HUP0202819A2 - Eljárás tiazolszármazékok előállítására és az új intermedierek - Google Patents

Eljárás tiazolszármazékok előállítására és az új intermedierek

Info

Publication number
HUP0202819A2
HUP0202819A2 HU0202819A HUP0202819A HUP0202819A2 HU P0202819 A2 HUP0202819 A2 HU P0202819A2 HU 0202819 A HU0202819 A HU 0202819A HU P0202819 A HUP0202819 A HU P0202819A HU P0202819 A2 HUP0202819 A2 HU P0202819A2
Authority
HU
Hungary
Prior art keywords
hydroxymethylthiazole
preparation
reacted
prepare
thiazole derivatives
Prior art date
Application number
HU0202819A
Other languages
English (en)
Inventor
Kevin Coppola
Original Assignee
Syngenta Participations Ag.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Syngenta Participations Ag. filed Critical Syngenta Participations Ag.
Publication of HUP0202819A2 publication Critical patent/HUP0202819A2/hu
Publication of HUP0202819A3 publication Critical patent/HUP0202819A3/hu

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/34—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/40—Unsubstituted amino or imino radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/50—Nitrogen atoms bound to hetero atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)

Abstract

A találmány szerinti eljárás során a (III) képletű vegyület éssavaddíciós sói előállítására 2-klór-5-hidroxi-metil-tiazolt vagy 2-hidroxi-5-hidroxi-metil-tiazolt, vagy 5-hidroxi-metil-tiazol-diazóniumsót sav jelenlétében egy klorid forrással reagáltatják. Az 5-hidroxi-metil-tiazol-diazónium só köztitermék előállítására 2-amino-5-hidroxi-metil-tiazolt vagy savaddíciós sóját sav jelenlétében egy alkálifém-nitrittel reagáltatják. 2-amino-5-hidroxi-metil-tiazol előállításáraaz (A) képletű vegyületet tiokarbamiddal reagáltatják. Ó
HU0202819A 1999-08-10 2000-08-08 Process for the preparation of thiazole derivatives and the new intermediates HUP0202819A3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/371,180 US6265553B1 (en) 1999-08-10 1999-08-10 Intermediate thiazoles and process for the preparation of 2-chloro-5-chloromethyl-thiazole
PCT/EP2000/007709 WO2001010852A1 (en) 1999-08-10 2000-08-08 Process for the preparation of thiazole derivatives

Publications (2)

Publication Number Publication Date
HUP0202819A2 true HUP0202819A2 (hu) 2002-12-28
HUP0202819A3 HUP0202819A3 (en) 2004-03-01

Family

ID=23462834

Family Applications (1)

Application Number Title Priority Date Filing Date
HU0202819A HUP0202819A3 (en) 1999-08-10 2000-08-08 Process for the preparation of thiazole derivatives and the new intermediates

Country Status (19)

Country Link
US (4) US6265553B1 (hu)
EP (1) EP1202979B1 (hu)
JP (1) JP2003506444A (hu)
KR (1) KR20020022796A (hu)
CN (2) CN1169800C (hu)
AR (1) AR030258A1 (hu)
AT (1) ATE294166T1 (hu)
AU (1) AU778367B2 (hu)
BR (1) BR0013235A (hu)
CA (1) CA2380838A1 (hu)
CZ (1) CZ2002483A3 (hu)
DE (1) DE60019763D1 (hu)
ES (1) ES2238029T3 (hu)
HU (1) HUP0202819A3 (hu)
MX (1) MXPA02001246A (hu)
RU (1) RU2002105516A (hu)
TR (2) TR200200304T2 (hu)
WO (1) WO2001010852A1 (hu)
ZA (1) ZA200201110B (hu)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2772017C (en) 2003-08-29 2016-05-31 Mitsui Chemicals, Inc. Agricultural/horticultural insecticide and method for using the same
WO2011101402A1 (en) * 2010-02-17 2011-08-25 Syngenta Participations Ag Isoxazoline derivatives as insecticides
EP2540701B1 (en) * 2010-02-26 2014-10-22 Sumitomo Chemical Co., Ltd Process for production of cyclopropanecarboxylic acid ester compound
CN104039755A (zh) * 2011-09-01 2014-09-10 百奥泰利加控股有限公司 由昆虫病原真菌分离的脂类杀虫剂及其用途
CN106749086B (zh) * 2016-12-27 2019-05-24 江苏振方生物化学有限公司 一种农药中间体2-氯-5-氯甲基噻唑的制备方法
CN111036158A (zh) * 2019-12-28 2020-04-21 邯郸市瑞田农药有限公司 一种2氯-5氯甲基噻唑合成反应系统

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3631538A1 (de) * 1986-09-17 1988-03-24 Bayer Ag Verfahren zur herstellung von 2-chlor-5-chlormethylthiazol
US5811555A (en) * 1995-11-22 1998-09-22 Kureha Chemical Industry Co., Ltd. Method for substitution of an amino group of a primary amine by a chlorine atom and a synthetic method by application thereof
JP2001508452A (ja) * 1997-01-22 2001-06-26 ノバルティス アクチェンゲゼルシャフト チアゾール誘導体の製造方法
US5773625A (en) * 1997-10-02 1998-06-30 Abbott Laboratories Process for the preparation of disubstituted carbonates
US6407251B1 (en) * 2000-12-28 2002-06-18 Takeda Chemical Industries, Ltd. Process for preparing 2-chloro-5-chloromethylthiazole

Also Published As

Publication number Publication date
US20030191321A1 (en) 2003-10-09
DE60019763D1 (de) 2005-06-02
CN1169800C (zh) 2004-10-06
HUP0202819A3 (en) 2004-03-01
ES2238029T3 (es) 2005-08-16
EP1202979B1 (en) 2005-04-27
MXPA02001246A (es) 2002-07-22
US6566530B2 (en) 2003-05-20
WO2001010852A1 (en) 2001-02-15
TR200202474T2 (tr) 2003-01-21
EP1202979A1 (en) 2002-05-08
CN1368966A (zh) 2002-09-11
US6265553B1 (en) 2001-07-24
ZA200201110B (en) 2002-11-27
BR0013235A (pt) 2002-04-23
ATE294166T1 (de) 2005-05-15
CZ2002483A3 (cs) 2002-05-15
JP2003506444A (ja) 2003-02-18
US20030055229A1 (en) 2003-03-20
RU2002105516A (ru) 2003-09-20
CN1626525A (zh) 2005-06-15
AR030258A1 (es) 2003-08-20
US6476230B1 (en) 2002-11-05
AU778367B2 (en) 2004-12-02
CA2380838A1 (en) 2001-02-15
TR200200304T2 (tr) 2002-06-21
KR20020022796A (ko) 2002-03-27
US6710182B2 (en) 2004-03-23
AU6836400A (en) 2001-03-05

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Legal Events

Date Code Title Description
FC4A Lapse of provisional application due to refusal