GR3035925T3 - 1-(4,5-Dihydro-2-thiazolyle)-3-azetidine thiol derivatives - Google Patents

1-(4,5-Dihydro-2-thiazolyle)-3-azetidine thiol derivatives

Info

Publication number
GR3035925T3
GR3035925T3 GR20010400749T GR20010400749T GR3035925T3 GR 3035925 T3 GR3035925 T3 GR 3035925T3 GR 20010400749 T GR20010400749 T GR 20010400749T GR 20010400749 T GR20010400749 T GR 20010400749T GR 3035925 T3 GR3035925 T3 GR 3035925T3
Authority
GR
Greece
Prior art keywords
azetidine
thiazolyle
dihydro
thiol derivatives
compounds
Prior art date
Application number
GR20010400749T
Other languages
English (en)
Inventor
Kazuhiko Hayashi
Chisato Sato
Satoshi Tamai
Original Assignee
Lederle Japan Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lederle Japan Ltd filed Critical Lederle Japan Ltd
Publication of GR3035925T3 publication Critical patent/GR3035925T3/el

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D477/00Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring
    • C07D477/10Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D477/12Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6
    • C07D477/16Heterocyclic compounds containing 1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. carbapenicillins, thienamycins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulphur-containing hetero ring with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 4, and with a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2 with hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, attached in position 6 with hetero atoms or carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 3
    • C07D477/20Sulfur atoms
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D417/00Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Solid-Sorbent Or Filter-Aiding Compositions (AREA)
  • Processing Of Solid Wastes (AREA)
  • Chemical Vapour Deposition (AREA)
GR20010400749T 1994-12-12 2001-05-24 1-(4,5-Dihydro-2-thiazolyle)-3-azetidine thiol derivatives GR3035925T3 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP33142394 1994-12-12
JP25728195 1995-09-11

Publications (1)

Publication Number Publication Date
GR3035925T3 true GR3035925T3 (en) 2001-08-31

Family

ID=26543132

Family Applications (1)

Application Number Title Priority Date Filing Date
GR20010400749T GR3035925T3 (en) 1994-12-12 2001-05-24 1-(4,5-Dihydro-2-thiazolyle)-3-azetidine thiol derivatives

Country Status (15)

Country Link
US (1) US5659043A (el)
EP (1) EP0717042B1 (el)
KR (1) KR100337053B1 (el)
AT (1) ATE201410T1 (el)
AU (1) AU703119B2 (el)
CA (1) CA2164918C (el)
DE (1) DE69521012T2 (el)
DK (1) DK0717042T3 (el)
ES (1) ES2156917T3 (el)
FI (1) FI120402B (el)
GR (1) GR3035925T3 (el)
HU (4) HU223477B1 (el)
IL (1) IL116331A (el)
NO (1) NO955007L (el)
PT (1) PT717042E (el)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
KR100451670B1 (ko) * 2001-09-14 2004-10-08 한국화학연구원 내성균에 대해 항생작용을 갖는 카바페넴 유도체 및 이의제조방법
KR100621782B1 (ko) * 2004-06-14 2006-09-19 한국과학기술연구원 1-베타메틸카바페넴 유도체 및 이의 제조방법
CN102532139A (zh) * 2010-12-07 2012-07-04 重庆医药工业研究院有限责任公司 一种替比培南的制备方法
CN102731502B (zh) * 2011-04-13 2016-08-03 石药集团中奇制药技术(石家庄)有限公司 一种碳青霉烯抗生素的制备方法
CN102731503B (zh) * 2011-04-13 2016-02-03 石药集团中奇制药技术(石家庄)有限公司 一种泰比培南的制备方法
CN102250080B (zh) * 2011-04-26 2015-06-03 广州白云山制药股份有限公司广州白云山制药总厂 一种1-(4,5-二氢-2-噻唑啉基)-3-巯基吖丁叮盐酸盐的制备方法
CN102757430B (zh) * 2011-04-29 2016-04-13 上海医药工业研究院 一种替比培南的制备方法
CN104292222B (zh) * 2013-07-17 2017-05-10 常州锐博生物科技有限公司 一种替比培南匹伏酯侧链的新的合成方法
RU2766579C2 (ru) 2015-07-02 2022-03-15 ХОРАЙЗОН ОРФАН ЭлЭлСи Цистеаминдиоксигеназа-резистентные аналоги цистеамина и их применение
CN112321582B (zh) * 2020-11-03 2021-12-03 江西富祥药业股份有限公司 一种泰比培南侧链的合成及中间体的精制方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU682510B2 (en) * 1993-07-01 1997-10-09 Pfizer Japan Inc. 2-(1-(1,3-thiazolin-2-yl)azetidin-3-yl)thio-carbapenem derivatives

Also Published As

Publication number Publication date
AU4035995A (en) 1996-06-20
ATE201410T1 (de) 2001-06-15
ES2156917T3 (es) 2001-08-01
DK0717042T3 (da) 2001-08-06
HU223477B1 (hu) 2004-07-28
AU703119B2 (en) 1999-03-18
IL116331A (en) 2000-02-17
EP0717042A1 (en) 1996-06-19
DE69521012D1 (de) 2001-06-28
FI955954A0 (fi) 1995-12-12
DE69521012T2 (de) 2001-09-06
HU0203890D0 (en) 2003-01-28
CA2164918A1 (en) 1996-06-13
KR960022512A (ko) 1996-07-18
IL116331A0 (en) 1996-03-31
EP0717042B1 (en) 2001-05-23
HU0203891D0 (en) 2003-01-28
HUT75098A (en) 1997-04-28
US5659043A (en) 1997-08-19
CA2164918C (en) 2007-09-25
HU223472B1 (hu) 2004-07-28
FI120402B (fi) 2009-10-15
FI955954A (fi) 1996-06-13
NO955007L (no) 1996-06-13
HU223536B1 (hu) 2004-08-30
NO955007D0 (no) 1995-12-11
PT717042E (pt) 2001-08-30
HU223476B1 (hu) 2004-07-28
KR100337053B1 (ko) 2002-11-07
HU9503548D0 (en) 1996-02-28
HU0203892D0 (en) 2003-01-28

Similar Documents

Publication Publication Date Title
NO942483D0 (no) Carbapenem-antibiotika
AU1114792A (en) Pyranyl cyanoguanidine derivatives
GR3035925T3 (en) 1-(4,5-Dihydro-2-thiazolyle)-3-azetidine thiol derivatives
GR3024653T3 (en) Process for producing alpha-ketoamide derivative
DE60000402D1 (de) Prozess zur herstellung von zwischebprodukten für imidazodeazepinen
AU689459B2 (en) Process for the preparation of aminotriazine derivatives
BR8502884A (pt) Derivado de azetidina e processo para preparar acido azetidino-3-carboxilico
NZ332245A (en) Substituted benzo-oxazolol carboxylic acid derivatives, process for their production and medicaments containing them
HU0204401D0 (en) Process for producing 2,6-dichlorophenol derivatives
ATE244228T1 (de) Verfahren zur herstellung von chloroacetylaminothiazoleaceticsäure derivate