HK1008898A1 - Hetero-aromatic ring substituted phenyloxazolidinone antimicrobials - Google Patents

Hetero-aromatic ring substituted phenyloxazolidinone antimicrobials

Info

Publication number
HK1008898A1
HK1008898A1 HK98109662A HK98109662A HK1008898A1 HK 1008898 A1 HK1008898 A1 HK 1008898A1 HK 98109662 A HK98109662 A HK 98109662A HK 98109662 A HK98109662 A HK 98109662A HK 1008898 A1 HK1008898 A1 HK 1008898A1
Authority
HK
Hong Kong
Prior art keywords
optionally substituted
hetero
alkoxy
pct
aromatic
Prior art date
Application number
HK98109662A
Other languages
English (en)
Inventor
Douglas K Hutchinson
Original Assignee
Upjohn Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Upjohn Co filed Critical Upjohn Co
Publication of HK1008898A1 publication Critical patent/HK1008898A1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
HK98109662A 1995-02-03 1998-08-04 Hetero-aromatic ring substituted phenyloxazolidinone antimicrobials HK1008898A1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US38427895A 1995-02-03 1995-02-03
PCT/US1996/000718 WO1996023788A1 (en) 1995-02-03 1996-01-29 Hetero-aromatic ring substituted phenyloxazolidinone antimicrobials

Publications (1)

Publication Number Publication Date
HK1008898A1 true HK1008898A1 (en) 1999-07-23

Family

ID=23516681

Family Applications (1)

Application Number Title Priority Date Filing Date
HK98109662A HK1008898A1 (en) 1995-02-03 1998-08-04 Hetero-aromatic ring substituted phenyloxazolidinone antimicrobials

Country Status (20)

Country Link
US (1) US5910504A (sv)
EP (1) EP0807112B1 (sv)
JP (1) JPH10513446A (sv)
KR (1) KR100441334B1 (sv)
CN (1) CN1075073C (sv)
AT (1) ATE205205T1 (sv)
BR (1) BR9607017A (sv)
CA (1) CA2208603A1 (sv)
CZ (1) CZ231497A3 (sv)
DE (1) DE69615002T2 (sv)
DK (1) DK0807112T3 (sv)
ES (1) ES2163004T3 (sv)
FI (1) FI973217A0 (sv)
HK (1) HK1008898A1 (sv)
NO (1) NO309526B1 (sv)
NZ (1) NZ302844A (sv)
PL (1) PL185872B1 (sv)
PT (1) PT807112E (sv)
RU (1) RU2154645C2 (sv)
WO (1) WO1996023788A1 (sv)

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EP2072514A1 (en) * 2007-12-17 2009-06-24 Ferrer Internacional, S.A. 1(2)H-tetrazol-5-yl-phenyl-oxazolidinones as antibacterial agents
WO2012171479A1 (zh) * 2011-06-17 2012-12-20 四川大学 噁唑烷酮类化合物及其在制备抗生素药物中的用途
EP2602248A1 (en) 2011-12-05 2013-06-12 University Of Leicester Novel pyrrole compounds
CN104364240B (zh) * 2012-06-08 2017-02-22 四川贝力克生物技术有限责任公司 一种用于预防或治疗分支杆菌疾病的药物
CN104873510B (zh) * 2014-02-28 2019-03-19 四川好医生药业集团有限公司 噁唑烷酮类化合物抗生物膜用途
CN103965183B (zh) * 2014-03-17 2017-05-03 上海应用技术学院 一种含氟噁唑烷酮类化合物及其制备方法和应用
CN105272976B (zh) * 2014-07-22 2018-11-20 四川好医生药业集团有限公司 一种噁唑烷酮类化合物
CN105399737B (zh) * 2014-09-10 2018-09-21 四川好医生药业集团有限公司 噁唑烷酮类化合物及其用途
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US9988369B2 (en) 2016-05-03 2018-06-05 Amgen Inc. Heterocyclic triazole compounds as agonists of the APJ receptor
US11191762B2 (en) 2016-11-16 2021-12-07 Amgen Inc. Alkyl substituted triazole compounds as agonists of the APJ Receptor
EP3541810B1 (en) 2016-11-16 2020-12-23 Amgen Inc. Triazole phenyl compounds as agonists of the apj receptor
EP3541803B1 (en) 2016-11-16 2020-12-23 Amgen Inc. Triazole pyridyl compounds as agonists of the apj receptor
US10736883B2 (en) 2016-11-16 2020-08-11 Amgen Inc. Triazole furan compounds as agonists of the APJ receptor
MA46827A (fr) 2016-11-16 2019-09-25 Amgen Inc Composés de triazole à substitution cycloalkyle en tant qu'agonistes du récepteur apj
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CN106831615B (zh) * 2017-02-15 2019-02-15 南京农业大学 一类1，2，3－三唑－5－酰胺类化合物作为农用杀菌剂的应用
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Also Published As

Publication number Publication date
FI973217A (sv) 1997-08-04
NO973550D0 (no) 1997-08-01
PT807112E (pt) 2002-02-28
ATE205205T1 (de) 2001-09-15
CA2208603A1 (en) 1996-08-08
CZ231497A3 (cs) 1998-08-12
RU2154645C2 (ru) 2000-08-20
AU4899896A (en) 1996-08-21
PL321663A1 (en) 1997-12-22
ES2163004T3 (es) 2002-01-16
KR100441334B1 (ko) 2004-10-20
NZ302844A (en) 1999-06-29
CN1172484A (zh) 1998-02-04
WO1996023788A1 (en) 1996-08-08
PL185872B1 (pl) 2003-08-29
EP0807112A1 (en) 1997-11-19
EP0807112B1 (en) 2001-09-05
NO309526B1 (no) 2001-02-12
DK0807112T3 (da) 2001-12-17
BR9607017A (pt) 1997-10-28
FI973217A0 (sv) 1997-08-04
AU703465B2 (en) 1999-03-25
KR19980701908A (ko) 1998-06-25
US5910504A (en) 1999-06-08
DE69615002D1 (de) 2001-10-11
JPH10513446A (ja) 1998-12-22
CN1075073C (zh) 2001-11-21
NO973550L (no) 1997-10-03
DE69615002T2 (de) 2002-06-13

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Effective date: 20060129