DE60000402D1 - Prozess zur herstellung von zwischebprodukten für imidazodeazepinen - Google Patents

Prozess zur herstellung von zwischebprodukten für imidazodeazepinen

Info

Publication number
DE60000402D1
DE60000402D1 DE60000402T DE60000402T DE60000402D1 DE 60000402 D1 DE60000402 D1 DE 60000402D1 DE 60000402 T DE60000402 T DE 60000402T DE 60000402 T DE60000402 T DE 60000402T DE 60000402 D1 DE60000402 D1 DE 60000402D1
Authority
DE
Germany
Prior art keywords
imidazodeacepines
production
intermediate products
compound
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
DE60000402T
Other languages
English (en)
Other versions
DE60000402T2 (de
Inventor
K Dhaon
Parvis Labib
A Davis
L Esser
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Abbott Laboratories
Original Assignee
Abbott Laboratories
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Abbott Laboratories filed Critical Abbott Laboratories
Application granted granted Critical
Publication of DE60000402D1 publication Critical patent/DE60000402D1/de
Publication of DE60000402T2 publication Critical patent/DE60000402T2/de
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
DE60000402T 1999-06-30 2000-06-15 Prozess zur herstellung von zwischebprodukten für imidazodeazepinen Expired - Fee Related DE60000402T2 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US09/343,317 US20010014738A1 (en) 1999-06-30 1999-06-30 Process for the preparation of imidazodiazepine intermediates
PCT/US2000/016476 WO2001000625A1 (en) 1999-06-30 2000-06-15 Process for the preparation of imidazodiazepine intermediates

Publications (2)

Publication Number Publication Date
DE60000402D1 true DE60000402D1 (de) 2002-10-10
DE60000402T2 DE60000402T2 (de) 2003-05-22

Family

ID=23345595

Family Applications (1)

Application Number Title Priority Date Filing Date
DE60000402T Expired - Fee Related DE60000402T2 (de) 1999-06-30 2000-06-15 Prozess zur herstellung von zwischebprodukten für imidazodeazepinen

Country Status (15)

Country Link
US (1) US20010014738A1 (de)
EP (2) EP1105392B1 (de)
JP (1) JP2003503410A (de)
KR (1) KR20010079706A (de)
CN (1) CN1315953A (de)
AT (1) ATE223414T1 (de)
AU (1) AU5874600A (de)
CA (1) CA2341524A1 (de)
DE (1) DE60000402T2 (de)
DK (1) DK1105392T3 (de)
ES (1) ES2185599T3 (de)
HK (1) HK1037617A1 (de)
IL (1) IL141394A0 (de)
PT (1) PT1105392E (de)
WO (1) WO2001000625A1 (de)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0211350D0 (en) 2002-05-16 2002-06-26 Rolls Royce Plc A gas turbine engine
IL156606A (en) 2003-06-23 2011-07-31 Aviad Kipnis Digital certificates
IT1399764B1 (it) * 2010-05-04 2013-05-03 F S I Fabbrica Italiana Sint Procedimento per la sintesi di 4h-imidazo [1,5-a][1,4]benzodiazepine, in particolare di midazolam.
CN103086986B (zh) * 2011-11-01 2015-11-04 上海医药工业研究院 1,4-苯二氮卓-n-亚硝胺类中间体的制备方法及其应用
CN103319486B (zh) * 2012-03-22 2017-10-10 徐州市心血管病研究所 合成4H‑咪唑并[1,5‑a][1,4]苯二氮卓,特别是咪达唑仑的方法
CN106032381A (zh) * 2015-03-16 2016-10-19 王志训 一种咪达唑仑衍生物的工业制造方法
CN106032380A (zh) * 2015-03-16 2016-10-19 王志训 一种咪达唑仑的工业制造方法
WO2018035246A1 (en) 2016-08-16 2018-02-22 Uwm Research Foundation, Inc. Gaba(a) receptor modulators and methods to control airway hyperresponsiveness and inflammation in asthma

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4440685A (en) * 1974-09-11 1984-04-03 Hoffmann-La Roche Inc. Imidazodiazepines and processes therefor
US4307237A (en) * 1974-09-11 1981-12-22 Hoffmann-La Roche Inc. Imidazoles
US4335042A (en) * 1980-04-21 1982-06-15 Hoffmann-La Roche Inc. Process to produce imidazobenzodiazepine intermediates

Also Published As

Publication number Publication date
ATE223414T1 (de) 2002-09-15
ES2185599T3 (es) 2003-05-01
DE60000402T2 (de) 2003-05-22
CN1315953A (zh) 2001-10-03
CA2341524A1 (en) 2001-01-04
JP2003503410A (ja) 2003-01-28
KR20010079706A (ko) 2001-08-22
PT1105392E (pt) 2002-12-31
HK1037617A1 (en) 2002-02-15
EP1105392A1 (de) 2001-06-13
AU5874600A (en) 2001-01-31
WO2001000625A1 (en) 2001-01-04
EP1199308A3 (de) 2002-05-02
EP1105392B1 (de) 2002-09-04
EP1199308A2 (de) 2002-04-24
DK1105392T3 (da) 2002-12-30
IL141394A0 (en) 2002-03-10
US20010014738A1 (en) 2001-08-16

Similar Documents

Publication Publication Date Title
ATE300528T1 (de) Synthese von cannabinoiden
DE602004024798D1 (de) Herstellung von quetiapin
ES2182061T3 (es) 1 - (2 - desoxi - 2 - fluor-4- tio-beta-d arabinofuranosil)citosina.
DE60000402D1 (de) Prozess zur herstellung von zwischebprodukten für imidazodeazepinen
NO894349D0 (no) Tienopyridin-type mevalonolaktoner.
PT829473E (pt) Processos para a preparacao de compostos ciclicos
PT1206452E (pt) Processo de preparacao de compostos benzoper-hidroisoindole
FI955954A (fi) Thiolyhdisteitä
BR0214445B1 (pt) processos para a produção de compostos.
DE60116201D1 (de) Verfahren zur Herstellung von Cephalosporin-Verbindungen und Zwischenprodukte für die Synthese dieser Verbindungen
ATE325159T1 (de) Verfahren zur herstellung von synergistischen stabilisatorgemischen
DE60112241D1 (de) Verfahren und zwischenverbindungen zur herstellung von imidazopyridinen
ATE247641T1 (de) Pyridin-zwischenprodukte, verwendbar zur herstellung von beta-adrenergischen rezeptor- agonisten
DK0439058T3 (da) Acycliske terpener
ATE348815T1 (de) Synthese von zwischenprodukten zur herstellung von tricyclischen verbindungen
DE50312447D1 (de) Verfahren zur herstellung von 4,6-dichlor-5-fluorpyrimidin
DE60127979D1 (de) Verfahren zur herstellung von 3,5-bisalkylphenolen
TW200420553A (en) Process for the synthesis of 3, 3a, 6, 6a-tetrahydro-2H-cyclopentan[b]furan-2-one
ATE244228T1 (de) Verfahren zur herstellung von chloroacetylaminothiazoleaceticsäure derivate
HU0001287D0 (en) New intermediate and process for its production
DE69816095D1 (de) Herstellung von beta-mehtylcarbapenem-zwischenprodukten

Legal Events

Date Code Title Description
8364 No opposition during term of opposition
8339 Ceased/non-payment of the annual fee