NO20010559L - Fremgangsmate for syntese av (1H)-benzo[c]kinolizin-3-ones derivater - Google Patents

Fremgangsmate for syntese av (1H)-benzo[c]kinolizin-3-ones derivater

Info

Publication number
NO20010559L
NO20010559L NO20010559A NO20010559A NO20010559L NO 20010559 L NO20010559 L NO 20010559L NO 20010559 A NO20010559 A NO 20010559A NO 20010559 A NO20010559 A NO 20010559A NO 20010559 L NO20010559 L NO 20010559L
Authority
NO
Norway
Prior art keywords
quinolizin
benzo
synthesis
ones derivatives
compounds
Prior art date
Application number
NO20010559A
Other languages
English (en)
Other versions
NO20010559D0 (no
Inventor
Antonio Guarna
Mario Serio
Ernesto Giovanni Occhiato
Original Assignee
Serono Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Serono Lab filed Critical Serono Lab
Publication of NO20010559D0 publication Critical patent/NO20010559D0/no
Publication of NO20010559L publication Critical patent/NO20010559L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D455/00Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
    • C07D455/03Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
    • C07D455/04Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing a quinolizine ring system condensed with only one six-membered carbocyclic ring, e.g. julolidine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/10Anti-acne agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/14Drugs for dermatological disorders for baldness or alopecia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Inorganic Compounds Of Heavy Metals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Carbon And Carbon Compounds (AREA)
NO20010559A 1998-08-03 2001-02-01 Fremgangsmate for syntese av (1H)-benzo[c]kinolizin-3-ones derivater NO20010559L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP98114524 1998-08-03
PCT/EP1999/005277 WO2000008019A1 (en) 1998-08-03 1999-07-23 Process for the synthesis of (1h)-benzo[c]quinolizin-3-ones derivatives

Publications (2)

Publication Number Publication Date
NO20010559D0 NO20010559D0 (no) 2001-02-01
NO20010559L true NO20010559L (no) 2001-02-01

Family

ID=8232396

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20010559A NO20010559L (no) 1998-08-03 2001-02-01 Fremgangsmate for syntese av (1H)-benzo[c]kinolizin-3-ones derivater

Country Status (29)

Country Link
US (1) US6723850B1 (no)
EP (1) EP1102765B1 (no)
JP (1) JP2002522435A (no)
KR (1) KR100624239B1 (no)
CN (1) CN1128148C (no)
AT (1) ATE250057T1 (no)
AU (1) AU751873B2 (no)
BG (1) BG65062B1 (no)
BR (1) BR9912870A (no)
CA (1) CA2338498C (no)
CZ (1) CZ291648B6 (no)
DE (1) DE69911430T2 (no)
DK (1) DK1102765T3 (no)
EA (1) EA003997B1 (no)
EE (1) EE04642B1 (no)
ES (1) ES2203169T3 (no)
HK (1) HK1037368A1 (no)
HU (1) HUP0103241A3 (no)
IL (2) IL141212A0 (no)
NO (1) NO20010559L (no)
NZ (1) NZ509243A (no)
PL (1) PL198963B1 (no)
PT (1) PT1102765E (no)
SI (1) SI1102765T1 (no)
SK (1) SK285438B6 (no)
TR (1) TR200100286T2 (no)
UA (1) UA67787C2 (no)
WO (1) WO2000008019A1 (no)
ZA (1) ZA200100365B (no)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20100074949A1 (en) 2008-08-13 2010-03-25 William Rowe Pharmaceutical composition and administration thereof
CN101006076B (zh) * 2004-06-24 2010-09-29 沃泰克斯药物股份有限公司 Atp-结合弹夹转运蛋白的调控剂
US8354427B2 (en) * 2004-06-24 2013-01-15 Vertex Pharmaceutical Incorporated Modulators of ATP-binding cassette transporters
JP2009521468A (ja) * 2005-12-24 2009-06-04 バーテックス ファーマシューティカルズ インコーポレイテッド Abc輸送体の調節因子としてのキノリン−4−オン誘導体
JP5409010B2 (ja) 2005-12-28 2014-02-05 バーテックス ファーマシューティカルズ インコーポレイテッド N−[2,4−ビス(1,1−ジメチルエチル)−5−ヒドロキシフェニル]−1,4−ジヒドロ−4−オキソキノリン−3−カルボキサミドの固体形態
EP2821400B1 (en) 2009-03-20 2017-09-27 Vertex Pharmaceuticals Incorporated Process for making modulators of cystic fibrosis transmembrane conductance regulator
US8802700B2 (en) 2010-12-10 2014-08-12 Vertex Pharmaceuticals Incorporated Modulators of ATP-Binding Cassette transporters
EP2651890B1 (en) * 2010-12-14 2014-09-10 Syngenta Participations AG Strigolactam derivatives and their use as plant growth regulators
MX2014010253A (es) 2012-02-27 2014-11-12 Vertex Pharma Composicion farmaceutica y administraciones de la misma.
WO2016057730A1 (en) 2014-10-07 2016-04-14 Strohmeier Mark Co-crystals of modulators of cystic fibrosis transmembrane conductance regulator
CN105001216B (zh) * 2015-07-08 2017-03-01 中国科学院兰州化学物理研究所 一种喹嗪酮的制备方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5064961A (en) * 1989-12-18 1991-11-12 E. R. Squibb & Sons, Inc. Process for preparing an optically active cyclobutane nucleoside
FR2696465B1 (fr) * 1992-10-02 1994-12-23 Adir Nouveaux dérivés d'ellipticine, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent.
IT1286545B1 (it) 1996-02-09 1998-07-15 Antonio Guarna Derivati benzo(c) chinolizinici,loro preparazione ed uso come inibitori delle 5-alfa-riduttasi
JPH09316076A (ja) * 1996-05-24 1997-12-09 Nippon Paper Ind Co Ltd 9−置換プリン誘導体及びその抗ウイルス剤としての用途

Also Published As

Publication number Publication date
CA2338498C (en) 2009-05-19
EP1102765B1 (en) 2003-09-17
BR9912870A (pt) 2001-10-16
IL141212A0 (en) 2002-03-10
NO20010559D0 (no) 2001-02-01
PL345802A1 (en) 2002-01-02
EE04642B1 (et) 2006-06-15
DE69911430D1 (de) 2003-10-23
JP2002522435A (ja) 2002-07-23
DK1102765T3 (da) 2004-02-02
EA200100213A1 (ru) 2001-08-27
SK285438B6 (sk) 2007-01-04
AU6312399A (en) 2000-02-28
KR100624239B1 (ko) 2006-09-13
EE200100060A (et) 2002-06-17
EP1102765A1 (en) 2001-05-30
HUP0103241A3 (en) 2002-10-28
SI1102765T1 (en) 2003-12-31
CZ2001434A3 (cs) 2001-08-15
WO2000008019A1 (en) 2000-02-17
ES2203169T3 (es) 2004-04-01
TR200100286T2 (tr) 2001-07-23
PT1102765E (pt) 2003-12-31
KR20010074684A (ko) 2001-08-09
CZ291648B6 (cs) 2003-04-16
UA67787C2 (uk) 2004-07-15
PL198963B1 (pl) 2008-08-29
NZ509243A (en) 2002-11-26
HUP0103241A2 (hu) 2002-01-28
CN1311788A (zh) 2001-09-05
BG65062B1 (bg) 2007-01-31
BG105198A (en) 2001-12-29
ATE250057T1 (de) 2003-10-15
HK1037368A1 (en) 2002-02-08
US6723850B1 (en) 2004-04-20
SK1672001A3 (en) 2001-08-06
ZA200100365B (en) 2001-07-26
EA003997B1 (ru) 2003-12-25
CN1128148C (zh) 2003-11-19
AU751873B2 (en) 2002-08-29
CA2338498A1 (en) 2000-02-17
DE69911430T2 (de) 2004-07-22
IL141212A (en) 2006-12-31

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Representative=s name: ONSAGERS AS, POSTBOKS 6963 ST OLAVS PLASS, 0130 OS

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