HUP9901820A3 - 4-amino pyrimidine derivatives, medicaments containing these compounds, their use and process for their production - Google Patents

4-amino pyrimidine derivatives, medicaments containing these compounds, their use and process for their production

Info

Publication number
HUP9901820A3
HUP9901820A3 HU9901820A HUP9901820A HUP9901820A3 HU P9901820 A3 HUP9901820 A3 HU P9901820A3 HU 9901820 A HU9901820 A HU 9901820A HU P9901820 A HUP9901820 A HU P9901820A HU P9901820 A3 HUP9901820 A3 HU P9901820A3
Authority
HU
Hungary
Prior art keywords
compounds
production
pyrimidine derivatives
medicaments containing
amino pyrimidine
Prior art date
Application number
HU9901820A
Other languages
English (en)
Hungarian (hu)
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE1996108631 external-priority patent/DE19608631A1/de
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of HUP9901820A2 publication Critical patent/HUP9901820A2/hu
Publication of HUP9901820A3 publication Critical patent/HUP9901820A3/hu

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Immunology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
HU9901820A 1996-03-06 1997-03-03 4-amino pyrimidine derivatives, medicaments containing these compounds, their use and process for their production HUP9901820A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE1996108631 DE19608631A1 (de) 1996-03-06 1996-03-06 4-Amino-pyrimidin-Derivate, diese Verbindungen enthaltende Arnzeimittel, deren Verwendung und Verfahren zu ihrer Herstellung
DE19629652A DE19629652A1 (de) 1996-03-06 1996-07-23 4-Amino-pyrimidin-Derivate, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung

Publications (2)

Publication Number Publication Date
HUP9901820A2 HUP9901820A2 (hu) 1999-09-28
HUP9901820A3 true HUP9901820A3 (en) 2001-10-29

Family

ID=26023531

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9901820A HUP9901820A3 (en) 1996-03-06 1997-03-03 4-amino pyrimidine derivatives, medicaments containing these compounds, their use and process for their production

Country Status (19)

Country Link
EP (1) EP0885226A1 (pt)
JP (1) JP2000506847A (pt)
KR (1) KR19990087550A (pt)
CN (1) CN1212695A (pt)
AU (1) AU710274B2 (pt)
BG (1) BG102708A (pt)
BR (1) BR9708312A (pt)
CA (1) CA2243994A1 (pt)
CZ (1) CZ281798A3 (pt)
DE (1) DE19629652A1 (pt)
EE (1) EE9800277A (pt)
HU (1) HUP9901820A3 (pt)
IL (1) IL125404A0 (pt)
NO (1) NO984084L (pt)
NZ (1) NZ331546A (pt)
PL (1) PL328771A1 (pt)
SK (1) SK120598A3 (pt)
TR (1) TR199801749T2 (pt)
WO (1) WO1997032881A1 (pt)

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EP0885198B1 (en) 1996-03-05 2001-12-19 AstraZeneca AB 4-anilinoquinazoline derivatives
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ES2306306T3 (es) 1999-11-05 2008-11-01 Astrazeneca Ab Nuevos derivados de quinazolina.
BRPI0411608A (pt) 2003-06-24 2006-08-08 Neurosearch As derivado de 8-aza-biciclo [3.2.1] octano, composição farmacêutica, uso do composto, e, método de tratamento, prevenção ou alìvio de uma doença, um distúrbio ou uma condição de um organismo animal vivo
CN101189238A (zh) * 2005-02-16 2008-05-28 先灵公司 具有cxcr3拮抗剂活性的哌嗪-哌啶
CA2742986C (en) 2008-11-07 2015-03-31 Triact Therapeutics, Inc. Use of catecholic butane derivatives in cancer therapy
CA2745041C (en) * 2008-12-01 2017-08-22 Kai Schiemann 2, 5-diamino-substituted pyrido [4, 3-d] pyrimidines as autotaxin inhibitors against cancer
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US8465912B2 (en) 2009-02-27 2013-06-18 OSI Pharmaceuticals, LLC Methods for the identification of agents that inhibit mesenchymal-like tumor cells or their formation
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Family Cites Families (2)

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Publication number Priority date Publication date Assignee Title
IL112249A (en) * 1994-01-25 2001-11-25 Warner Lambert Co Pharmaceutical compositions containing di and tricyclic pyrimidine derivatives for inhibiting tyrosine kinases of the epidermal growth factor receptor family and some new such compounds
DE4431867A1 (de) * 1994-09-07 1996-03-14 Thomae Gmbh Dr K Pyrimido[5,4-d]pyrimidine, diese Verbindungen enthaltende Arzneimittel, deren Verwendung und Verfahren zu ihrer Herstellung

Also Published As

Publication number Publication date
JP2000506847A (ja) 2000-06-06
CA2243994A1 (en) 1997-09-12
BG102708A (en) 1999-09-30
IL125404A0 (en) 1999-03-12
EE9800277A (et) 1999-02-15
BR9708312A (pt) 1999-08-03
NO984084D0 (no) 1998-09-04
WO1997032881A1 (de) 1997-09-12
DE19629652A1 (de) 1998-01-29
TR199801749T2 (xx) 1998-12-21
NO984084L (no) 1998-09-04
SK120598A3 (en) 1999-06-11
AU710274B2 (en) 1999-09-16
EP0885226A1 (de) 1998-12-23
CZ281798A3 (cs) 1999-02-17
AU1925197A (en) 1997-09-22
CN1212695A (zh) 1999-03-31
NZ331546A (en) 2000-03-27
KR19990087550A (ko) 1999-12-27
PL328771A1 (en) 1999-02-15
HUP9901820A2 (hu) 1999-09-28

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