HK1135705A1 - Piperidine gpcr agonists - Google Patents

Piperidine gpcr agonists

Info

Publication number
HK1135705A1
HK1135705A1 HK10103733.4A HK10103733A HK1135705A1 HK 1135705 A1 HK1135705 A1 HK 1135705A1 HK 10103733 A HK10103733 A HK 10103733A HK 1135705 A1 HK1135705 A1 HK 1135705A1
Authority
HK
Hong Kong
Prior art keywords
gpcr agonists
piperidine
piperidine gpcr
agonists
gpcr
Prior art date
Application number
HK10103733.4A
Other languages
English (en)
Inventor
Matthew Colin Thor Fyfe
Revathy Perpetua Jeevaratnam
John Keily
Simon Andrew Swain
Lisa Sarah Bertram
Original Assignee
Prosidion Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0700125A external-priority patent/GB0700125D0/en
Priority claimed from GB0708746A external-priority patent/GB0708746D0/en
Priority claimed from GB0719763A external-priority patent/GB0719763D0/en
Application filed by Prosidion Ltd filed Critical Prosidion Ltd
Publication of HK1135705A1 publication Critical patent/HK1135705A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Peptides Or Proteins (AREA)
  • Pyridine Compounds (AREA)
HK10103733.4A 2007-01-04 2010-04-16 Piperidine gpcr agonists HK1135705A1 (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB0700125A GB0700125D0 (en) 2007-01-04 2007-01-04 GPCR agonists
GB0708746A GB0708746D0 (en) 2007-05-08 2007-05-08 GPCR agonists
GB0719763A GB0719763D0 (en) 2007-10-10 2007-10-10 GPCR agonists
PCT/GB2008/050013 WO2008081207A1 (en) 2007-01-04 2008-01-04 Piperidine gpcr agonists

Publications (1)

Publication Number Publication Date
HK1135705A1 true HK1135705A1 (en) 2010-06-11

Family

ID=39199058

Family Applications (1)

Application Number Title Priority Date Filing Date
HK10103733.4A HK1135705A1 (en) 2007-01-04 2010-04-16 Piperidine gpcr agonists

Country Status (21)

Country Link
US (1) US20100105732A1 (sl)
EP (2) EP2114935B1 (sl)
JP (1) JP2010514831A (sl)
AR (1) AR064735A1 (sl)
AT (1) ATE517103T1 (sl)
BR (1) BRPI0806500A2 (sl)
CA (1) CA2674455A1 (sl)
CL (1) CL2008000018A1 (sl)
CY (1) CY1112474T1 (sl)
DK (1) DK2114935T3 (sl)
EA (1) EA015130B1 (sl)
HK (1) HK1135705A1 (sl)
HR (1) HRP20110750T1 (sl)
PE (1) PE20081659A1 (sl)
PL (1) PL2114935T3 (sl)
PT (1) PT2114935E (sl)
RS (1) RS51943B (sl)
SA (1) SA08280757B1 (sl)
SI (1) SI2114935T1 (sl)
TW (1) TW200835482A (sl)
WO (1) WO2008081207A1 (sl)

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Also Published As

Publication number Publication date
AR064735A1 (es) 2009-04-22
US20100105732A1 (en) 2010-04-29
EP2114935B1 (en) 2011-07-20
EP2114935A1 (en) 2009-11-11
SI2114935T1 (sl) 2011-11-30
RS51943B (en) 2012-02-29
JP2010514831A (ja) 2010-05-06
WO2008081207A1 (en) 2008-07-10
CA2674455A1 (en) 2008-07-10
BRPI0806500A2 (pt) 2014-04-22
DK2114935T3 (da) 2011-10-31
EA015130B1 (ru) 2011-06-30
ATE517103T1 (de) 2011-08-15
SA08280757B1 (ar) 2011-01-15
TW200835482A (en) 2008-09-01
PE20081659A1 (es) 2008-10-24
CY1112474T1 (el) 2015-12-09
CL2008000018A1 (es) 2008-08-01
PL2114935T3 (pl) 2012-03-30
EP2377864A1 (en) 2011-10-19
PT2114935E (pt) 2011-10-17
EA200900880A1 (ru) 2010-02-26
HRP20110750T1 (hr) 2011-11-30

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PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20150104