DK161080C - Krystallinsk hydrat af oralt anvendeligt cephalosporin og praeparat dermed - Google Patents

Krystallinsk hydrat af oralt anvendeligt cephalosporin og praeparat dermed

Info

Publication number
DK161080C
DK161080C DK336487A DK336487A DK161080C DK 161080 C DK161080 C DK 161080C DK 336487 A DK336487 A DK 336487A DK 336487 A DK336487 A DK 336487A DK 161080 C DK161080 C DK 161080C
Authority
DK
Denmark
Prior art keywords
crystallic
hydrate
preparation
oral
used cephalosporin
Prior art date
Application number
DK336487A
Other languages
Danish (da)
English (en)
Other versions
DK161080B (da
DK336487D0 (da
DK336487A (da
Inventor
Yoshio Hamashima
Kyoji Minami
Kyozo Kawata
Teruo Sakamoto
Toyohiko Takeda
Yusuke Suzuki
Masanori Tujikawa
Original Assignee
Shionogi & Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP61156954A external-priority patent/JP2544113B2/ja
Priority claimed from JP21626086A external-priority patent/JPH0717651B2/ja
Application filed by Shionogi & Co filed Critical Shionogi & Co
Publication of DK336487D0 publication Critical patent/DK336487D0/da
Publication of DK336487A publication Critical patent/DK336487A/da
Publication of DK161080B publication Critical patent/DK161080B/da
Application granted granted Critical
Publication of DK161080C publication Critical patent/DK161080C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D501/14—Compounds having a nitrogen atom directly attached in position 7
    • C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
    • C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/542—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/545—Compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins, cefaclor, or cephalexine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Cephalosporin Compounds (AREA)
DK336487A 1986-07-02 1987-06-30 Krystallinsk hydrat af oralt anvendeligt cephalosporin og praeparat dermed DK161080C (da)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP61156954A JP2544113B2 (ja) 1986-07-02 1986-07-02 安定なカプセル製剤
JP15695486 1986-07-02
JP21626086A JPH0717651B2 (ja) 1986-09-12 1986-09-12 経口投与用セフアロスポリン水和物結晶
JP21626086 1986-09-12

Publications (4)

Publication Number Publication Date
DK336487D0 DK336487D0 (da) 1987-06-30
DK336487A DK336487A (da) 1988-01-03
DK161080B DK161080B (da) 1991-05-27
DK161080C true DK161080C (da) 1991-11-11

Family

ID=26484565

Family Applications (1)

Application Number Title Priority Date Filing Date
DK336487A DK161080C (da) 1986-07-02 1987-06-30 Krystallinsk hydrat af oralt anvendeligt cephalosporin og praeparat dermed

Country Status (27)

Country Link
US (2) US4812561A (cs)
KR (1) KR950005302B1 (cs)
CN (1) CN1015106B (cs)
AR (1) AR243893A1 (cs)
AT (1) AT392472B (cs)
AU (1) AU594167B2 (cs)
BE (1) BE1001691A4 (cs)
CA (1) CA1283405C (cs)
CH (1) CH672788A5 (cs)
DE (1) DE3721913A1 (cs)
DK (1) DK161080C (cs)
ES (2) ES2004952A6 (cs)
FI (1) FI89052C (cs)
FR (1) FR2601014B1 (cs)
GB (1) GB2192183B (cs)
GR (1) GR871014B (cs)
HK (1) HK47893A (cs)
HU (1) HU200777B (cs)
IE (1) IE59613B1 (cs)
IL (1) IL83059A (cs)
IT (1) IT1211469B (cs)
NL (1) NL193136C (cs)
NO (1) NO170889C (cs)
NZ (1) NZ220764A (cs)
PL (1) PL159180B1 (cs)
RU (1) RU1829932C (cs)
SE (1) SE466257B (cs)

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JP5619743B2 (ja) 2008-08-20 2014-11-05 メルク・シャープ・アンド・ドーム・コーポレーションＭｅｒｃｋ Ｓｈａｒｐ ＆ Ｄｏｈｍｅ Ｃｏｒｐ． エテニル置換ピリジンおよびピリミジン誘導体およびウイルス感染の治療におけるそれらの使用
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JP2012528195A (ja) 2009-05-29 2012-11-12 メルク・シャープ・アンド・ドーム・コーポレーション Ｃ型肝炎などの疾患を処置するための３つの結合アリール部分で構成された抗菌性化合物
DK2451445T3 (da) 2009-07-06 2019-06-24 Boehringer Ingelheim Int Fremgangsmåde til at tørre bibw2992, dets salte og faste farmaceutiske formuleringer omfattende denne aktive ingrediens
JP2013512246A (ja) 2009-11-25 2013-04-11 メルク・シャープ・アンド・ドーム・コーポレーション ウイルス疾患治療に有用な縮合型三環式化合物およびその誘導体
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WO2013033899A1 (en) 2011-09-08 2013-03-14 Merck Sharp & Dohme Corp. Substituted benzofuran compounds and methods of use thereof for the treatment of viral diseases
WO2013033901A1 (en) 2011-09-08 2013-03-14 Merck Sharp & Dohme Corp. Heterocyclic-substituted benzofuran derivatives and methods of use thereof for the treatment of viral diseases
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Also Published As

Publication number Publication date
AT392472B (de) 1991-04-10
NO170889C (no) 1992-12-23
PL159180B1 (pl) 1992-11-30
KR950005302B1 (ko) 1995-05-23
NO872729D0 (no) 1987-06-30
SE8702705L (sv) 1988-01-03
IE871738L (en) 1988-01-02
SE466257B (sv) 1992-01-20
IT8767566A0 (it) 1987-07-01
AU7504087A (en) 1988-01-07
IL83059A0 (en) 1987-12-31
NO170889B (no) 1992-09-14
IT1211469B (it) 1989-11-03
CA1283405C (en) 1991-04-23
AU594167B2 (en) 1990-03-01
NL193136C (nl) 1998-12-04
FI872903L (fi) 1988-01-03
ES2004952A6 (es) 1989-02-16
DK161080B (da) 1991-05-27
BE1001691A4 (fr) 1990-02-13
FR2601014B1 (fr) 1990-09-14
HK47893A (en) 1993-05-27
SE8702705D0 (sv) 1987-06-30
CH672788A5 (cs) 1989-12-29
DK336487D0 (da) 1987-06-30
FR2601014A1 (fr) 1988-01-08
KR880001670A (ko) 1988-04-26
US4812561A (en) 1989-03-14
US4933443A (en) 1990-06-12
PL266567A1 (en) 1988-07-21
DE3721913A1 (de) 1988-01-07
GB2192183B (en) 1990-05-16
FI89052B (fi) 1993-04-30
IE59613B1 (en) 1994-03-09
RU1829932C (ru) 1993-07-23
NO872729L (no) 1988-01-04
AR243893A1 (es) 1993-09-30
GB2192183A (en) 1988-01-06
ATA165887A (de) 1990-09-15
CN1015106B (zh) 1991-12-18
GB8715064D0 (en) 1987-08-05
NL193136B (nl) 1998-08-03
FI89052C (fi) 1993-08-10
DK336487A (da) 1988-01-03
CN87105009A (zh) 1988-03-23
HU200777B (en) 1990-08-28
NL8701507A (nl) 1988-02-01
ES2008759A6 (es) 1989-08-01
IL83059A (en) 1992-03-29
HUT44257A (en) 1988-02-29
GR871014B (en) 1987-11-02
FI872903A0 (fi) 1987-07-01
NZ220764A (en) 1989-09-27

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