HK1091480A1 - Quinazoline derivatives as tyrosine kinase inhibitors - Google Patents

Quinazoline derivatives as tyrosine kinase inhibitors

Info

Publication number
HK1091480A1
HK1091480A1 HK06111949A HK06111949A HK1091480A1 HK 1091480 A1 HK1091480 A1 HK 1091480A1 HK 06111949 A HK06111949 A HK 06111949A HK 06111949 A HK06111949 A HK 06111949A HK 1091480 A1 HK1091480 A1 HK 1091480A1
Authority
HK
Hong Kong
Prior art keywords
tyrosine kinase
kinase inhibitors
quinazoline derivatives
quinazoline
derivatives
Prior art date
Application number
HK06111949A
Other languages
English (en)
Inventor
Hennequin Laurent Francois Andre
Halsall Christopher Thomas
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34315440&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HK1091480(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GBGB0321620.7A external-priority patent/GB0321620D0/en
Priority claimed from GB0406163A external-priority patent/GB0406163D0/en
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of HK1091480A1 publication Critical patent/HK1091480A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C04—CEMENTS; CONCRETE; ARTIFICIAL STONE; CERAMICS; REFRACTORIES
    • C04B—LIME, MAGNESIA; SLAG; CEMENTS; COMPOSITIONS THEREOF, e.g. MORTARS, CONCRETE OR LIKE BUILDING MATERIALS; ARTIFICIAL STONE; CERAMICS; REFRACTORIES; TREATMENT OF NATURAL STONE
    • C04B35/00—Shaped ceramic products characterised by their composition; Ceramics compositions; Processing powders of inorganic compounds preparatory to the manufacturing of ceramic products
    • C04B35/622—Forming processes; Processing powders of inorganic compounds preparatory to the manufacturing of ceramic products
    • C04B35/626—Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B
    • C04B35/63—Preparing or treating the powders individually or as batches ; preparing or treating macroscopic reinforcing agents for ceramic products, e.g. fibres; mechanical aspects section B using additives specially adapted for forming the products, e.g.. binder binders
    • C04B35/632—Organic additives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/14—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing three or more hetero rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Ceramic Engineering (AREA)
  • Health & Medical Sciences (AREA)
  • Manufacturing & Machinery (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Inorganic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Structural Engineering (AREA)
  • Materials Engineering (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
HK06111949A 2003-09-16 2006-10-31 Quinazoline derivatives as tyrosine kinase inhibitors HK1091480A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GBGB0321620.7A GB0321620D0 (en) 2003-09-16 2003-09-16 Quinazoline derivatives
GB0406163A GB0406163D0 (en) 2004-03-19 2004-03-19 Quinazoline derivatives
PCT/GB2004/003923 WO2005026150A1 (en) 2003-09-16 2004-09-13 Quinazoline derivatives as tyrosine kinase inhibitors

Publications (1)

Publication Number Publication Date
HK1091480A1 true HK1091480A1 (en) 2007-01-19

Family

ID=34315440

Family Applications (1)

Application Number Title Priority Date Filing Date
HK06111949A HK1091480A1 (en) 2003-09-16 2006-10-31 Quinazoline derivatives as tyrosine kinase inhibitors

Country Status (25)

Country Link
US (2) US7569577B2 (pt)
EP (1) EP1667991B1 (pt)
JP (1) JP4795952B2 (pt)
AR (1) AR045663A1 (pt)
AT (1) ATE395346T1 (pt)
AU (1) AU2004272348B2 (pt)
BR (1) BRPI0414489A8 (pt)
CA (1) CA2538884C (pt)
CO (1) CO5690594A2 (pt)
CY (1) CY1108186T1 (pt)
DE (1) DE602004013806D1 (pt)
DK (1) DK1667991T3 (pt)
ES (1) ES2305844T3 (pt)
HK (1) HK1091480A1 (pt)
HR (1) HRP20080329T3 (pt)
IL (1) IL174261A0 (pt)
MX (1) MXPA06002964A (pt)
NO (1) NO20061322L (pt)
PL (1) PL1667991T3 (pt)
PT (1) PT1667991E (pt)
RU (1) RU2378268C2 (pt)
SI (1) SI1667991T1 (pt)
TW (1) TW200519104A (pt)
UA (1) UA84167C2 (pt)
WO (1) WO2005026150A1 (pt)

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US20070032513A1 (en) * 2003-09-16 2007-02-08 Hennequin Laurent F A Quinazoline derivatives
US20070032508A1 (en) * 2003-09-16 2007-02-08 Bradbury Robert H Quinazoline derivatives as tyrosine kinase inhibitors
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GB0322409D0 (en) * 2003-09-25 2003-10-29 Astrazeneca Ab Quinazoline derivatives
GB0326459D0 (en) * 2003-11-13 2003-12-17 Astrazeneca Ab Quinazoline derivatives
US8017321B2 (en) * 2004-01-23 2011-09-13 The Regents Of The University Of Colorado, A Body Corporate Gefitinib sensitivity-related gene expression and products and methods related thereto
US20080113874A1 (en) * 2004-01-23 2008-05-15 The Regents Of The University Of Colorado Gefitinib sensitivity-related gene expression and products and methods related thereto
WO2005075439A1 (en) * 2004-02-03 2005-08-18 Astrazeneca Ab Quinazoline derivatives
CA2567293C (en) * 2004-05-27 2017-05-16 The Regents Of The University Of Colorado Methods for prediction of clinical outcome to epidermal growth factor receptor inhibitors by cancer patients
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AU2006223086A1 (en) * 2005-03-11 2006-09-21 The Regents Of The University Of Colorado Histone deacetylase inhibitors sensitize cancer cells to epidermal growth factor inhibitors
GB0508715D0 (en) * 2005-04-29 2005-06-08 Astrazeneca Ab Chemical compounds
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CN102452988B (zh) 2010-10-27 2016-01-27 中国科学院化学研究所 一种喹唑啉衍生物及其制备方法
EP2680844B1 (en) 2011-03-04 2016-10-19 GlaxoSmithKline Intellectual Property Development Limited Amino-quinolines as kinase inhibitors
TWI547494B (zh) 2011-08-18 2016-09-01 葛蘭素史克智慧財產發展有限公司 作為激酶抑制劑之胺基喹唑啉類
TWI592417B (zh) * 2012-09-13 2017-07-21 葛蘭素史克智慧財產發展有限公司 胺基喹唑啉激酶抑制劑之前藥
TW201425307A (zh) 2012-09-13 2014-07-01 Glaxosmithkline Llc 作為激酶抑制劑之胺基－喹啉類
RU2662810C2 (ru) 2013-02-21 2018-07-31 Глэксосмитклайн Интеллекчуал Проперти Дивелопмент Лимитед Хиназолины в качестве ингибиторов киназы
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Also Published As

Publication number Publication date
CA2538884A1 (en) 2005-03-24
RU2006112599A (ru) 2007-11-10
AR045663A1 (es) 2005-11-02
ES2305844T3 (es) 2008-11-01
HRP20080329T3 (en) 2008-08-31
SI1667991T1 (sl) 2008-10-31
CO5690594A2 (es) 2006-10-31
ATE395346T1 (de) 2008-05-15
CA2538884C (en) 2010-09-21
RU2378268C2 (ru) 2010-01-10
US7569577B2 (en) 2009-08-04
NO20061322L (no) 2006-06-15
JP4795952B2 (ja) 2011-10-19
DE602004013806D1 (en) 2008-06-26
DK1667991T3 (da) 2008-08-18
IL174261A0 (en) 2006-08-01
TW200519104A (en) 2005-06-16
US20070043009A1 (en) 2007-02-22
EP1667991B1 (en) 2008-05-14
BRPI0414489A8 (pt) 2019-01-15
PT1667991E (pt) 2008-07-14
PL1667991T3 (pl) 2008-12-31
AU2004272348A1 (en) 2005-03-24
MXPA06002964A (es) 2006-06-14
WO2005026150A1 (en) 2005-03-24
EP1667991A1 (en) 2006-06-14
BRPI0414489A (pt) 2006-11-14
AU2004272348B2 (en) 2008-09-04
US20090312343A1 (en) 2009-12-17
UA84167C2 (ru) 2008-09-25
JP2007505872A (ja) 2007-03-15
CY1108186T1 (el) 2014-02-12

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