HK47893A - A crystalline oral cephalosporin hydrate and its compositions - Google Patents

A crystalline oral cephalosporin hydrate and its compositions Download PDF

Info

Publication number
HK47893A
HK47893A HK478/93A HK47893A HK47893A HK 47893 A HK47893 A HK 47893A HK 478/93 A HK478/93 A HK 478/93A HK 47893 A HK47893 A HK 47893A HK 47893 A HK47893 A HK 47893A
Authority
HK
Hong Kong
Prior art keywords
hydrate
crystalline
compositions
oral cephalosporin
gelatin
Prior art date
Application number
HK478/93A
Other languages
English (en)
Inventor
Hamashima Yoshio
Minami Kyoji
Kawata Kyozo
Sakamoto Teruo
Takeda Toyohiko
Suzuki Yusuke
Tujikawa Masonori
Original Assignee
Shionogi Seiyaku Kabushiki Kaisha
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP61156954A external-priority patent/JP2544113B2/ja
Priority claimed from JP21626086A external-priority patent/JPH0717651B2/ja
Application filed by Shionogi Seiyaku Kabushiki Kaisha filed Critical Shionogi Seiyaku Kabushiki Kaisha
Publication of HK47893A publication Critical patent/HK47893A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Cephalosporin Compounds (AREA)
HK478/93A 1986-07-02 1993-05-20 A crystalline oral cephalosporin hydrate and its compositions HK47893A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP61156954A JP2544113B2 (ja) 1986-07-02 1986-07-02 安定なカプセル製剤
JP21626086A JPH0717651B2 (ja) 1986-09-12 1986-09-12 経口投与用セフアロスポリン水和物結晶

Publications (1)

Publication Number Publication Date
HK47893A true HK47893A (en) 1993-05-27

Family

ID=26484565

Family Applications (1)

Application Number Title Priority Date Filing Date
HK478/93A HK47893A (en) 1986-07-02 1993-05-20 A crystalline oral cephalosporin hydrate and its compositions

Country Status (27)

Country Link
US (2) US4812561A (cs)
KR (1) KR950005302B1 (cs)
CN (1) CN1015106B (cs)
AR (1) AR243893A1 (cs)
AT (1) AT392472B (cs)
AU (1) AU594167B2 (cs)
BE (1) BE1001691A4 (cs)
CA (1) CA1283405C (cs)
CH (1) CH672788A5 (cs)
DE (1) DE3721913A1 (cs)
DK (1) DK161080C (cs)
ES (2) ES2004952A6 (cs)
FI (1) FI89052C (cs)
FR (1) FR2601014B1 (cs)
GB (1) GB2192183B (cs)
GR (1) GR871014B (cs)
HK (1) HK47893A (cs)
HU (1) HU200777B (cs)
IE (1) IE59613B1 (cs)
IL (1) IL83059A (cs)
IT (1) IT1211469B (cs)
NL (1) NL193136C (cs)
NO (1) NO170889C (cs)
NZ (1) NZ220764A (cs)
PL (1) PL159180B1 (cs)
RU (1) RU1829932C (cs)
SE (1) SE466257B (cs)

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RU2010111550A (ru) * 2007-08-29 2011-10-10 Шеринг Корпорейшн (US) 2,3-замещенные индольные производные для лечения вирусных инфекций
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US8980920B2 (en) 2009-05-29 2015-03-17 Merck Sharp & Dohme Corp. Antiviral compounds of three linked aryl moieties to treat diseases such as hepatitis C
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US20120276047A1 (en) 2009-11-25 2012-11-01 Rosenblum Stuart B Fused tricyclic compounds and derivatives thereof useful for the treatment of viral diseases
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WO2011103441A1 (en) 2010-02-18 2011-08-25 Schering Corporation Substituted pyridine and pyrimidine derivatives and their use in treating viral infections
KR20130008040A (ko) 2010-03-09 2013-01-21 머크 샤프 앤드 돔 코포레이션 융합된 트리시클릭 실릴 화합물 및 바이러스성 질환의 치료를 위한 그의 사용 방법
EP2566449B1 (en) 2010-05-04 2014-10-08 Mahmut Bilgic Pharmaceutical compositions comprising ceftibuten
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US9242965B2 (en) 2013-12-31 2016-01-26 Boehringer Ingelheim International Gmbh Process for the manufacture of (E)-4-N,N-dialkylamino crotonic acid in HX salt form and use thereof for synthesis of EGFR tyrosine kinase inhibitors
CN103948932B (zh) * 2014-04-17 2016-03-16 海南日中天制药有限公司 一种头孢克肟组合物及其制备方法
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CN106432271A (zh) * 2016-09-21 2017-02-22 临沂草之美医药科技有限公司 一种治疗外科手术感染的药物头孢布烯晶体化合物
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Also Published As

Publication number Publication date
AU7504087A (en) 1988-01-07
NO170889B (no) 1992-09-14
FI872903A0 (fi) 1987-07-01
NZ220764A (en) 1989-09-27
DK336487D0 (da) 1987-06-30
DK161080C (da) 1991-11-11
CA1283405C (en) 1991-04-23
IL83059A0 (en) 1987-12-31
IT1211469B (it) 1989-11-03
IE59613B1 (en) 1994-03-09
AU594167B2 (en) 1990-03-01
DE3721913A1 (de) 1988-01-07
AT392472B (de) 1991-04-10
NO872729D0 (no) 1987-06-30
FR2601014B1 (fr) 1990-09-14
US4812561A (en) 1989-03-14
GB2192183A (en) 1988-01-06
FI89052C (fi) 1993-08-10
DK161080B (da) 1991-05-27
IE871738L (en) 1988-01-02
AR243893A1 (es) 1993-09-30
GB2192183B (en) 1990-05-16
NL193136B (nl) 1998-08-03
NO170889C (no) 1992-12-23
SE8702705L (sv) 1988-01-03
RU1829932C (ru) 1993-07-23
SE466257B (sv) 1992-01-20
CN1015106B (zh) 1991-12-18
GB8715064D0 (en) 1987-08-05
FI872903L (fi) 1988-01-03
PL266567A1 (en) 1988-07-21
FI89052B (fi) 1993-04-30
FR2601014A1 (fr) 1988-01-08
PL159180B1 (pl) 1992-11-30
IT8767566A0 (it) 1987-07-01
ES2004952A6 (es) 1989-02-16
KR880001670A (ko) 1988-04-26
US4933443A (en) 1990-06-12
KR950005302B1 (ko) 1995-05-23
SE8702705D0 (sv) 1987-06-30
DK336487A (da) 1988-01-03
HU200777B (en) 1990-08-28
IL83059A (en) 1992-03-29
CH672788A5 (cs) 1989-12-29
CN87105009A (zh) 1988-03-23
NL193136C (nl) 1998-12-04
GR871014B (en) 1987-11-02
HUT44257A (en) 1988-02-29
ATA165887A (de) 1990-09-15
NO872729L (no) 1988-01-04
ES2008759A6 (es) 1989-08-01
NL8701507A (nl) 1988-02-01
BE1001691A4 (fr) 1990-02-13

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Effective date: 20070625