CO6491117A2 - Derivados de n1-acil-5-fluoropirimidinona - Google Patents
Derivados de n1-acil-5-fluoropirimidinonaInfo
- Publication number
- CO6491117A2 CO6491117A2 CO12019954A CO12019954A CO6491117A2 CO 6491117 A2 CO6491117 A2 CO 6491117A2 CO 12019954 A CO12019954 A CO 12019954A CO 12019954 A CO12019954 A CO 12019954A CO 6491117 A2 CO6491117 A2 CO 6491117A2
- Authority
- CO
- Colombia
- Prior art keywords
- compounds
- formulations
- formula
- present description
- fluoropirimidinona
- Prior art date
Links
- 238000009472 formulation Methods 0.000 abstract 4
- 239000000203 mixture Substances 0.000 abstract 4
- 150000001875 compounds Chemical class 0.000 abstract 3
- 241000235349 Ascomycota Species 0.000 abstract 1
- 241000221198 Basidiomycota Species 0.000 abstract 1
- 241000233654 Oomycetes Species 0.000 abstract 1
- 239000003905 agrochemical Substances 0.000 abstract 1
- 239000000417 fungicide Substances 0.000 abstract 1
- 239000007788 liquid Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000843 powder Substances 0.000 abstract 1
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
- C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
- A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Agronomy & Crop Science (AREA)
- Pest Control & Pesticides (AREA)
- Plant Pathology (AREA)
- Health & Medical Sciences (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US23222309P | 2009-08-07 | 2009-08-07 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CO6491117A2 true CO6491117A2 (es) | 2012-07-31 |
Family
ID=43535292
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CO12019954A CO6491117A2 (es) | 2009-08-07 | 2012-02-06 | Derivados de n1-acil-5-fluoropirimidinona |
Country Status (33)
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| PE20120691A1 (es) * | 2009-08-07 | 2012-06-08 | Dow Agrosciences Llc | Derivados de n1-sulfonil-5-fluoropirimidinona |
| US8658660B2 (en) | 2011-08-17 | 2014-02-25 | Dow Agrosciences, Llc. | 5-fluoro-4-imino-3,4-dihydropyrimidin-2-(1H)-ones derivatives |
| EP2938194B1 (en) | 2012-12-28 | 2019-11-27 | Adama Makhteshim Ltd. | N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxylate derivatives |
| US9321734B2 (en) | 2012-12-28 | 2016-04-26 | Dow Agrosciences Llc | N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1(2H)-carboxamide derivatives |
| CN104994859B (zh) * | 2012-12-28 | 2018-10-26 | 阿达玛马克西姆股份有限公司 | 1-(取代的苯甲酰基)-5-氟-4-亚氨基-3-甲基-3,4-二氢嘧啶-2(1h)-酮衍生物 |
| RU2644014C2 (ru) | 2012-12-31 | 2018-02-07 | Адама Мактешим Лтд. | Производные 3-алкил-5-фтор-4-замещенного-имино-3,4-дигидропиримидин-2(н)-она в качестве фунгицидов |
| WO2015103261A1 (en) | 2013-12-31 | 2015-07-09 | Dow Agrosciences Llc | Synergistic fungicidal mixtures for fungal control in cereals |
| UA122200C2 (uk) | 2013-12-31 | 2020-10-12 | Адама Махтешім Лтд. | 5-фтор-4-іміно-3-(алкіл/заміщений алкіл)-1-(арилсульфоніл)-3,4-дигідропіримідин-2(1h)-он і способи його одержання |
| JP6734267B2 (ja) | 2014-09-26 | 2020-08-05 | ザ ケマーズ カンパニー エフシー リミテッド ライアビリティ カンパニー | イソシアネート由来のオルガノシラン |
| EP3655396A1 (en) | 2017-07-17 | 2020-05-27 | Adama Makhteshim Ltd. | Polymorphs of 5-fluoro-4-imino-3-methyl-1-tosyl-3,4-dihydropyrimidin-2-one |
| EA202191250A1 (ru) | 2018-11-05 | 2021-08-20 | Адама Мактешим Лтд. | Смеси и композиции, включающие 5-фтор-4-имино-3-метил-1-тозил-3,4-дигидропиримидин-2-он, и способы их применения |
| TWI808347B (zh) | 2019-09-23 | 2023-07-11 | 以色列商亞當馬赫特希姆有限公司 | 用於製備5-氟-4-亞胺基-3-甲基-1-甲苯磺醯基-3,4-二氫嘧啶-2(1h)-酮及該化合物的衍生物之方法 |
Family Cites Families (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH421973A (de) * | 1962-05-01 | 1966-10-15 | Hoffmann La Roche | Verfahren zur Herstellung eines Cytosin-Derivates |
| US3309359A (en) | 1965-10-22 | 1967-03-14 | Hoffmann La Roche | N-mono-acyl-5-fluorocytosine derivatives and process |
| US3368938A (en) * | 1966-01-13 | 1968-02-13 | Hoffmann La Roche | Controlling fungi with 5-fluorocytosine |
| US3868373A (en) | 1970-01-27 | 1975-02-25 | Hoffmann La Roche | 4-Amino-5-fluoro-2-tri(lower alkyl) silyloxypyrimidines |
| CH579057A5 (cg-RX-API-DMAC10.html) | 1973-09-07 | 1976-08-31 | Hoffmann La Roche | |
| FR2530636A1 (fr) | 1982-07-23 | 1984-01-27 | Rhone Poulenc Agrochimie | Nouveaux derives de la tetrahydro-2,3,6,7 5h-thiazolo (3,2-a) pyrimidine, leur preparation et leur utilisation comme herbicides |
| GR80171B (en) | 1983-08-29 | 1985-01-02 | Ciba Geigy Ag | N-(2-nitrophenyl)-4-aminopyrimidine derivatives process for the preparation thereof and use |
| US4845081A (en) | 1984-10-18 | 1989-07-04 | University Of Florida | Aminomethyl derivatives of biologically active substances, and enhanced delivery thereof across topical membranes |
| EP0332579B1 (de) | 1988-03-09 | 1994-08-10 | Ciba-Geigy Ag | Mittel zum Schutz von Pflanzen gegen Krankheiten |
| DE3821711A1 (de) | 1988-06-28 | 1990-02-08 | Bayer Ag | Thiazolopyrimidin-derivate, verfahren zu ihrer herstellung und ihre verwendung als schaedlingsbekaempfungsmittel |
| JP3217191B2 (ja) | 1992-07-16 | 2001-10-09 | ビーエーエスエフ アクチェンゲゼルシャフト | ヘテロ芳香族化合物およびこれを含有する植物保護剤 |
| EP0836602B1 (en) | 1995-07-05 | 2002-01-30 | E.I. Du Pont De Nemours And Company | Fungicidal pyrimidinones |
| EA001148B1 (ru) * | 1996-03-11 | 2000-10-30 | Новартис Аг | Производные пиримидин-4-она |
| HRP970239B1 (en) | 1997-05-09 | 2004-04-30 | Inst Ru Er Bouekovic | Process for the preparation of sulfonyl-pyrimidine derivatives with antitumor activity |
| GT199900185A (es) | 1998-11-06 | 2001-04-18 | Novedosa pirimidin-4-enamina como fungicida. | |
| WO2003018051A1 (en) | 2001-08-27 | 2003-03-06 | Vic Jira | Anti-fungal composition |
| JPWO2005095419A1 (ja) | 2004-04-01 | 2008-02-21 | 武田薬品工業株式会社 | チアゾロピリミジン誘導体 |
| WO2008005303A2 (en) | 2006-06-30 | 2008-01-10 | Janssen Pharmaceutica N.V. | Thiazolopyrimidine modulators of trpv1 |
| RU2522430C2 (ru) | 2008-01-22 | 2014-07-10 | ДАУ АГРОСАЙЕНСИЗ ЭлЭлСи | 5-фторпиримидиновые производные в качестве фунгицидов |
| ES2456272T3 (es) | 2008-08-01 | 2014-04-21 | Dow Agrosciences Llc | Uso de 5-fluorocitosina como un fungicida |
| CA2750413C (en) | 2009-01-23 | 2016-06-21 | Northlake Biosciences Llc | Hydroxamic acid derivatives |
| PE20120691A1 (es) | 2009-08-07 | 2012-06-08 | Dow Agrosciences Llc | Derivados de n1-sulfonil-5-fluoropirimidinona |
-
2010
- 2010-05-08 UA UAA201202731A patent/UA106889C2/uk unknown
- 2010-08-05 HR HRP20190919TT patent/HRP20190919T1/hr unknown
- 2010-08-05 KR KR1020127005927A patent/KR101792285B1/ko not_active Expired - Fee Related
- 2010-08-05 NZ NZ597570A patent/NZ597570A/en unknown
- 2010-08-05 TR TR2019/08180T patent/TR201908180T4/tr unknown
- 2010-08-05 WO PCT/US2010/044576 patent/WO2011017538A1/en not_active Ceased
- 2010-08-05 PE PE2012000169A patent/PE20120688A1/es not_active Application Discontinuation
- 2010-08-05 JP JP2012523950A patent/JP5748754B2/ja active Active
- 2010-08-05 HU HUE10807171A patent/HUE045290T2/hu unknown
- 2010-08-05 SI SI201031893T patent/SI2519512T1/sl unknown
- 2010-08-05 ES ES10807171T patent/ES2728966T3/es active Active
- 2010-08-05 DK DK10807171.3T patent/DK2519512T3/da active
- 2010-08-05 CN CN201080045370.7A patent/CN102548981B/zh active Active
- 2010-08-05 PL PL10807171T patent/PL2519512T3/pl unknown
- 2010-08-05 AU AU2010279402A patent/AU2010279402B2/en not_active Ceased
- 2010-08-05 EP EP10807171.3A patent/EP2519512B1/en active Active
- 2010-08-05 LT LTEP10807171.3T patent/LT2519512T/lt unknown
- 2010-08-05 MX MX2012001620A patent/MX2012001620A/es active IP Right Grant
- 2010-08-05 CA CA2768510A patent/CA2768510C/en not_active Expired - Fee Related
- 2010-08-05 US US12/851,236 patent/US8470839B2/en active Active - Reinstated
- 2010-08-05 EA EA201270253A patent/EA023411B1/ru not_active IP Right Cessation
- 2010-08-05 PT PT10807171T patent/PT2519512T/pt unknown
- 2010-08-05 IN IN539DEN2012 patent/IN2012DN00539A/en unknown
- 2010-08-05 BR BR112012002810-3A patent/BR112012002810B1/pt active IP Right Grant
-
2012
- 2012-01-18 CR CR20120030A patent/CR20120030A/es unknown
- 2012-02-02 HN HN2012000269A patent/HN2012000269A/es unknown
- 2012-02-02 ZA ZA2012/00819A patent/ZA201200819B/en unknown
- 2012-02-03 NI NI201200022A patent/NI201200022A/es unknown
- 2012-02-05 IL IL217952A patent/IL217952A/en active IP Right Grant
- 2012-02-06 CO CO12019954A patent/CO6491117A2/es active IP Right Grant
- 2012-02-06 CL CL2012000316A patent/CL2012000316A1/es unknown
- 2012-02-07 EC ECSP12011653 patent/ECSP12011653A/es unknown
-
2019
- 2019-06-06 CY CY20191100603T patent/CY1122115T1/el unknown
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CO6491117A2 (es) | Derivados de n1-acil-5-fluoropirimidinona | |
| ECSP15032846A (es) | Derivados de n-(sustituido)-5-fluoro-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2h)-carboximida | |
| MX381341B (es) | Derivados de 3-alquil-5-fluoro-4-sustituido-imino-3,4-dihidropirimidin-2(1h)-ona como fungicidas. | |
| SV2017005461A (es) | Benzamidas sustituidas con 1,3-tiazol-2-ilo | |
| ECSP15032926A (es) | Derivados de 1-(benzoílo-sustituido)-5-fluoro-4-imino-3-metil-3,4-dihidropirimidin-2(1h)-ona | |
| MX357150B (es) | Composicion de acaros que comprende un acaro depredador y una presa inmovilizada que se pone pone en contacto con un agente reductor de hongos y metodos y usos relacionados con el uso de dicha composicion. | |
| CL2012002896A1 (es) | Compuestos para tratamiento de enfermedades asociadas con proteinas amiloides o tipo amiloide; composicion farmacéutica que lo comprende; uso del compuesto para retener o incrementar la memoria cognitiva. | |
| GT201200334A (es) | Morfolinopirimidinas y su uso en terapia | |
| BR112012024822B8 (pt) | Composto, uso de um composto e composição farmacêutica | |
| CL2014002087A1 (es) | Composición veterinaria masticable que comprende como agente activo un compuesto derivado de isoxazolina; y su uso para el tratamiento y/o prevención de una infestación y/o infección por parásitos en un animal. | |
| CR20110059A (es) | Compuestos organicos | |
| UY35040A (es) | Pirrolopirimidinilamino-benzotiazolonas sustituidas | |
| CL2013001009A1 (es) | Compuestos heterociclicos fusionados; composicion farmaceutica que los comprende, y uso en el tratamiento de un trastorno proliferativo tal como cancer. | |
| CL2011002930A1 (es) | Compuestos derivados de 8-oxo-9-[3-(1h-bencimidazol-2-iloxi)-fenil]-4,5,6,7,8,9-hexahidro-2h-pirrolo[3,4-b]quinolina-3-carboxilato de etilo; procedimiento de preparacion; composicion farmaceutica que lo comprende; compuestos intermediarios; y uso del compuesto como inhibidor selectivo de quinasas aurora a y b para tratar el cancer. | |
| AR088622A1 (es) | 18-METIL-6,7-METILEN-3-OXO-17-PREGN-4-EN-21,17b-CARBOLACTONA, PREPARADOS FARMACEUTICOS QUE CONTIENEN LOS COMPUESTOS MENCIONADOS Y SU USO EN LA TERAPIA DE LA ENDOMETRIOSIS | |
| ECSP15032859A (es) | Derivados de n-(sustituido)-5-fluoro-4-imino-3-metil-2-oxo-3,4-dihidropirimidin-1(2h)-carboxilato | |
| DOP2015000170A (es) | Compuestos químicos | |
| MY172413A (en) | Fungicide formulations for soft pvc | |
| CR20150314A (es) | Pirimido-[4,5-b]-quinolina-4,5 (3h, 10h)-dionas como supresoras de mutación sin sentido | |
| CL2013000735A1 (es) | Uso de una composicion que comprende compuestos derivados de 1-h-imidazol-4-il sustituido para el tratamiento de enfermedades y condiciones de la piel, tales como rosacea, daño solar cronico, psoriasis, entre otras; kit farmaceutico. | |
| DOP2016000007A (es) | Pirazolpiridinas sustituidas | |
| SV2017005466A (es) | Pirazolpiridinaminas como inhibidores de mknk1 y mknk2 | |
| CL2015002466A1 (es) | Formulaciones de compuestos orgánicos | |
| BRPI0916571A2 (pt) | composto derivado de alquilaminometiloxazolidinona tricíclo, medicamento e composição farmacêutica que o contém e uso do composto | |
| DOP2015000298A (es) | Compuestos nuevos para el tratamiento del cáncer |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FG | Application granted |