HRP20190919T1 - Derivati n1-acil- 5-fluoropirimidinona - Google Patents

Derivati n1-acil- 5-fluoropirimidinona Download PDF

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Publication number
HRP20190919T1
HRP20190919T1 HRP20190919TT HRP20190919T HRP20190919T1 HR P20190919 T1 HRP20190919 T1 HR P20190919T1 HR P20190919T T HRP20190919T T HR P20190919TT HR P20190919 T HRP20190919 T HR P20190919T HR P20190919 T1 HRP20190919 T1 HR P20190919T1
Authority
HR
Croatia
Prior art keywords
alkyl
benzyl
optionally substituted
phenyl
compound
Prior art date
Application number
HRP20190919TT
Other languages
English (en)
Croatian (hr)
Inventor
Timothy Boebel
Kristy Bryan
Beth Lorsbach
Timothy Martin
W. Owen
Mark Pobanz
Scott Thornburgh
Jeffery Webster
Chenglin Yao
Original Assignee
Adama Makhteshim Ltd.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=43535292&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HRP20190919(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Adama Makhteshim Ltd. filed Critical Adama Makhteshim Ltd.
Publication of HRP20190919T1 publication Critical patent/HRP20190919T1/hr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
    • C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Dentistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
HRP20190919TT 2009-08-07 2010-08-05 Derivati n1-acil- 5-fluoropirimidinona HRP20190919T1 (hr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US23222309P 2009-08-07 2009-08-07
EP10807171.3A EP2519512B1 (en) 2009-08-07 2010-08-05 N1-acyl- 5-fluoropyrimidinone derivatives
PCT/US2010/044576 WO2011017538A1 (en) 2009-08-07 2010-08-05 N1-acyl-5-fluoropyrimidinone derivatives

Publications (1)

Publication Number Publication Date
HRP20190919T1 true HRP20190919T1 (hr) 2019-09-20

Family

ID=43535292

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20190919TT HRP20190919T1 (hr) 2009-08-07 2010-08-05 Derivati n1-acil- 5-fluoropirimidinona

Country Status (33)

Country Link
US (1) US8470839B2 (cg-RX-API-DMAC10.html)
EP (1) EP2519512B1 (cg-RX-API-DMAC10.html)
JP (1) JP5748754B2 (cg-RX-API-DMAC10.html)
KR (1) KR101792285B1 (cg-RX-API-DMAC10.html)
CN (1) CN102548981B (cg-RX-API-DMAC10.html)
AU (1) AU2010279402B2 (cg-RX-API-DMAC10.html)
BR (1) BR112012002810B1 (cg-RX-API-DMAC10.html)
CA (1) CA2768510C (cg-RX-API-DMAC10.html)
CL (1) CL2012000316A1 (cg-RX-API-DMAC10.html)
CO (1) CO6491117A2 (cg-RX-API-DMAC10.html)
CR (1) CR20120030A (cg-RX-API-DMAC10.html)
CY (1) CY1122115T1 (cg-RX-API-DMAC10.html)
DK (1) DK2519512T3 (cg-RX-API-DMAC10.html)
EA (1) EA023411B1 (cg-RX-API-DMAC10.html)
EC (1) ECSP12011653A (cg-RX-API-DMAC10.html)
ES (1) ES2728966T3 (cg-RX-API-DMAC10.html)
HN (1) HN2012000269A (cg-RX-API-DMAC10.html)
HR (1) HRP20190919T1 (cg-RX-API-DMAC10.html)
HU (1) HUE045290T2 (cg-RX-API-DMAC10.html)
IL (1) IL217952A (cg-RX-API-DMAC10.html)
IN (1) IN2012DN00539A (cg-RX-API-DMAC10.html)
LT (1) LT2519512T (cg-RX-API-DMAC10.html)
MX (1) MX2012001620A (cg-RX-API-DMAC10.html)
NI (1) NI201200022A (cg-RX-API-DMAC10.html)
NZ (1) NZ597570A (cg-RX-API-DMAC10.html)
PE (1) PE20120688A1 (cg-RX-API-DMAC10.html)
PL (1) PL2519512T3 (cg-RX-API-DMAC10.html)
PT (1) PT2519512T (cg-RX-API-DMAC10.html)
SI (1) SI2519512T1 (cg-RX-API-DMAC10.html)
TR (1) TR201908180T4 (cg-RX-API-DMAC10.html)
UA (1) UA106889C2 (cg-RX-API-DMAC10.html)
WO (1) WO2011017538A1 (cg-RX-API-DMAC10.html)
ZA (1) ZA201200819B (cg-RX-API-DMAC10.html)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PE20120691A1 (es) * 2009-08-07 2012-06-08 Dow Agrosciences Llc Derivados de n1-sulfonil-5-fluoropirimidinona
US8658660B2 (en) 2011-08-17 2014-02-25 Dow Agrosciences, Llc. 5-fluoro-4-imino-3,4-dihydropyrimidin-2-(1H)-ones derivatives
EP2938194B1 (en) 2012-12-28 2019-11-27 Adama Makhteshim Ltd. N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxylate derivatives
US9321734B2 (en) 2012-12-28 2016-04-26 Dow Agrosciences Llc N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxamide derivatives
CN104994859B (zh) * 2012-12-28 2018-10-26 阿达玛马克西姆股份有限公司 1-(取代的苯甲酰基)-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2(1h)-酮衍生物
RU2644014C2 (ru) 2012-12-31 2018-02-07 Адама Мактешим Лтд. Производные 3-алкил-5-фтор-4-замещенного-имино-3,4-дигидропиримидин-2(н)-она в качестве фунгицидов
WO2015103261A1 (en) 2013-12-31 2015-07-09 Dow Agrosciences Llc Synergistic fungicidal mixtures for fungal control in cereals
UA122200C2 (uk) 2013-12-31 2020-10-12 Адама Махтешім Лтд. 5-фтор-4-іміно-3-(алкіл/заміщений алкіл)-1-(арилсульфоніл)-3,4-дигідропіримідин-2(1h)-он і способи його одержання
JP6734267B2 (ja) 2014-09-26 2020-08-05 ザ ケマーズ カンパニー エフシー リミテッド ライアビリティ カンパニー イソシアネート由来のオルガノシラン
EP3655396A1 (en) 2017-07-17 2020-05-27 Adama Makhteshim Ltd. Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one
EA202191250A1 (ru) 2018-11-05 2021-08-20 Адама Мактешим Лтд. Смеси и композиции, включающие 5-фтор-4-имино-3-метил-1-тозил-3,4-дигидропиримидин-2-он, и способы их применения
TWI808347B (zh) 2019-09-23 2023-07-11 以色列商亞當馬赫特希姆有限公司 用於製備5-氟-4-亞胺基-3-甲基-1-甲苯磺醯基-3,4-二氫嘧啶-2(1h)-酮及該化合物的衍生物之方法

Family Cites Families (22)

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Publication number Priority date Publication date Assignee Title
CH421973A (de) * 1962-05-01 1966-10-15 Hoffmann La Roche Verfahren zur Herstellung eines Cytosin-Derivates
US3309359A (en) 1965-10-22 1967-03-14 Hoffmann La Roche N-mono-acyl-5-fluorocytosine derivatives and process
US3368938A (en) * 1966-01-13 1968-02-13 Hoffmann La Roche Controlling fungi with 5-fluorocytosine
US3868373A (en) 1970-01-27 1975-02-25 Hoffmann La Roche 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines
CH579057A5 (cg-RX-API-DMAC10.html) 1973-09-07 1976-08-31 Hoffmann La Roche
FR2530636A1 (fr) 1982-07-23 1984-01-27 Rhone Poulenc Agrochimie Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides
GR80171B (en) 1983-08-29 1985-01-02 Ciba Geigy Ag N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use
US4845081A (en) 1984-10-18 1989-07-04 University Of Florida Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes
EP0332579B1 (de) 1988-03-09 1994-08-10 Ciba-Geigy Ag Mittel zum Schutz von Pflanzen gegen Krankheiten
DE3821711A1 (de) 1988-06-28 1990-02-08 Bayer Ag Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel
JP3217191B2 (ja) 1992-07-16 2001-10-09 ビーエーエスエフ アクチェンゲゼルシャフト ヘテロ芳香族化合物およびこれを含有する植物保護剤
EP0836602B1 (en) 1995-07-05 2002-01-30 E.I. Du Pont De Nemours And Company Fungicidal pyrimidinones
EA001148B1 (ru) * 1996-03-11 2000-10-30 Новартис Аг Производные пиримидин-4-она
HRP970239B1 (en) 1997-05-09 2004-04-30 Inst Ru Er Bouekovic Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity
GT199900185A (es) 1998-11-06 2001-04-18 Novedosa pirimidin-4-enamina como fungicida.
WO2003018051A1 (en) 2001-08-27 2003-03-06 Vic Jira Anti-fungal composition
JPWO2005095419A1 (ja) 2004-04-01 2008-02-21 武田薬品工業株式会社 チアゾロピリミジン誘導体
WO2008005303A2 (en) 2006-06-30 2008-01-10 Janssen Pharmaceutica N.V. Thiazolopyrimidine modulators of trpv1
RU2522430C2 (ru) 2008-01-22 2014-07-10 ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи 5-фторпиримидиновые производные в качестве фунгицидов
ES2456272T3 (es) 2008-08-01 2014-04-21 Dow Agrosciences Llc Uso de 5-fluorocitosina como un fungicida
CA2750413C (en) 2009-01-23 2016-06-21 Northlake Biosciences Llc Hydroxamic acid derivatives
PE20120691A1 (es) 2009-08-07 2012-06-08 Dow Agrosciences Llc Derivados de n1-sulfonil-5-fluoropirimidinona

Also Published As

Publication number Publication date
WO2011017538A1 (en) 2011-02-10
BR112012002810B1 (pt) 2018-12-11
UA106889C2 (uk) 2014-10-27
IL217952A0 (en) 2012-03-29
EA201270253A1 (ru) 2012-07-30
IN2012DN00539A (cg-RX-API-DMAC10.html) 2015-06-12
CN102548981A (zh) 2012-07-04
LT2519512T (lt) 2019-07-25
PT2519512T (pt) 2019-06-04
IL217952A (en) 2017-11-30
HK1172894A1 (en) 2013-05-03
NZ597570A (en) 2014-04-30
AU2010279402B2 (en) 2015-04-16
ZA201200819B (en) 2013-05-29
HN2012000269A (es) 2015-04-27
JP2013501723A (ja) 2013-01-17
CO6491117A2 (es) 2012-07-31
BR112012002810A2 (pt) 2015-09-15
CL2012000316A1 (es) 2014-06-27
CN102548981B (zh) 2015-05-13
EA023411B1 (ru) 2016-06-30
KR20120041786A (ko) 2012-05-02
US20110034490A1 (en) 2011-02-10
CA2768510A1 (en) 2011-02-10
SI2519512T1 (sl) 2019-09-30
US8470839B2 (en) 2013-06-25
PE20120688A1 (es) 2012-06-06
NI201200022A (es) 2012-05-22
EP2519512B1 (en) 2019-03-20
AU2010279402A1 (en) 2012-02-02
ECSP12011653A (es) 2012-03-30
HUE045290T2 (hu) 2019-12-30
DK2519512T3 (da) 2019-05-27
CR20120030A (es) 2012-03-28
PL2519512T3 (pl) 2019-09-30
EP2519512A4 (en) 2013-01-16
CY1122115T1 (el) 2020-11-25
MX2012001620A (es) 2012-04-11
ES2728966T3 (es) 2019-10-29
EP2519512A1 (en) 2012-11-07
JP5748754B2 (ja) 2015-07-15
CA2768510C (en) 2018-05-15
TR201908180T4 (tr) 2019-06-21
KR101792285B1 (ko) 2017-10-31

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