REN | Ceased due to non-payment of the annual fee |