KR920004353A - 4,5,6,7-테트라하이드로-3-아릴-인다졸, 그의 제조방법 및 제초제로의 용도 - Google Patents

4,5,6,7-테트라하이드로-3-아릴-인다졸, 그의 제조방법 및 제초제로의 용도 Download PDF

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KR920004353A
KR920004353A KR1019910013458A KR910013458A KR920004353A KR 920004353 A KR920004353 A KR 920004353A KR 1019910013458 A KR1019910013458 A KR 1019910013458A KR 910013458 A KR910013458 A KR 910013458A KR 920004353 A KR920004353 A KR 920004353A
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alkyl
compound
phenyl
formula
alkoxy
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KR1019910013458A
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슐쯔 라이너
바우어 클라우스
비어링거 헤르만
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마이어,라피체
훽스트 아크티엔게젤샤프트
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Publication of KR920004353A publication Critical patent/KR920004353A/ko

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
    • C07D231/06—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/28—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N<
    • A01N47/38—Ureas or thioureas containing the groups >N—CO—N< or >N—CS—N< containing the group >N—CO—N< where at least one nitrogen atom is part of a heterocyclic ring; Thio analogues thereof
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/56—1,2-Diazoles; Hydrogenated 1,2-diazoles
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/16—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof the nitrogen atom being part of a heterocyclic ring
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N47/00—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid
    • A01N47/08—Biocides, pest repellants or attractants, or plant growth regulators containing organic compounds containing a carbon atom not being member of a ring and having no bond to a carbon or hydrogen atom, e.g. derivatives of carbonic acid the carbon atom having one or more single bonds to nitrogen atoms
    • A01N47/10—Carbamic acid derivatives, i.e. containing the group —O—CO—N<; Thio analogues thereof
    • A01N47/22—O-Aryl or S-Aryl esters thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
    • C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
    • C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles

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  • Life Sciences & Earth Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Dentistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Plant Pathology (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

내용 없음

Description

4,5,6,7-테트라하이드로-3-아릴-인다졸, 그의 제조방법 및 제초제로의 용도
본 내용은 요부공개 건이므로 전문내용을 수록하지 않았음

Claims (9)

  1. 하기 일반식(Ⅰ) 또는 (Ⅰ')화합물:
    상기 식에서 X는 산소 또는 황원자이고, R1은 H,C1-C6알킬, C2-C6은 알케닐, C2-C6알키닐, C1-C6할로알킬,(C1-C4-알콕시)-C1-C4알킬, (C1-C6-알콕시)카보닐,아릴톡시카보닐, (C1-C6-알킬)아미노카보닐, 아릴 아미노카보닐, 페닐, 치환된 페닐 또는 아실이고, R2는 펜리 또는 치환된 페닐이고, R3는 서로 독립적으로 또는 아실이고, R2는 페닐 또는 치환된 페닐이고, R3는 서로 독립적으로H또는 C1-C5알킬이고, n은 0 내지 6의 정수이다.
  2. 제1항에 있어서, R1이 H, C1-C4-알킬, C2-C4알케닐, C2-C4알키닐, C1-C4할로알킬, (C1-C2-알콕시)-C1-C4-알킬, (C1-C4-알콕시)카보닐, (C1-C4-알킬)아미노카보닐, 페닐록시카보닐, 페닐아미노카보닐, 페닐(여기에서, 페닐록시카보닐, 페닐아미노카보닐 및 페닐 그룹은 각각의 경우 페닐 고리에서 비치환되거나 또는 할로겐, C1-C4-알킬, C1-C4할로알킬, C1-C4알콕시, C1-C4할로알콕시, 니트로, 카복실 및 카복실의 산 유도체를 포함하는 그룹으로부터 선택된 하나 이상의 라디칼로 치환된다)이거나 또는 아실인 화합물.
  3. 제1항 또는 제2항에 있어서, R2가 치환되지 않거나 또는 할로겐, 니트로 C1-C4-알킬, C1-C4-할로알킬 및 C1-C4-알킬설포닐을 포함하는 그룹중에서 선택된 1 내지 3개의 라디칼로 치환된 페닐인 화합물.
  4. 제1항 내지 제3항중 어느 한 항에 있어서, R3라디칼이 서로 독립적으로 바람직하게 H또는 메틸이고, n이 0 내지 4의 정수인 화합물.
  5. 제1항 내지 제4항중 어느 한 항에 있어서, 상기 정의한 일반식(Ⅰ)을 갖는 화합물.
  6. 염기의 존재하에서 a)하기 일반식(Ⅱ)의 화합물을 하기 일반식(Ⅲ)의 하이드라진 유도체와 반응시키거나, 또는 b)R1이 알킬인 일반식(Ⅰ)또는 (Ⅰ')의 화합물을 제조하는 경우, R1이 수소원자인 언급한 일반식(Ⅰ)또는 (Ⅰ')화합물을 적합한 알킬화제와 반응시키거나, 또는 c)일반식(Ⅰ')의 화합물을 제조하는 경우를 제외하고, 하기 일반식(Ⅳ)의 사이클로헥산-1,3-디온을 하기 일반식(Ⅴ)의 클로로하이드라존과 반응시켜 언급한 일반식(Ⅰ)의 화합물을 수득함을 포함하는, 제1항에서, 정의한 바와같은 일반식(Ⅰ)또는(Ⅰ')화합물의 제조방법 :
    상기 식에서, X는 산소 또는 황원자이고, R1은 H, C1-C6-알킬, C2-C6-알케닐,C2-C6알키닐, C1-C6할로알킬, (C1-C4-알콕시)-C1-C4알킬, (C1-C6-알콕시)카보닐,아릴톡시카보닐, (C1-C6-알킬)아미노카보닐, 아릴아미노카보닐, 페닐. 치환된 페닐 또는 아실이고, R2는 페닐 또는 치환된 페닐이고, R3는 서로 독립적으로 H또는 C1-C5알킬이고, n은 0 내지 6의 정수이다.
  7. 제1항 내지 제5항중 어느 한 항에 청구된 일반식(Ⅰ)또는(Ⅰ')의 화합물과 통상적이 제형화 보조제를 함유하는 제초제.
  8. 제1항 내지 제5항중 어느 한 항에 청구된 일반식(Ⅰ)또는 (Ⅰ')의 화합물의 제초제로의 용도.
  9. 제1항 내지 제5항중 어느 한 항에 정의된 화합물 효과량을 식물, 식물의 종자, 또는 재배 지역에 적용함을 포함하는, 유해 식물을 선택적으로 방제하는 방법.
    ※ 참고사항 : 최초출원 내용에 의하여 공개하는 것임.
KR1019910013458A 1990-08-04 1991-08-03 4,5,6,7-테트라하이드로-3-아릴-인다졸, 그의 제조방법 및 제초제로의 용도 KR920004353A (ko)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DEP4024862.3 1990-08-04
DE4024862A DE4024862A1 (de) 1990-08-04 1990-08-04 4,5,6,7-tetrahydro-3-aryl-indazole, verfahren zu ihrer herstellung und ihre verwendung als herbizide

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KR920004353A true KR920004353A (ko) 1992-03-27

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US (1) US5104442A (ko)
EP (1) EP0470489A1 (ko)
JP (1) JPH04234368A (ko)
KR (1) KR920004353A (ko)
DE (1) DE4024862A1 (ko)
IE (1) IE912770A1 (ko)
PT (1) PT98549A (ko)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5444038A (en) * 1992-03-09 1995-08-22 Zeneca Limited Arylindazoles and their use as herbicides
DE4232544A1 (de) * 1992-09-29 1994-03-31 Thomae Gmbh Dr K Arzneimittel enthaltend 1,5,6,7-Tetrahydro-4H-indazol-4-one, neue 1,5,6,7-Tetrahydro-4H-indazol-4-one und Verfahren zu ihrer Herstellung
CA2156652A1 (en) * 1994-08-31 1996-03-01 Minoru Takano Epoxyphenol derivatives and herbicides containing them as active ingredients
US5939324A (en) * 1997-12-02 1999-08-17 The United States Of America As Represented By The United States Department Of Energy Performance evaluation soil samples utilizing encapsulation technology
US6545033B1 (en) 1999-10-06 2003-04-08 3-Dimensional Pharmaceuticals, Inc. Fused 1-(2,6-dichloro-4-trifluoromethylphenyl)-pyrazoles, the synthesis thereof and the use thereof as pesticides
TWI382015B (zh) * 2005-02-25 2013-01-11 Serenex Inc 苯、吡啶及噠嗪衍生物
US20070185184A1 (en) * 2005-09-16 2007-08-09 Serenex, Inc. Carbazole derivatives
WO2007101156A1 (en) * 2006-02-27 2007-09-07 Serenex, Inc. Cyclohexylamino, benzene, pyridine, and pyridazine derivatives
EP2391627B1 (en) 2009-01-28 2013-12-25 Cara Therapeutics, Inc. Bicyclic pyrazolo-heterocycles
US7741350B1 (en) * 2009-01-28 2010-06-22 Cara Therapeutics, Inc. Bicyclic pyrazolo-heterocycles
CN107428740A (zh) 2014-09-11 2017-12-01 埃萨内克斯股份有限公司 吲唑基‑和吲哚基‑苯甲酰胺衍生物

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4059434A (en) * 1975-10-15 1977-11-22 E. I. Du Pont De Nemours And Company Cycloalkanapyrazole herbicides
PH18938A (en) * 1982-09-28 1985-11-11 Sumitomo Chemical Co 2-substituted phenyl-4,5,6,7-tetrahydro-2h-indazoles and their use
GR80558B (en) * 1983-10-08 1985-02-06 Nippon Kayaku Kk Derivative of pyrazole and use thereof as a herbicide

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PT98549A (pt) 1993-11-30
DE4024862A1 (de) 1992-02-13
JPH04234368A (ja) 1992-08-24
IE912770A1 (en) 1992-02-12
US5104442A (en) 1992-04-14
EP0470489A1 (de) 1992-02-12

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