EE200100060A - (1H)benso[c]kinolisiin-3-ooni derivaatide sünteesi meetod - Google Patents
(1H)benso[c]kinolisiin-3-ooni derivaatide sünteesi meetodInfo
- Publication number
- EE200100060A EE200100060A EEP200100060A EEP200100060A EE200100060A EE 200100060 A EE200100060 A EE 200100060A EE P200100060 A EEP200100060 A EE P200100060A EE P200100060 A EEP200100060 A EE P200100060A EE 200100060 A EE200100060 A EE 200100060A
- Authority
- EE
- Estonia
- Prior art keywords
- quinolizin
- benzo
- derivatives
- synthesis
- compounds
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D455/00—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
- C07D455/03—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine
- C07D455/04—Heterocyclic compounds containing quinolizine ring systems, e.g. emetine alkaloids, protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing quinolizine ring systems directly condensed with at least one six-membered carbocyclic ring, e.g. protoberberine; Alkylenedioxy derivatives of dibenzo [a, g] quinolizines, e.g. berberine containing a quinolizine ring system condensed with only one six-membered carbocyclic ring, e.g. julolidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/10—Anti-acne agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/14—Drugs for dermatological disorders for baldness or alopecia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Inorganic Compounds Of Heavy Metals (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Carbon And Carbon Compounds (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP98114524 | 1998-08-03 | ||
PCT/EP1999/005277 WO2000008019A1 (en) | 1998-08-03 | 1999-07-23 | Process for the synthesis of (1h)-benzo[c]quinolizin-3-ones derivatives |
Publications (2)
Publication Number | Publication Date |
---|---|
EE200100060A true EE200100060A (et) | 2002-06-17 |
EE04642B1 EE04642B1 (et) | 2006-06-15 |
Family
ID=8232396
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
EEP200100060A EE04642B1 (et) | 1998-08-03 | 1999-07-23 | (1H)benso[c]kinolisiin-3-ooni derivaatide sünteesi meetod |
Country Status (29)
Country | Link |
---|---|
US (1) | US6723850B1 (et) |
EP (1) | EP1102765B1 (et) |
JP (1) | JP2002522435A (et) |
KR (1) | KR100624239B1 (et) |
CN (1) | CN1128148C (et) |
AT (1) | ATE250057T1 (et) |
AU (1) | AU751873B2 (et) |
BG (1) | BG65062B1 (et) |
BR (1) | BR9912870A (et) |
CA (1) | CA2338498C (et) |
CZ (1) | CZ291648B6 (et) |
DE (1) | DE69911430T2 (et) |
DK (1) | DK1102765T3 (et) |
EA (1) | EA003997B1 (et) |
EE (1) | EE04642B1 (et) |
ES (1) | ES2203169T3 (et) |
HK (1) | HK1037368A1 (et) |
HU (1) | HUP0103241A3 (et) |
IL (2) | IL141212A0 (et) |
NO (1) | NO20010559L (et) |
NZ (1) | NZ509243A (et) |
PL (1) | PL198963B1 (et) |
PT (1) | PT1102765E (et) |
SI (1) | SI1102765T1 (et) |
SK (1) | SK285438B6 (et) |
TR (1) | TR200100286T2 (et) |
UA (1) | UA67787C2 (et) |
WO (1) | WO2000008019A1 (et) |
ZA (1) | ZA200100365B (et) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20100074949A1 (en) | 2008-08-13 | 2010-03-25 | William Rowe | Pharmaceutical composition and administration thereof |
BR122018075478B8 (pt) * | 2004-06-24 | 2023-10-31 | Vertex Pharma | moduladores de transportadores de cassete de ligação de atp |
US8354427B2 (en) | 2004-06-24 | 2013-01-15 | Vertex Pharmaceutical Incorporated | Modulators of ATP-binding cassette transporters |
US20090105272A1 (en) * | 2005-12-24 | 2009-04-23 | Grootenhuis Peter D J | Prodrugs of modulators of ABC transporters |
HUE049976T2 (hu) | 2005-12-28 | 2020-11-30 | Vertex Pharma | N-[2,4-bisz(1,1-dimetil-etil)-5-hidroxi-fenil]-1,4-dihidro-4-oxo-kinolin-3-karboxamid amorf alakjának gyógyászati kompozíciói |
SG10201504084QA (en) | 2009-03-20 | 2015-06-29 | Vertex Pharma | Process for making modulators of cystic fibrosis transmembrane conductance regulator |
US8802700B2 (en) | 2010-12-10 | 2014-08-12 | Vertex Pharmaceuticals Incorporated | Modulators of ATP-Binding Cassette transporters |
MX2013006497A (es) * | 2010-12-14 | 2013-06-28 | Syngenta Participations Ag | Derivados de estrigolactama y su uso como reguladores del crecimiento de plantas. |
CN109966264A (zh) | 2012-02-27 | 2019-07-05 | 沃泰克斯药物股份有限公司 | 药物组合物及其施用 |
CN107250113B (zh) | 2014-10-07 | 2019-03-29 | 弗特克斯药品有限公司 | 囊性纤维化跨膜传导调节蛋白的调节剂的共晶 |
CN105001216B (zh) * | 2015-07-08 | 2017-03-01 | 中国科学院兰州化学物理研究所 | 一种喹嗪酮的制备方法 |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5064961A (en) * | 1989-12-18 | 1991-11-12 | E. R. Squibb & Sons, Inc. | Process for preparing an optically active cyclobutane nucleoside |
FR2696465B1 (fr) * | 1992-10-02 | 1994-12-23 | Adir | Nouveaux dérivés d'ellipticine, leur procédé de préparation et les compositions pharmaceutiques qui les contiennent. |
IT1286545B1 (it) * | 1996-02-09 | 1998-07-15 | Antonio Guarna | Derivati benzo(c) chinolizinici,loro preparazione ed uso come inibitori delle 5-alfa-riduttasi |
JPH09316076A (ja) * | 1996-05-24 | 1997-12-09 | Nippon Paper Ind Co Ltd | 9−置換プリン誘導体及びその抗ウイルス剤としての用途 |
-
1999
- 1999-07-23 TR TR2001/00286T patent/TR200100286T2/xx unknown
- 1999-07-23 AT AT99941269T patent/ATE250057T1/de not_active IP Right Cessation
- 1999-07-23 UA UA2001020777A patent/UA67787C2/uk unknown
- 1999-07-23 DK DK99941269T patent/DK1102765T3/da active
- 1999-07-23 SI SI9930419T patent/SI1102765T1/xx unknown
- 1999-07-23 US US09/743,373 patent/US6723850B1/en not_active Expired - Fee Related
- 1999-07-23 CZ CZ2001434A patent/CZ291648B6/cs not_active IP Right Cessation
- 1999-07-23 PL PL345802A patent/PL198963B1/pl not_active IP Right Cessation
- 1999-07-23 NZ NZ509243A patent/NZ509243A/xx not_active IP Right Cessation
- 1999-07-23 CA CA002338498A patent/CA2338498C/en not_active Expired - Fee Related
- 1999-07-23 JP JP2000563652A patent/JP2002522435A/ja active Pending
- 1999-07-23 IL IL14121299A patent/IL141212A0/xx active IP Right Grant
- 1999-07-23 KR KR1020017000325A patent/KR100624239B1/ko not_active IP Right Cessation
- 1999-07-23 CN CN99809204A patent/CN1128148C/zh not_active Expired - Fee Related
- 1999-07-23 ES ES99941269T patent/ES2203169T3/es not_active Expired - Lifetime
- 1999-07-23 AU AU63123/99A patent/AU751873B2/en not_active Ceased
- 1999-07-23 EA EA200100213A patent/EA003997B1/ru not_active IP Right Cessation
- 1999-07-23 SK SK167-2001A patent/SK285438B6/sk not_active IP Right Cessation
- 1999-07-23 BR BR9912870-5A patent/BR9912870A/pt not_active Application Discontinuation
- 1999-07-23 HU HU0103241A patent/HUP0103241A3/hu unknown
- 1999-07-23 PT PT99941269T patent/PT1102765E/pt unknown
- 1999-07-23 DE DE69911430T patent/DE69911430T2/de not_active Expired - Fee Related
- 1999-07-23 WO PCT/EP1999/005277 patent/WO2000008019A1/en active IP Right Grant
- 1999-07-23 EE EEP200100060A patent/EE04642B1/et not_active IP Right Cessation
- 1999-07-23 EP EP99941269A patent/EP1102765B1/en not_active Expired - Lifetime
-
2001
- 2001-01-12 ZA ZA200100365A patent/ZA200100365B/en unknown
- 2001-01-30 BG BG105198A patent/BG65062B1/bg unknown
- 2001-02-01 IL IL141212A patent/IL141212A/en not_active IP Right Cessation
- 2001-02-01 NO NO20010559A patent/NO20010559L/no not_active Application Discontinuation
- 2001-11-20 HK HK01108153A patent/HK1037368A1/xx not_active IP Right Cessation
Also Published As
Similar Documents
Publication | Publication Date | Title |
---|---|---|
MX9707706A (es) | Compuestos intermediarios novedosos y proceso para la manufactura de derivados de la camptotecina (cpt-11) y compuestos relacionados. | |
DE69709938D1 (de) | N-benzylpiperidin- und tetrahydropyridin-derivate | |
NO20061793L (no) | 1,4-disubstituerte isoquinilonderlvater som RAF-kinaseinhibitorer nyttige for behandling av proliferative sykdommer | |
EA200000358A1 (ru) | Способ получения диарилпиридинов, полезных в качестве ингибиторов cox-2 | |
EE04642B1 (et) | (1H)benso[c]kinolisiin-3-ooni derivaatide sünteesi meetod | |
WO2001090097A3 (en) | Novel compounds having antiinflammatory activity: process for their preparation and pharmaceutical compositions containing them | |
ZA200404752B (en) | 6-aminomorphinane derivatives method for the production and use thereof | |
TNSN06167A1 (en) | Method for producing (3-oxo-2,3-dihydro-1h-isoindol-1-yl) acetylguanidine derivatives | |
NO20052197L (no) | Fremgangsmate for fremstilling av pyrazol | |
WO2006013049A3 (en) | Benzyloxy derivatives as maob inhibitors | |
MXPA05006587A (es) | Compuestos de tiazol como derivados de antagonistas del receptor de la integrina. | |
DE60009945D1 (de) | Beta-d-thioxylos-derivate, verfahren zur herstellung und verwendung als arzneimittel | |
WO2002008227A3 (en) | Bicyclic hydantoin derivatives and combinatorial libraries thereof | |
DE60335960D1 (de) | 1,2,4-triazolderivat, verfahren zu dessenherstellung, und dieses enthaltende pharmazeutische zusammensetzung | |
FR2784682B1 (fr) | Nouveaux derives 2-halogene de 5-0-desosaminylerythronolide a, leur procede de preparation et leur application comme medicaments | |
DE60006125D1 (de) | Herstellung von 2-(2-arylmorpholin-2-yl)ethanolderivaten und zwischenprodukte | |
DE60329721D1 (de) | Regiospezifische synthese von nikotinderivaten | |
NO20020561L (no) | Fremgangsmåte for fremstilling av syrer via alfa-klorepoksi- estere | |
FR2835835B1 (fr) | Nouveaux derives de la pyridazine, leur utilisation comme medicaments, compositions pharmaceutiques et leur procede de preparation | |
AU1392600A (en) | Alkyl esters of 3-(3,4-dihalogenophenyl)-2,6-dioxopiperidine-3-propionic acid useful as intermediates | |
MXPA03003466A (es) | Derivados de piranosido. | |
DE50107619D1 (de) | Verfahren zur herstellung von 4-brom-anilin-derivaten | |
CY1115291T1 (el) | Ινδολη, αζαϊνδολη και σχετικα ετεροκυκλικα αμιδια 4-αλκενυλ πιπεριδινης | |
EE200200465A (et) | Asendatud 8,8a-dihüdro-3aH-indeno[1,2-d]tiasoolid, nende valmistamismeetod ja kasutamine ravimitena | |
NO20014530L (no) | Fremgangsmåte for fremstilling av 4, 4-dimetyl-3<beta>- hydroksy-pregna-8, 14-dien-21-karboksylsyreestere ogmellomprodukter ved fremgangsmåten |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
KB4A | Valid patent at the end of a year |
Effective date: 20061231 |
|
GB1A | Change in the ownership or in the address of the owner | ||
KB4A | Valid patent at the end of a year |
Effective date: 20071231 |
|
KB4A | Valid patent at the end of a year |
Effective date: 20081231 |
|
KB4A | Valid patent at the end of a year |
Effective date: 20101231 |
|
MM4A | Lapsed by not paying the annual fees |
Effective date: 20100723 |