HRP20171807T1 - Spojevi policikličkog karbamoilpiridona i njihova uporaba za liječenje hiv infekcija - Google Patents

Spojevi policikličkog karbamoilpiridona i njihova uporaba za liječenje hiv infekcija Download PDF

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Publication number
HRP20171807T1
HRP20171807T1 HRP20171807TT HRP20171807T HRP20171807T1 HR P20171807 T1 HRP20171807 T1 HR P20171807T1 HR P20171807T T HRP20171807T T HR P20171807TT HR P20171807 T HRP20171807 T HR P20171807T HR P20171807 T1 HRP20171807 T1 HR P20171807T1
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HR
Croatia
Prior art keywords
image
compound according
hydrogen
alkyl
following formula
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HRP20171807TT
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English (en)
Croatian (hr)
Inventor
Mingzhe Ji
Teresa Alejandra Trejo Martin
Manoj C. Desai
Haolun Jin
Hyung-Jung Pyun
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Gilead Sciences, Inc.
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Application filed by Gilead Sciences, Inc. filed Critical Gilead Sciences, Inc.
Publication of HRP20171807T1 publication Critical patent/HRP20171807T1/hr

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • A61P31/18—Antivirals for RNA viruses for HIV
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/14—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/18—Bridged systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Virology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Molecular Biology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • AIDS & HIV (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Pyridine Compounds (AREA)
HRP20171807TT 2013-07-12 2014-07-11 Spojevi policikličkog karbamoilpiridona i njihova uporaba za liječenje hiv infekcija HRP20171807T1 (hr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361845807P 2013-07-12 2013-07-12
EP14745053.0A EP3019499B1 (en) 2013-07-12 2014-07-11 Polycyclic-carbamoylpyridone compounds and their use for the treatment of hiv infections
PCT/US2014/046415 WO2015006733A1 (en) 2013-07-12 2014-07-11 Polycyclic-carbamoylpyridone compounds and their use for the treatment of hiv infections

Publications (1)

Publication Number Publication Date
HRP20171807T1 true HRP20171807T1 (hr) 2018-01-26

Family

ID=51257630

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20171807TT HRP20171807T1 (hr) 2013-07-12 2014-07-11 Spojevi policikličkog karbamoilpiridona i njihova uporaba za liječenje hiv infekcija

Country Status (18)

Country Link
US (6) US9458159B2 (forum.php)
EP (2) EP3252053B1 (forum.php)
JP (1) JP6411492B2 (forum.php)
AU (3) AU2014286995B2 (forum.php)
CA (1) CA2918055C (forum.php)
CY (1) CY1119545T1 (forum.php)
DK (1) DK3019499T3 (forum.php)
ES (2) ES2856867T3 (forum.php)
HR (1) HRP20171807T1 (forum.php)
HU (1) HUE037343T2 (forum.php)
LT (1) LT3019499T (forum.php)
NO (1) NO2865735T3 (forum.php)
PL (1) PL3019499T3 (forum.php)
PT (1) PT3019499T (forum.php)
RS (1) RS56539B1 (forum.php)
SI (2) SI3019499T1 (forum.php)
SM (1) SMT201700525T1 (forum.php)
WO (1) WO2015006733A1 (forum.php)

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TW202133858A (zh) 2019-11-28 2021-09-16 日商鹽野義製藥股份有限公司 以組合整合酶阻礙劑及抗ｈｉｖ藥為特徵之ｈｉｖ感染症的預防及治療用醫藥
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CN116390924A (zh) * 2020-09-30 2023-07-04 吉利德科学公司 桥连三环氨基甲酰基吡啶酮化合物及其用途
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