GT201400042A - Compuesto de benzotiazolona - Google Patents

Compuesto de benzotiazolona

Info

Publication number
GT201400042A
GT201400042A GT201400042A GT201400042A GT201400042A GT 201400042 A GT201400042 A GT 201400042A GT 201400042 A GT201400042 A GT 201400042A GT 201400042 A GT201400042 A GT 201400042A GT 201400042 A GT201400042 A GT 201400042A
Authority
GT
Guatemala
Prior art keywords
benzotiazolona
composite
provides
compound
pharmaceutically acceptable
Prior art date
Application number
GT201400042A
Other languages
English (en)
Spanish (es)
Inventor
Cao Jun
Erb Bernhard
Fairhurst Robin Alec
Grandeury Arnaud
Hatakeyama Shinji
Koziczak-Holbro Magdalena
Lai Xinzhong
Lustenberger Philipp
Riebesehl Bernd
Tufilli Nicola
Ullrich Thomas
Wu Xiang
Zhou Jianguang
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=47010668&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=GT201400042(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed filed Critical
Publication of GT201400042A publication Critical patent/GT201400042A/es

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/425—Thiazoles
    • A61K31/428—Thiazoles condensed with carbocyclic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
    • C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D277/62—Benzothiazoles
    • C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/16—Amides, e.g. hydroxamic acids
    • A61K31/165—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167—Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00—Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06—Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00—Drugs for disorders of the muscular or neuromuscular system
    • A61P21/04—Drugs for disorders of the muscular or neuromuscular system for myasthenia gravis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C53/00—Saturated compounds having only one carboxyl group bound to an acyclic carbon atom or hydrogen
    • C07C53/08—Acetic acid
    • C07C53/10—Salts thereof
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/07—Optical isomers
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Neurology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Hematology (AREA)
  • Diabetes (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Emergency Medicine (AREA)
  • Cosmetics (AREA)
  • Addition Polymer Or Copolymer, Post-Treatments, Or Chemical Modifications (AREA)
  • Macromonomer-Based Addition Polymer (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
GT201400042A 2011-09-06 2014-03-04 Compuesto de benzotiazolona GT201400042A (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CN2011079379 2011-09-06

Publications (1)

Publication Number Publication Date
GT201400042A true GT201400042A (es) 2015-02-19

Family

ID=47010668

Family Applications (1)

Application Number Title Priority Date Filing Date
GT201400042A GT201400042A (es) 2011-09-06 2014-03-04 Compuesto de benzotiazolona

Country Status (39)

Country Link
US (6) US8933108B2 (enExample)
EP (1) EP2753609B1 (enExample)
JP (2) JP6130835B2 (enExample)
KR (2) KR101800140B1 (enExample)
CN (2) CN106187942B (enExample)
AP (1) AP3830A (enExample)
AR (1) AR087787A1 (enExample)
AU (1) AU2013200422C1 (enExample)
BR (1) BR112014004732A2 (enExample)
CA (1) CA2845766A1 (enExample)
CL (1) CL2014000493A1 (enExample)
CO (1) CO6900147A2 (enExample)
CR (1) CR20140114A (enExample)
CU (1) CU24303B1 (enExample)
CY (1) CY1118585T1 (enExample)
DK (1) DK2753609T3 (enExample)
EA (1) EA022909B1 (enExample)
ES (1) ES2615052T3 (enExample)
GT (1) GT201400042A (enExample)
HR (1) HRP20170075T1 (enExample)
HU (1) HUE030530T2 (enExample)
IL (1) IL231235A (enExample)
JO (1) JO3192B1 (enExample)
LT (1) LT2753609T (enExample)
MX (1) MX345405B (enExample)
MY (1) MY163301A (enExample)
PE (1) PE20141993A1 (enExample)
PH (1) PH12014500399A1 (enExample)
PL (1) PL2753609T3 (enExample)
PT (1) PT2753609T (enExample)
RS (1) RS55468B1 (enExample)
SG (1) SG2014013114A (enExample)
SI (1) SI2753609T1 (enExample)
TN (1) TN2014000060A1 (enExample)
TW (1) TWI555738B (enExample)
UA (1) UA114295C2 (enExample)
UY (1) UY34312A (enExample)
WO (1) WO2013035047A1 (enExample)
ZA (2) ZA201401112B (enExample)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JO3192B1 (ar) 2011-09-06 2018-03-08 Novartis Ag مركب بنزوثيازولون
UA117092C2 (uk) 2011-09-06 2018-06-25 Байєр Інтеллектуал Проперті Гмбх Амінозаміщені імідазопіридазини
SI2890687T1 (sl) * 2012-08-30 2017-10-30 Novartis Ag Soli benzotiazolonske spojine kot agonist beta-2-adrenoceptorja
ES2646916T3 (es) 2012-11-19 2017-12-18 Bayer Pharma Aktiengesellschaft Aminoimidazopiridazinas como inhibidores de MKNK1 cinasa
WO2014132205A1 (en) 2013-02-28 2014-09-04 Novartis Ag Formulation comprising benzothiazolone compound
US10967119B1 (en) 2019-04-01 2021-04-06 Azizi Bilal Wearable medication injecting device

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EP1144387A1 (en) 1998-12-04 2001-10-17 Neurosearch A/S New benzimidazolone-, benzoxazolone-, or benzothiazolone derivatives as ion channel modulating agents
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JP2005187357A (ja) 2003-12-25 2005-07-14 Nippon Suisan Kaisha Ltd 選択的なβ2受容体アゴニスト活性を有するベンゾチアゾロン誘導体の製造方法
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GB201009801D0 (en) 2010-06-11 2010-07-21 Astrazeneca Ab Compounds 950
GB201107985D0 (en) 2011-05-13 2011-06-29 Astrazeneca Ab Process
JO3192B1 (ar) 2011-09-06 2018-03-08 Novartis Ag مركب بنزوثيازولون
SI2890687T1 (sl) * 2012-08-30 2017-10-30 Novartis Ag Soli benzotiazolonske spojine kot agonist beta-2-adrenoceptorja
WO2014132205A1 (en) 2013-02-28 2014-09-04 Novartis Ag Formulation comprising benzothiazolone compound

Also Published As

Publication number Publication date
JP2017132781A (ja) 2017-08-03
CA2845766A1 (en) 2013-03-14
JP6340103B2 (ja) 2018-06-06
PE20141993A1 (es) 2014-12-17
BR112014004732A2 (pt) 2017-03-28
TW201317221A (zh) 2013-05-01
CO6900147A2 (es) 2014-03-20
US9913828B2 (en) 2018-03-13
CL2014000493A1 (es) 2014-10-03
NZ621089A (en) 2015-07-31
WO2013035047A1 (en) 2013-03-14
LT2753609T (lt) 2017-01-10
CN106187942B (zh) 2020-06-26
KR20160038079A (ko) 2016-04-06
RS55468B1 (sr) 2017-04-28
JP2014525472A (ja) 2014-09-29
UY34312A (es) 2013-04-30
PT2753609T (pt) 2017-02-08
AU2013200422C1 (en) 2015-01-15
US20160075670A1 (en) 2016-03-17
MX345405B (es) 2017-01-30
PL2753609T3 (pl) 2017-05-31
KR101800140B1 (ko) 2017-11-21
EP2753609B1 (en) 2016-11-09
IL231235A (en) 2017-09-28
CU20140028A7 (es) 2014-05-27
US20150094346A1 (en) 2015-04-02
SG2014013114A (en) 2014-07-30
CU24303B1 (es) 2018-01-10
JO3192B1 (ar) 2018-03-08
US20180140582A1 (en) 2018-05-24
SI2753609T1 (sl) 2017-03-31
EP2753609A1 (en) 2014-07-16
CY1118585T1 (el) 2017-07-12
AR087787A1 (es) 2014-04-16
KR20140057382A (ko) 2014-05-12
AP3830A (en) 2016-09-30
US8933108B2 (en) 2015-01-13
AP2014007462A0 (en) 2014-02-28
CN103781771B (zh) 2016-08-24
HRP20170075T1 (hr) 2017-03-24
ZA201500790B (en) 2017-04-26
UA114295C2 (uk) 2017-05-25
US20150336914A1 (en) 2015-11-26
ZA201401112B (en) 2016-01-27
AU2013200422A1 (en) 2013-03-21
MY163301A (en) 2017-09-15
PH12014500399A1 (en) 2021-06-02
IL231235A0 (en) 2014-04-30
CN103781771A (zh) 2014-05-07
AU2013200422B2 (en) 2014-08-07
KR101628585B1 (ko) 2016-06-08
EA022909B1 (ru) 2016-03-31
TWI555738B (zh) 2016-11-01
US10251868B2 (en) 2019-04-09
HUE030530T2 (en) 2017-05-29
MX2014002688A (es) 2014-04-14
CN106187942A (zh) 2016-12-07
US20160279107A1 (en) 2016-09-29
EA201490573A1 (ru) 2014-06-30
ES2615052T3 (es) 2017-06-05
JP6130835B2 (ja) 2017-05-17
US20130245080A1 (en) 2013-09-19
DK2753609T3 (en) 2017-02-06
TN2014000060A1 (en) 2015-07-01
CR20140114A (es) 2014-05-06

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