ID22838A - Oksazolidina sebagai antagonis 5-ht2a - Google Patents

Oksazolidina sebagai antagonis 5-ht2a

Info

Publication number
ID22838A
ID22838A IDW990813D ID990813D ID22838A ID 22838 A ID22838 A ID 22838A ID W990813 D IDW990813 D ID W990813D ID 990813 D ID990813 D ID 990813D ID 22838 A ID22838 A ID 22838A
Authority
ID
Indonesia
Prior art keywords
oksazolidina
ht2a antagonists
ht2a
antagonists
Prior art date
Application number
IDW990813D
Other languages
English (en)
Inventor
Henning Bottcher
Helmut Prucher
Helmut Greiner
Gerd Bartoszyk
Christoph Seyfried
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of ID22838A publication Critical patent/ID22838A/id

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D413/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/10Drugs for genital or sexual disorders; Contraceptives for impotence
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/18Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/20Hypnotics; Sedatives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/22Anxiolytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/30Drugs for disorders of the nervous system for treating abuse or dependence
    • A61P25/36Opioid-abuse
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/04Anorexiants; Antiobesity agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
IDW990813D 1997-02-26 1998-02-06 Oksazolidina sebagai antagonis 5-ht2a ID22838A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19707628A DE19707628A1 (de) 1997-02-26 1997-02-26 Oxazolidinone

Publications (1)

Publication Number Publication Date
ID22838A true ID22838A (id) 1999-12-09

Family

ID=7821498

Family Applications (1)

Application Number Title Priority Date Filing Date
IDW990813D ID22838A (id) 1997-02-26 1998-02-06 Oksazolidina sebagai antagonis 5-ht2a

Country Status (25)

Country Link
US (1) US6462056B1 (id)
EP (1) EP0964863B1 (id)
JP (2) JP4402175B2 (id)
KR (1) KR20000075697A (id)
CN (1) CN1177847C (id)
AR (1) AR010899A1 (id)
AT (1) ATE240954T1 (id)
AU (1) AU739251B2 (id)
BR (1) BR9807765A (id)
CA (1) CA2281918C (id)
CZ (1) CZ299199A3 (id)
DE (2) DE19707628A1 (id)
DK (1) DK0964863T3 (id)
ES (1) ES2197466T3 (id)
HU (1) HUP0001093A3 (id)
ID (1) ID22838A (id)
NO (1) NO313415B1 (id)
PL (1) PL335100A1 (id)
PT (1) PT964863E (id)
RU (1) RU2196140C2 (id)
SK (1) SK112799A3 (id)
TW (1) TW531538B (id)
UA (1) UA58542C2 (id)
WO (1) WO1998038189A1 (id)
ZA (1) ZA981579B (id)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2787328A1 (fr) 1998-12-22 2000-06-23 Sanofi Sa Utilisation d'un antagoniste des recepteurs 5ht2a pour la preparation de medicaments utiles dans le traitement des ronflements et du syndrome de haute resistance ou de resistance des voies aeriennes superieures
CA2360683A1 (en) * 1999-01-28 2000-08-03 Joseph P. Yevich Antidepressant heterocyclic compounds
ES2165274B1 (es) 1999-06-04 2003-04-01 Almirall Prodesfarma Sa Nuevos derivados de indolilpiperidina como agentes antihistaminicos y antialergicos.
AU5567000A (en) * 1999-06-24 2001-01-09 Toray Industries, Inc. Alpha1b-adrenergic receptor antagonists
GB9928568D0 (en) 1999-12-03 2000-02-02 Zeneca Ltd Chemical compounds
GB0009803D0 (en) * 2000-04-25 2000-06-07 Astrazeneca Ab Chemical compounds
ES2172436B1 (es) 2000-10-31 2004-01-16 Almirall Prodesfarma Sa Derivados de indolilpiperidina como agentes antihistaminicos y antialergicos.
DE60212959T2 (de) * 2001-04-07 2007-02-15 Astrazeneca Ab Eine sulfonimid-gruppe enthaltende oxazolidinone als antibiotika
WO2004069828A1 (ja) * 2003-02-04 2004-08-19 Mitsubishi Pharma Corporation ピペリジン化合物およびその医薬用途
CA2548917C (en) 2003-12-11 2014-09-23 Sepracor Inc. Combination of a sedative and a neurotransmitter modulator, and methods for improving sleep quality and treating depression
CL2008001002A1 (es) * 2007-04-11 2008-10-17 Actelion Pharmaceuticals Ltd Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana.
BRPI0820985A2 (pt) * 2007-12-18 2015-06-16 Actelion Pharmaceuticals Ltd Composto derivado de 5-aminociclometil-oxazondin-2-ona, medicamento e composição farmacêutica que os contém e uso dos mesmos
WO2010041218A2 (en) * 2008-10-10 2010-04-15 Actelion Pharmaceuticals Ltd Oxazolidinyl antibiotics
WO2014046544A1 (en) 2012-09-21 2014-03-27 Aapa B.V. Substituted 3-heteroaryloxy-3-(hetero)aryl-propylamines as serotonin transporter and serotonin ht2c receptor modulators

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3723797A1 (de) 1987-07-18 1989-01-26 Merck Patent Gmbh Oxazolidinone
DE4005371A1 (de) * 1990-02-21 1991-08-22 Merck Patent Gmbh Oxazolidinone
DE4017211A1 (de) * 1990-05-29 1991-12-05 Merck Patent Gmbh Oxazolidinone
DK152090D0 (da) * 1990-06-22 1990-06-22 Lundbaek A S H Piperidylsubstituerede indolderivater
DK158590D0 (da) * 1990-07-02 1990-07-02 Lundbeck & Co As H Indolderivater
DE4324393A1 (de) 1993-07-21 1995-01-26 Merck Patent Gmbh 4-Aryloxy- und 4-Arylthiopiperidinderivate
DE4414113A1 (de) * 1994-04-22 1995-10-26 Merck Patent Gmbh 3-Indolylpiperidine
ZA954689B (en) * 1994-06-08 1996-01-29 Lundbeck & Co As H 4-Aryl-1-(indanmethyl dihydrobenzofuranmethyl or dihydrobenzothiophenemethyl) piperidines tetrahydropyridines or piperazines
DE19500689A1 (de) 1995-01-12 1996-07-18 Merck Patent Gmbh Indolpiperidin-Derivate

Also Published As

Publication number Publication date
NO994106L (no) 1999-10-19
JP2001513764A (ja) 2001-09-04
TW531538B (en) 2003-05-11
US6462056B1 (en) 2002-10-08
JP2009256363A (ja) 2009-11-05
PT964863E (pt) 2003-10-31
DE59808461D1 (de) 2003-06-26
CZ299199A3 (cs) 1999-11-17
EP0964863A1 (de) 1999-12-22
NO994106D0 (no) 1999-08-25
ATE240954T1 (de) 2003-06-15
AR010899A1 (es) 2000-07-12
ES2197466T3 (es) 2004-01-01
ZA981579B (en) 1999-03-17
HUP0001093A3 (en) 2001-07-30
CN1177847C (zh) 2004-12-01
PL335100A1 (en) 2000-04-10
CA2281918C (en) 2007-04-03
WO1998038189A1 (de) 1998-09-03
HUP0001093A2 (hu) 2001-06-28
EP0964863B1 (de) 2003-05-21
AU739251B2 (en) 2001-10-04
DK0964863T3 (da) 2003-08-04
JP4402175B2 (ja) 2010-01-20
KR20000075697A (ko) 2000-12-26
UA58542C2 (uk) 2003-08-15
NO313415B1 (no) 2002-09-30
CN1248973A (zh) 2000-03-29
CA2281918A1 (en) 1998-09-03
AU6394998A (en) 1998-09-18
BR9807765A (pt) 2000-02-22
DE19707628A1 (de) 1998-08-27
SK112799A3 (en) 2000-06-12
RU2196140C2 (ru) 2003-01-10

Similar Documents

Publication Publication Date Title
ID18003A (id) Antagonis muskarinik
ID19623A (id) Antagonis reseptor vitronektin
ID16742A (id) Antagonis reseptor endotelin
EE200000171A (et) Uued NPY antagonistid
ATE255098T1 (de) Substituierte chromanderivate
ID26223A (id) Antagonis reseptor vitronektin
ID22838A (id) Oksazolidina sebagai antagonis 5-ht2a
ATE255099T1 (de) Substituierte chromanderivate
ID26665A (id) Antagonis vla-4
NO993460D0 (no) Paroxetine-preparater
ID27845A (id) Turunan tetrahidrokuilina sebagai antagonis glisilina
ID24468A (id) 2-asilaminopropanamina sebagai antagonis reseptor tachykinin
ID28811A (id) Antagonis reseptor vitronektin
PT969815E (pt) Composicoes farmaceuticas
EP0986553A4 (en) DIHYDROPYRIMIDONE DERIVATIVES AS NPY ANTAGONISTS
PT964867E (pt) Antagonistas da taquicinima
ID23054A (id) Turunan-turunan piperazino sebagai antagonis neurokinin
EE200000330A (et) Farmatseutilised kompositsioonid
ATE378327T1 (de) Substituierte cyclobutylaminderivate
ID24309A (id) 2-asilaminopropanamina sebagai antagonis reseptor tachykinin
ID26508A (id) Oksim-oksim tersubstitusi sebagai antagonis-antagonis neurokinin
DE29719467U1 (de) Abrollbock
ID22978A (id) Antagonis reseptor endotelin
NO994436D0 (no) Farmasöytiske sammensetninger
DE29722763U1 (de) Tischkonstruktion