HRP20080552A9 - Benzimidazole derivative and use thereof - Google Patents

Benzimidazole derivative and use thereof

Info

Publication number
HRP20080552A9
HRP20080552A9 HR20080552A HRP20080552A HRP20080552A9 HR P20080552 A9 HRP20080552 A9 HR P20080552A9 HR 20080552 A HR20080552 A HR 20080552A HR P20080552 A HRP20080552 A HR P20080552A HR P20080552 A9 HRP20080552 A9 HR P20080552A9
Authority
HR
Croatia
Prior art keywords
methyl
benzimidazole derivative
oxo
pharmaceutical agent
benzimidazole
Prior art date
Application number
HR20080552A
Other languages
English (en)
Croatian (hr)
Inventor
Kuroita Takanobu
Ojima Mami
Ban Junko
Original Assignee
Takeda Pharmaceutical Company Limited
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Takeda Pharmaceutical Company Limited filed Critical Takeda Pharmaceutical Company Limited
Publication of HRP20080552A2 publication Critical patent/HRP20080552A2/xx
Publication of HRP20080552A9 publication Critical patent/HRP20080552A9/xx

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245—Oxadiazoles
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HR20080552A 2005-03-30 2008-10-29 Benzimidazole derivative and use thereof HRP20080552A9 (en)

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BRPI0916847A2 (pt) * 2008-07-31 2016-02-10 Takeda Pharmaceutical preparação sólida, e, métodos para estabilizar um composto e para melhorar a propriedade de dissolução de um composto.
JP5559689B2 (ja) 2008-08-06 2014-07-23 協和発酵キリン株式会社 ３環系化合物
AR073380A1 (es) 2008-09-25 2010-11-03 Takeda Pharmaceutical Composicion farmaceutica solida. comprimido multicapa
US9233955B2 (en) * 2011-02-08 2016-01-12 Jubilant Life Sciences, Ltd. Process for the preparation of azilsartan medoxomil
CZ304252B6 (cs) * 2011-04-11 2014-01-29 Zentiva, K. S. Způsob výroby 2-ethoxy-1-((2´-(5-oxo-4,5-dihydro-1,2,4-oxadiazol-3-yl)bifenyl-4-yl)methyl)-1H-benzo[d]imidazol-7-karboxylátů a jejich převedení na azilsartan
KR101275092B1 (ko) * 2011-05-19 2013-06-17 한미정밀화학주식회사 아질사르탄의 개선된 제조방법
CN102827153B (zh) * 2011-06-14 2016-10-05 江苏豪森药业集团有限公司 阿齐沙坦的晶型及其制备方法
JP6281735B2 (ja) * 2013-03-19 2018-02-21 トーアエイヨー株式会社 急性心不全治療薬の評価方法、及び、急性心不全モデルの作製方法

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JP4795362B2 (ja) 2011-10-19
CY1111168T1 (el) 2015-06-11
CR9432A (es) 2008-02-04
MY146254A (en) 2012-07-31
SI1863801T1 (sl) 2010-12-31
WO2006107062A3 (en) 2006-12-14
PL1863801T3 (pl) 2011-03-31
NO20075399L (no) 2007-12-19
US20090054502A1 (en) 2009-02-26
RU2007139928A (ru) 2009-05-10
CA2602624A1 (en) 2006-10-12
US20120172401A1 (en) 2012-07-05
TW200724539A (en) 2007-07-01
IL185726A0 (en) 2008-01-06
GEP20115138B (en) 2011-01-10
KR20070116648A (ko) 2007-12-10
RU2407742C2 (ru) 2010-12-27
HRP20080552A2 (en) 2009-03-31
IL185726A (en) 2012-07-31
RS20080510A (xx) 2009-07-15
DE602006017183D1 (de) 2010-11-11
AU2006231418A1 (en) 2006-10-12
AR055755A1 (es) 2007-09-05
EP1863801B1 (en) 2010-09-29
JP2008534434A (ja) 2008-08-28
PT1863801E (pt) 2010-11-19
DK1863801T3 (da) 2010-11-15
PE20061195A1 (es) 2006-12-21
AU2006231418B2 (en) 2011-10-13
BRPI0608944A2 (pt) 2010-11-16
NZ562887A (en) 2010-10-29
MA29438B1 (fr) 2008-05-02
JP2011190265A (ja) 2011-09-29
EP1863801A2 (en) 2007-12-12
WO2006107062A2 (en) 2006-10-12
HK1115584A1 (en) 2008-12-05
MEP33308A (en) 2010-10-10

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