HUP0202331A2 - Eljárás 5- és/vagy 6-helyzetben szubsztituált 2-hidroxi-benzoesav-észterek előállítására - Google Patents
Eljárás 5- és/vagy 6-helyzetben szubsztituált 2-hidroxi-benzoesav-észterek előállításáraInfo
- Publication number
- HUP0202331A2 HUP0202331A2 HU0202331A HUP0202331A HUP0202331A2 HU P0202331 A2 HUP0202331 A2 HU P0202331A2 HU 0202331 A HU0202331 A HU 0202331A HU P0202331 A HUP0202331 A HU P0202331A HU P0202331 A2 HUP0202331 A2 HU P0202331A2
- Authority
- HU
- Hungary
- Prior art keywords
- general formula
- substituted
- preparation
- acid esters
- hydroxybenzoic acid
- Prior art date
Links
- 238000000034 method Methods 0.000 title abstract 2
- -1 6-substituted-2-hydroxybenzoic acid esters Chemical class 0.000 title 1
- 125000000217 alkyl group Chemical group 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- UFHFLCQGNIYNRP-UHFFFAOYSA-N Hydrogen Chemical compound [H][H] UFHFLCQGNIYNRP-UHFFFAOYSA-N 0.000 abstract 1
- WDJHALXBUFZDSR-UHFFFAOYSA-M acetoacetate Chemical compound CC(=O)CC([O-])=O WDJHALXBUFZDSR-UHFFFAOYSA-M 0.000 abstract 1
- 125000002777 acetyl group Chemical group [H]C([H])([H])C(*)=O 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- RWCCWEUUXYIKHB-UHFFFAOYSA-N benzophenone Chemical compound C=1C=CC=CC=1C(=O)C1=CC=CC=C1 RWCCWEUUXYIKHB-UHFFFAOYSA-N 0.000 abstract 1
- 239000012965 benzophenone Substances 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 125000002485 formyl group Chemical class [H]C(*)=O 0.000 abstract 1
- 239000000417 fungicide Substances 0.000 abstract 1
- 125000005843 halogen group Chemical group 0.000 abstract 1
- 229910052739 hydrogen Inorganic materials 0.000 abstract 1
- 239000001257 hydrogen Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 239000005445 natural material Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000002904 solvent Substances 0.000 abstract 1
- 239000007858 starting material Substances 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C67/00—Preparation of carboxylic acid esters
- C07C67/30—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group
- C07C67/333—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton
- C07C67/343—Preparation of carboxylic acid esters by modifying the acid moiety of the ester, such modification not being an introduction of an ester group by isomerisation; by change of size of the carbon skeleton by increase in the number of carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C45/00—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds
- C07C45/45—Preparation of compounds having >C = O groups bound only to carbon or hydrogen atoms; Preparation of chelates of such compounds by condensation
- C07C45/46—Friedel-Crafts reactions
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
A találmány tárgya egylépéses eljárás az általános képletű vegyületek- ahol R alkilcsoport; R1 és R2 egymástól függetlenül hidrogénatom vagyalkilcsoport; és X halogénatom vagy acetilcsoport - előállítására egyáltalános képletű acetoacetátnak és egy általános képletű aldehidnekegy alkilkarbonsavsó és egy oldószer jelenlétében végzettreakciójával. Az (I) általános képletű vegyületek kiindulási anyagkéntalkalmazhatók természetes anyagok szintézisében és benzofenon gombaölőszerek gyártásában. Ó
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US35403799A | 1999-07-15 | 1999-07-15 | |
| PCT/US2000/018768 WO2001005739A1 (en) | 1999-07-15 | 2000-07-10 | Process for the preparation of 5- and/or 6-substituted-2-hydroxybenzoic acid esters |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| HUP0202331A2 true HUP0202331A2 (hu) | 2002-11-28 |
| HUP0202331A3 HUP0202331A3 (en) | 2005-01-28 |
| HU229906B1 HU229906B1 (en) | 2014-12-29 |
Family
ID=23391634
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| HU0202331A HU229906B1 (en) | 1999-07-15 | 2000-07-10 | Process for the preparation of 5- and/or 6-substituted-2-hydroxybenzoic acid esters |
Country Status (19)
| Country | Link |
|---|---|
| US (1) | US6441219B1 (hu) |
| EP (1) | EP1196370B1 (hu) |
| JP (1) | JP3779615B2 (hu) |
| KR (1) | KR100651090B1 (hu) |
| CN (1) | CN1160304C (hu) |
| AT (1) | ATE249415T1 (hu) |
| AU (1) | AU5926300A (hu) |
| BR (1) | BR0012493B1 (hu) |
| CA (1) | CA2379342C (hu) |
| CZ (1) | CZ300511B6 (hu) |
| DE (1) | DE60005193T2 (hu) |
| DK (1) | DK1196370T3 (hu) |
| ES (1) | ES2207528T3 (hu) |
| HU (1) | HU229906B1 (hu) |
| IL (2) | IL147027A0 (hu) |
| MX (1) | MXPA02000395A (hu) |
| RU (1) | RU2245325C2 (hu) |
| SK (1) | SK286835B6 (hu) |
| WO (1) | WO2001005739A1 (hu) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6559336B2 (en) * | 1999-07-15 | 2003-05-06 | Basf Aktiengesellschaft | Process for the preparation of 5- and/or 6-substituted-2-hydroxybenzoic acid esters |
| DE60034254T2 (de) * | 2000-12-23 | 2007-12-20 | Basf Ag | Verfahren zur herstellung von 5- und/oder 6-substituierten 2-hydroxybenzoesäureestern |
| BR112014017780A8 (pt) | 2012-01-18 | 2017-07-11 | Zafgen Inc | Compostos de sulfona tricíclicos e métodos para fazer e usar os mesmos |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2107958C3 (de) | 1971-02-19 | 1980-08-21 | Basf Ag, 6700 Ludwigshafen | Verfahren zur Herstellung von a -Naphtholen |
| US5773663A (en) * | 1996-05-01 | 1998-06-30 | American Cyanamid Company | Fungicidal methods, compounds and compositions containing benzophenones |
| US5945567A (en) | 1997-08-20 | 1999-08-31 | American Cyanamid Company | Fungicidal 2-methoxybenzophenones |
-
2000
- 2000-07-10 CA CA002379342A patent/CA2379342C/en not_active Expired - Fee Related
- 2000-07-10 DK DK00945295T patent/DK1196370T3/da active
- 2000-07-10 WO PCT/US2000/018768 patent/WO2001005739A1/en active IP Right Grant
- 2000-07-10 HU HU0202331A patent/HU229906B1/hu not_active IP Right Cessation
- 2000-07-10 AT AT00945295T patent/ATE249415T1/de active
- 2000-07-10 IL IL14702700A patent/IL147027A0/xx active IP Right Grant
- 2000-07-10 DE DE60005193T patent/DE60005193T2/de not_active Expired - Lifetime
- 2000-07-10 BR BRPI0012493-1A patent/BR0012493B1/pt not_active IP Right Cessation
- 2000-07-10 JP JP2001511400A patent/JP3779615B2/ja not_active Expired - Fee Related
- 2000-07-10 AU AU59263/00A patent/AU5926300A/en not_active Abandoned
- 2000-07-10 EP EP00945295A patent/EP1196370B1/en not_active Expired - Lifetime
- 2000-07-10 RU RU2002102233/04A patent/RU2245325C2/ru not_active IP Right Cessation
- 2000-07-10 CZ CZ20020112A patent/CZ300511B6/cs not_active IP Right Cessation
- 2000-07-10 KR KR1020027000513A patent/KR100651090B1/ko not_active IP Right Cessation
- 2000-07-10 SK SK68-2002A patent/SK286835B6/sk not_active IP Right Cessation
- 2000-07-10 ES ES00945295T patent/ES2207528T3/es not_active Expired - Lifetime
- 2000-07-10 CN CNB008101779A patent/CN1160304C/zh not_active Expired - Lifetime
- 2000-07-10 MX MXPA02000395A patent/MXPA02000395A/es active IP Right Grant
- 2000-10-30 US US09/699,775 patent/US6441219B1/en not_active Expired - Lifetime
-
2001
- 2001-12-11 IL IL147027A patent/IL147027A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| DE60005193T2 (de) | 2004-07-01 |
| HUP0202331A3 (en) | 2005-01-28 |
| CZ2002112A3 (cs) | 2002-05-15 |
| US6441219B1 (en) | 2002-08-27 |
| SK286835B6 (sk) | 2009-06-05 |
| KR100651090B1 (ko) | 2006-11-29 |
| JP2003505355A (ja) | 2003-02-12 |
| BR0012493B1 (pt) | 2011-02-22 |
| ES2207528T3 (es) | 2004-06-01 |
| AU5926300A (en) | 2001-02-05 |
| CN1160304C (zh) | 2004-08-04 |
| CN1360564A (zh) | 2002-07-24 |
| HU229906B1 (en) | 2014-12-29 |
| SK682002A3 (en) | 2002-08-06 |
| WO2001005739A1 (en) | 2001-01-25 |
| IL147027A (en) | 2006-12-31 |
| MXPA02000395A (es) | 2002-07-02 |
| EP1196370B1 (en) | 2003-09-10 |
| CA2379342C (en) | 2007-01-02 |
| EP1196370A1 (en) | 2002-04-17 |
| DE60005193D1 (de) | 2003-10-16 |
| BR0012493A (pt) | 2002-04-02 |
| IL147027A0 (en) | 2002-08-14 |
| CA2379342A1 (en) | 2001-01-25 |
| KR20020012629A (ko) | 2002-02-16 |
| DK1196370T3 (da) | 2004-01-12 |
| ATE249415T1 (de) | 2003-09-15 |
| RU2245325C2 (ru) | 2005-01-27 |
| CZ300511B6 (cs) | 2009-06-03 |
| JP3779615B2 (ja) | 2006-05-31 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MM4A | Lapse of definitive patent protection due to non-payment of fees |