HK1147094A1 - Alkylsulfonyl-substituted thiazolide compounds - Google Patents

Alkylsulfonyl-substituted thiazolide compounds

Info

Publication number
HK1147094A1
HK1147094A1 HK11101101.1A HK11101101A HK1147094A1 HK 1147094 A1 HK1147094 A1 HK 1147094A1 HK 11101101 A HK11101101 A HK 11101101A HK 1147094 A1 HK1147094 A1 HK 1147094A1
Authority
HK
Hong Kong
Prior art keywords
alkylsulfonyl
thiazolide compounds
substituted
substituted thiazolide
compounds
Prior art date
Application number
HK11101101.1A
Other languages
English (en)
Inventor
J Edward Semple
Jean-Francois Rossignol
Original Assignee
Romark Lab Lc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39791394&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1147094(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Romark Lab Lc filed Critical Romark Lab Lc
Publication of HK1147094A1 publication Critical patent/HK1147094A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
    • C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D277/38—Nitrogen atoms
    • C07D277/44—Acylated amino or imino radicals
    • C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12—Antivirals
    • A61P31/14—Antivirals for RNA viruses
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
HK11101101.1A 2007-08-03 2011-02-02 Alkylsulfonyl-substituted thiazolide compounds HK1147094A1 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US95375807P 2007-08-03 2007-08-03
US4695608P 2008-04-22 2008-04-22
US5636908P 2008-05-27 2008-05-27
PCT/US2008/071990 WO2009035788A1 (en) 2007-08-03 2008-08-01 Alkylsulfonyl-substituted thiazolide compounds

Publications (1)

Publication Number Publication Date
HK1147094A1 true HK1147094A1 (en) 2011-07-29

Family

ID=39791394

Family Applications (1)

Application Number Title Priority Date Filing Date
HK11101101.1A HK1147094A1 (en) 2007-08-03 2011-02-02 Alkylsulfonyl-substituted thiazolide compounds

Country Status (16)

Country Link
US (2) US8124632B2 (ja)
EP (1) EP2178852B9 (ja)
JP (1) JP5676258B2 (ja)
CN (1) CN101835765B (ja)
AR (1) AR068334A1 (ja)
AU (1) AU2008299781B2 (ja)
BR (1) BRPI0815057B8 (ja)
CA (1) CA2695517C (ja)
CL (1) CL2008002295A1 (ja)
EA (1) EA019357B1 (ja)
ES (1) ES2550755T3 (ja)
HK (1) HK1147094A1 (ja)
MX (1) MX2010001358A (ja)
PT (1) PT2178852E (ja)
TW (1) TWI453018B (ja)
WO (1) WO2009035788A1 (ja)

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US9333193B2 (en) 2010-09-20 2016-05-10 University Of Virginia Patent Foundation Compositions and methods for treating tuberculosis
CN103269593A (zh) * 2010-11-01 2013-08-28 罗马克实验室有限公司 烷基亚磺酰基取代的噻唑化物化合物
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CN106565626B (zh) * 2016-10-10 2022-06-10 淮海工学院 2-氨基-4-芳基-5-甲硫基噻唑类化合物的合成方法
WO2018107332A1 (zh) * 2016-12-12 2018-06-21 中山大学 一类手性芳杂胺类衍生物及其合成方法和应用
CN108610301B (zh) * 2016-12-12 2021-08-31 中山大学 一类手性芳杂胺类衍生物及其合成方法和应用
WO2018195035A1 (en) 2017-04-18 2018-10-25 Romark Laboratories L.C. Inhibition of protein disulfide-isomerase a3
CN111848601B (zh) * 2019-04-30 2022-06-21 南京海璞医药科技有限公司 一种含稠环的化合物、其应用及含其的药物组合物
CN112480104A (zh) * 2019-09-11 2021-03-12 北京美倍他药物研究有限公司 硝唑尼特衍生物及其医药用途
US20230303504A1 (en) 2020-07-20 2023-09-28 Romark Laboratories, L.C. Crystalline salts of tizoxanide and 2-hydroxy-n-(5-chloro-1,3-thiazol-2-yl)benzamide (rm-4848) with ethanolamine, morpholine, propanolamine, piperazine and n-methylpiperazine
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Also Published As

Publication number Publication date
US20090036467A1 (en) 2009-02-05
EA019357B1 (ru) 2014-03-31
CA2695517C (en) 2016-09-20
PT2178852E (pt) 2015-11-12
JP2010535712A (ja) 2010-11-25
BRPI0815057B8 (pt) 2021-05-25
CN101835765B (zh) 2013-05-29
US8124632B2 (en) 2012-02-28
TWI453018B (zh) 2014-09-21
AU2008299781B2 (en) 2013-11-14
WO2009035788A1 (en) 2009-03-19
ES2550755T3 (es) 2015-11-12
AR068334A1 (es) 2009-11-11
CL2008002295A1 (es) 2009-03-27
TW200911239A (en) 2009-03-16
CN101835765A (zh) 2010-09-15
AU2008299781A1 (en) 2009-03-19
MX2010001358A (es) 2010-04-09
US8895752B2 (en) 2014-11-25
US20120122939A1 (en) 2012-05-17
BRPI0815057B1 (pt) 2020-11-10
BRPI0815057A2 (pt) 2015-07-28
JP5676258B2 (ja) 2015-02-25
EP2178852A1 (en) 2010-04-28
EP2178852B1 (en) 2015-07-22
EP2178852B9 (en) 2016-06-22
EA201070182A1 (ru) 2010-10-29
CA2695517A1 (en) 2009-03-19

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Legal Events

Date Code Title Description
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20230801