HUP9900492A2 - 3,6-Ketál és enol-éter makrolid antibiotikumok és ezeket tartalmazó gyógyszerkészítmények - Google Patents
3,6-Ketál és enol-éter makrolid antibiotikumok és ezeket tartalmazó gyógyszerkészítményekInfo
- Publication number
- HUP9900492A2 HUP9900492A2 HU9900492A HUP9900492A HUP9900492A2 HU P9900492 A2 HUP9900492 A2 HU P9900492A2 HU 9900492 A HU9900492 A HU 9900492A HU P9900492 A HUP9900492 A HU P9900492A HU P9900492 A2 HUP9900492 A2 HU P9900492A2
- Authority
- HU
- Hungary
- Prior art keywords
- contg
- ketal
- pharmaceuticals
- enol ether
- macrolide antibiotics
- Prior art date
Links
- 239000003814 drug Substances 0.000 title 1
- 150000002084 enol ethers Chemical class 0.000 title 1
- 239000003120 macrolide antibiotic agent Substances 0.000 title 1
- 208000035143 Bacterial infection Diseases 0.000 abstract 2
- 206010017533 Fungal infection Diseases 0.000 abstract 2
- 208000031888 Mycoses Diseases 0.000 abstract 2
- 208000030852 Parasitic disease Diseases 0.000 abstract 2
- 230000001580 bacterial effect Effects 0.000 abstract 2
- 208000022362 bacterial infectious disease Diseases 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 230000003071 parasitic effect Effects 0.000 abstract 2
- 241000251468 Actinopterygii Species 0.000 abstract 1
- 241000271566 Aves Species 0.000 abstract 1
- 241000124008 Mammalia Species 0.000 abstract 1
- 239000000825 pharmaceutical preparation Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/04—Antineoplastic agents specific for metastasis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Animal Behavior & Ethology (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Oncology (AREA)
- Communicable Diseases (AREA)
- Tropical Medicine & Parasitology (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Biotechnology (AREA)
- Genetics & Genomics (AREA)
- Molecular Biology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Abstract
A találmány tárgya (1) vagy (2) általánős képletű vegyület, melyalkalmas baktériűm, parazita vagy prőtőzőőn őkőzta fertőzések,valamint baktériűm, parazita vagy prőtőzőőn őkőzta fertőzésselkapcsőlatős betegségek kezelésére emlősöknél, halaknál és madaraknál.A találmány tővábbi tárgyát képezik az (1) vagy (2) általánős képletűvegyületet tartalmaz gyógyszerkészítmények is. ŕ
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US7663098P | 1998-03-03 | 1998-03-03 |
Publications (3)
Publication Number | Publication Date |
---|---|
HU9900492D0 HU9900492D0 (en) | 1999-04-28 |
HUP9900492A2 true HUP9900492A2 (hu) | 1999-09-28 |
HUP9900492A3 HUP9900492A3 (en) | 2001-08-28 |
Family
ID=22133253
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
HU9900492A HUP9900492A3 (en) | 1998-03-03 | 1999-03-02 | 3,6-ketal and enol ether macrolide antibiotics and pharmaceuticals contg. them |
Country Status (17)
Country | Link |
---|---|
US (1) | US6043226A (hu) |
EP (1) | EP0941998B1 (hu) |
JP (1) | JP3666788B2 (hu) |
CN (1) | CN1244532A (hu) |
AR (1) | AR016715A1 (hu) |
AT (1) | ATE275151T1 (hu) |
AU (1) | AU741435B2 (hu) |
BR (1) | BR9900856A (hu) |
CA (1) | CA2263203C (hu) |
DE (1) | DE69919769T2 (hu) |
DK (1) | DK0941998T3 (hu) |
ES (1) | ES2226282T3 (hu) |
HU (1) | HUP9900492A3 (hu) |
NO (1) | NO312366B1 (hu) |
NZ (1) | NZ334442A (hu) |
PT (1) | PT941998E (hu) |
ZA (1) | ZA991664B (hu) |
Families Citing this family (29)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AP9801420A0 (en) * | 1998-01-02 | 1998-12-31 | Pfizer Prod Inc | Novel macrolides. |
AP1060A (en) * | 1998-01-02 | 2002-04-23 | Pfizer Prod Inc | Novel erythromycin derivatives. |
HUP0104192A3 (en) | 1998-11-03 | 2003-12-29 | Pfizer Prod Inc | Novel macrolide antibiotics |
US6939861B2 (en) | 1999-04-16 | 2005-09-06 | Kosan Biosciences, Inc. | Amido macrolides |
US6451768B1 (en) * | 1999-04-16 | 2002-09-17 | Kosan Biosciences, Inc. | Macrolide antiinfective agents |
WO2000063224A2 (en) | 1999-04-16 | 2000-10-26 | Kosan Biosciences, Inc. | Macrolide antiinfective agents |
US6590083B1 (en) * | 1999-04-16 | 2003-07-08 | Ortho-Mcneil Pharmaceutical, Inc. | Ketolide antibacterials |
US6514944B2 (en) * | 1999-04-16 | 2003-02-04 | Kosan Biosciences, Inc. | Macrolide antiinfective agents |
IL145739A0 (en) * | 1999-05-24 | 2002-07-25 | Pfizer Prod Inc | 13-methyl-erythromycin derivatives |
EP1146051A3 (en) * | 2000-04-10 | 2001-10-31 | Pfizer Products Inc. | Erythromycin A derivatives |
CA2428158C (en) * | 2000-11-07 | 2010-06-29 | Morphotek, Inc. | Methods for isolating novel antimicrobial agents from hypermutable mammalian cells |
US8063021B2 (en) * | 2002-01-17 | 2011-11-22 | Kosan Biosciences Incorporated | Ketolide anti-infective compounds |
ITMI20021726A1 (it) | 2002-08-01 | 2004-02-02 | Zambon Spa | Macrolidi ad attivita' antiinfiammatoria. |
ITMI20022292A1 (it) * | 2002-10-29 | 2004-04-30 | Zambon Spa | 9a-azalidi ad attivita' antiinfiammatoria. |
US20060141470A1 (en) * | 2003-02-14 | 2006-06-29 | Kalayoglu Murat V | Chlamydia pneumoniae associated chronic intraocular disorders and treatment thereof |
EA011281B1 (ru) * | 2004-12-21 | 2009-02-27 | Пфайзер Продактс Инк. | Макролиды |
US7517859B2 (en) * | 2005-05-04 | 2009-04-14 | Enanta Pharmaceuticals, Inc. | Spirocyclic bicyclolides |
EP2203435B1 (en) * | 2007-09-17 | 2018-07-18 | Enanta Pharmaceuticals, Inc. | 6, 11-bridged biaryl macrolides |
WO2018193126A1 (en) * | 2017-04-20 | 2018-10-25 | Novintum Biotechnology Gmbh | Azithromycin derivatives containing a phosphonium ion as antibacterial agents |
GB201706299D0 (en) * | 2017-04-20 | 2017-06-07 | Novintum Biotechnology Gmbh | Compounds |
WO2018193111A1 (en) * | 2017-04-20 | 2018-10-25 | Novintum Biotechnology Gmbh | Azithromycin derivatives containing a phosphonium ion as anticancer agents |
CN111148750A (zh) * | 2017-04-20 | 2020-05-12 | 来兴泰德基金会 | 作为抗癌剂的包含鏻离子的阿奇霉素衍生物 |
US11560395B2 (en) | 2017-04-20 | 2023-01-24 | Rising Tide Foundation | Azithromycin derivatives containing a phosphonium ion as anticancer agents |
WO2018193116A1 (en) * | 2017-04-20 | 2018-10-25 | Novintum Biotechnology Gmbh | Azithromycin derivatives containing a phosphonium ion as anticancer agents |
US11229657B2 (en) | 2017-04-21 | 2022-01-25 | Lunella Biotech, Inc. | Targeting hypoxic cancer stem cells (CSCs) with doxycycline: implications for improving anti-angiogenic therapy |
US11197872B2 (en) | 2017-04-21 | 2021-12-14 | Lunella Biotech, Inc. | Vitamin C and doxycycline: a synthetic lethal combination therapy for eradicating cancer stem cells (CSCs) |
KR20200010343A (ko) | 2017-05-19 | 2020-01-30 | 루넬라 바이오테크 인코포레이티드 | 안티미토신: 암 줄기 세포를 근절하기 위한 미토콘드리아 생물발생의 표적화 억제제 |
SG11201913134UA (en) | 2017-06-26 | 2020-01-30 | Lunella Biotech Inc | Mitoketoscins: mitochondrial-based therapeutics targeting ketone metabolism in cancer cells |
GB201817083D0 (en) * | 2018-10-19 | 2018-12-05 | Novintum Biotechnology Gmbh | Compounds |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8721165D0 (en) * | 1987-09-09 | 1987-10-14 | Beecham Group Plc | Chemical compounds |
EP0344106A3 (de) * | 1988-05-24 | 1990-01-31 | Ciba-Geigy Ag | Blaue Dispersionsfarbstoffe und Mischungen blauer Dispersionsfarbstoffe |
US5302705A (en) * | 1989-10-07 | 1994-04-12 | Taisho Pharmaceutical Co., Ltd. | 6-O-methylerythromycin a oxime derivatives |
US5602239A (en) * | 1993-01-26 | 1997-02-11 | Taisho Pharmaceutical Co., Ltd. | 5-O-desosaminylerythronolide derivatives |
AU2340797A (en) * | 1996-05-07 | 1997-11-26 | Abbott Laboratories | 6-o-substituted erythromycins and method for making them |
-
1999
- 1999-02-23 EP EP99301325A patent/EP0941998B1/en not_active Expired - Lifetime
- 1999-02-23 DK DK99301325T patent/DK0941998T3/da active
- 1999-02-23 DE DE69919769T patent/DE69919769T2/de not_active Expired - Fee Related
- 1999-02-23 PT PT99301325T patent/PT941998E/pt unknown
- 1999-02-23 AT AT99301325T patent/ATE275151T1/de not_active IP Right Cessation
- 1999-02-23 ES ES99301325T patent/ES2226282T3/es not_active Expired - Lifetime
- 1999-02-25 US US09/257,709 patent/US6043226A/en not_active Expired - Fee Related
- 1999-03-01 AR ARP990100858A patent/AR016715A1/es unknown
- 1999-03-01 CA CA002263203A patent/CA2263203C/en not_active Expired - Fee Related
- 1999-03-02 NZ NZ334442A patent/NZ334442A/xx unknown
- 1999-03-02 ZA ZA9901664A patent/ZA991664B/xx unknown
- 1999-03-02 HU HU9900492A patent/HUP9900492A3/hu unknown
- 1999-03-02 NO NO19991012A patent/NO312366B1/no not_active IP Right Cessation
- 1999-03-02 JP JP05371599A patent/JP3666788B2/ja not_active Expired - Fee Related
- 1999-03-03 AU AU18562/99A patent/AU741435B2/en not_active Ceased
- 1999-03-03 BR BR9900856-4A patent/BR9900856A/pt not_active IP Right Cessation
- 1999-03-03 CN CN99105681A patent/CN1244532A/zh active Pending
Also Published As
Publication number | Publication date |
---|---|
DK0941998T3 (da) | 2004-09-20 |
AU741435B2 (en) | 2001-11-29 |
NZ334442A (en) | 2000-03-27 |
CA2263203C (en) | 2002-09-03 |
NO991012D0 (no) | 1999-03-02 |
NO312366B1 (no) | 2002-04-29 |
AR016715A1 (es) | 2001-07-25 |
HUP9900492A3 (en) | 2001-08-28 |
DE69919769D1 (de) | 2004-10-07 |
CN1244532A (zh) | 2000-02-16 |
EP0941998B1 (en) | 2004-09-01 |
HU9900492D0 (en) | 1999-04-28 |
ATE275151T1 (de) | 2004-09-15 |
ES2226282T3 (es) | 2005-03-16 |
JPH11315093A (ja) | 1999-11-16 |
DE69919769T2 (de) | 2005-01-27 |
EP0941998A3 (en) | 1999-10-06 |
US6043226A (en) | 2000-03-28 |
AU1856299A (en) | 1999-09-16 |
CA2263203A1 (en) | 1999-09-03 |
JP3666788B2 (ja) | 2005-06-29 |
NO991012L (no) | 1999-09-06 |
EP0941998A2 (en) | 1999-09-15 |
PT941998E (pt) | 2004-12-31 |
ZA991664B (en) | 2000-10-12 |
BR9900856A (pt) | 2000-04-25 |
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