HRP20120798T1 - Kappa-opijatni agonisti za lijeäśenje dijareja-predominantnog i naizmjeniäśnog sindroma iritabilnog crijeva - Google Patents

Kappa-opijatni agonisti za lijeäśenje dijareja-predominantnog i naizmjeniäśnog sindroma iritabilnog crijeva Download PDF

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Publication number
HRP20120798T1
HRP20120798T1 HRP20120798AT HRP20120798T HRP20120798T1 HR P20120798 T1 HRP20120798 T1 HR P20120798T1 HR P20120798A T HRP20120798A T HR P20120798AT HR P20120798 T HRP20120798 T HR P20120798T HR P20120798 T1 HRP20120798 T1 HR P20120798T1
Authority
HR
Croatia
Prior art keywords
hydroxypyrrolidin
phenyl
ethyl
methyl
diphenylacetamide
Prior art date
Application number
HRP20120798AT
Other languages
English (en)
Croatian (hr)
Inventor
Allen Mangel
Original Assignee
Tioga Pharmaceuticals, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Tioga Pharmaceuticals, Inc. filed Critical Tioga Pharmaceuticals, Inc.
Publication of HRP20120798T1 publication Critical patent/HRP20120798T1/hr

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4015—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil having oxo groups directly attached to the heterocyclic ring, e.g. piracetam, ethosuximide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/10—Laxatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/12—Antidiarrhoeals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

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  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Pyrrole Compounds (AREA)
HRP20120798AT 2007-03-30 2008-03-07 Kappa-opijatni agonisti za lijeäśenje dijareja-predominantnog i naizmjeniäśnog sindroma iritabilnog crijeva HRP20120798T1 (hr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US92084107P 2007-03-30 2007-03-30
PCT/US2008/056317 WO2008121496A1 (en) 2007-03-30 2008-03-07 Kappa-opiate agonists for the treatment of diarrhea-predominant and alternating irritable bowel syndrome

Publications (1)

Publication Number Publication Date
HRP20120798T1 true HRP20120798T1 (hr) 2012-11-30

Family

ID=39795494

Family Applications (1)

Application Number Title Priority Date Filing Date
HRP20120798AT HRP20120798T1 (hr) 2007-03-30 2008-03-07 Kappa-opijatni agonisti za lijeäśenje dijareja-predominantnog i naizmjeniäśnog sindroma iritabilnog crijeva

Country Status (19)

Country Link
US (2) US7960429B2 (enExample)
EP (3) EP2561870A1 (enExample)
JP (2) JP5416085B2 (enExample)
KR (2) KR101208326B1 (enExample)
CN (2) CN102641265A (enExample)
AU (1) AU2008232954A1 (enExample)
BR (1) BRPI0809651A2 (enExample)
CA (1) CA2682608A1 (enExample)
CY (1) CY1113317T1 (enExample)
DK (1) DK2136801T3 (enExample)
ES (1) ES2393815T3 (enExample)
HR (1) HRP20120798T1 (enExample)
IL (1) IL201226A0 (enExample)
MX (1) MX2009010409A (enExample)
PL (1) PL2136801T3 (enExample)
PT (1) PT2136801E (enExample)
RU (1) RU2441655C2 (enExample)
SI (1) SI2136801T1 (enExample)
WO (1) WO2008121496A1 (enExample)

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US11246905B2 (en) 2016-08-15 2022-02-15 President And Fellows Of Harvard College Treating infections using IdsD from Proteus mirabilis
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EP3932390A1 (en) 2020-07-02 2022-01-05 Dr. August Wolff GmbH & Co. KG Arzneimittel Topical gel formulation containing asimadoline
JP7464744B2 (ja) * 2020-10-20 2024-04-09 セトラスホールディングス株式会社 診療支援装置、診療支援方法、診療支援プログラム及び診療支援システム
WO2022155332A1 (en) * 2021-01-13 2022-07-21 Blue Therapeutics, Inc. Methods of treating irritable bowel syndrome

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Also Published As

Publication number Publication date
KR20100016004A (ko) 2010-02-12
EP2136801A4 (en) 2010-05-26
DK2136801T3 (da) 2012-12-17
PL2136801T3 (pl) 2013-01-31
SI2136801T1 (sl) 2013-01-31
JP2010523492A (ja) 2010-07-15
CN102641265A (zh) 2012-08-22
US7960429B2 (en) 2011-06-14
BRPI0809651A2 (pt) 2014-10-07
CY1113317T1 (el) 2016-04-13
US20110046174A1 (en) 2011-02-24
KR101208326B1 (ko) 2012-12-05
US8877800B2 (en) 2014-11-04
PT2136801E (pt) 2012-12-06
AU2008232954A2 (en) 2011-12-01
JP2013173790A (ja) 2013-09-05
JP5416085B2 (ja) 2014-02-12
CN101677997B (zh) 2012-05-09
ES2393815T3 (es) 2012-12-28
HK1139860A1 (en) 2010-09-30
IL201226A0 (en) 2010-05-31
EP2561870A1 (en) 2013-02-27
AU2008232954A1 (en) 2008-10-09
KR101263225B1 (ko) 2013-05-13
RU2441655C2 (ru) 2012-02-10
EP2136801A1 (en) 2009-12-30
EP2636407A3 (en) 2013-11-06
MX2009010409A (es) 2010-03-29
CN101677997A (zh) 2010-03-24
KR20120058614A (ko) 2012-06-07
EP2636407A2 (en) 2013-09-11
US20080242720A1 (en) 2008-10-02
CA2682608A1 (en) 2008-10-09
RU2009140042A (ru) 2011-05-10
EP2136801B1 (en) 2012-08-29
WO2008121496A1 (en) 2008-10-09

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