GB902703A - Penicillins - Google Patents
PenicillinsInfo
- Publication number
- GB902703A GB902703A GB29345/60A GB2934560A GB902703A GB 902703 A GB902703 A GB 902703A GB 29345/60 A GB29345/60 A GB 29345/60A GB 2934560 A GB2934560 A GB 2934560A GB 902703 A GB902703 A GB 902703A
- Authority
- GB
- United Kingdom
- Prior art keywords
- penicillanic acid
- acid
- amino
- aminophenylacetamido
- pencillin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 150000002960 penicillins Chemical class 0.000 title abstract 2
- 229930182555 Penicillin Natural products 0.000 title 1
- 150000003839 salts Chemical class 0.000 abstract 2
- NGHVIOIJCVXTGV-ALEPSDHESA-N 6-aminopenicillanic acid Chemical compound [O-]C(=O)[C@H]1C(C)(C)S[C@@H]2[C@H]([NH3+])C(=O)N21 NGHVIOIJCVXTGV-ALEPSDHESA-N 0.000 abstract 1
- NGHVIOIJCVXTGV-UHFFFAOYSA-N 6beta-amino-penicillanic acid Natural products OC(=O)C1C(C)(C)SC2C(N)C(=O)N21 NGHVIOIJCVXTGV-UHFFFAOYSA-N 0.000 abstract 1
- 125000003277 amino group Chemical group 0.000 abstract 1
- AVKUERGKIZMTKX-NJBDSQKTSA-N ampicillin Chemical compound C1([C@@H](N)C(=O)N[C@H]2[C@H]3SC([C@@H](N3C2=O)C(O)=O)(C)C)=CC=CC=C1 AVKUERGKIZMTKX-NJBDSQKTSA-N 0.000 abstract 1
- 238000009903 catalytic hydrogenation reaction Methods 0.000 abstract 1
- 230000008878 coupling Effects 0.000 abstract 1
- 238000010168 coupling process Methods 0.000 abstract 1
- 238000005859 coupling reaction Methods 0.000 abstract 1
- 230000006378 damage Effects 0.000 abstract 1
- 231100000252 nontoxic Toxicity 0.000 abstract 1
- 230000003000 nontoxic effect Effects 0.000 abstract 1
- 125000006239 protecting group Chemical group 0.000 abstract 1
- UQDJGEHQDNVPGU-UHFFFAOYSA-N serine phosphoethanolamine Chemical compound [NH3+]CCOP([O-])(=O)OCC([NH3+])C([O-])=O UQDJGEHQDNVPGU-UHFFFAOYSA-N 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
- C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
- C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
- C07D499/64—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms
- C07D499/68—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms with aromatic rings as additional substituents on the carbon chain
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
- C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Priority Applications (8)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB29345/60A GB902703A (en) | 1960-08-25 | 1960-08-25 | Penicillins |
| SE539061A SE219929C1 (enrdf_load_stackoverflow) | 1960-08-25 | 1961-05-23 | |
| BE604187A BE604187R (fr) | 1960-08-25 | 1961-05-25 | Perfectionnements apportés aux dérivés de la pénicilline |
| CH638961A CH407126A (de) | 1958-10-06 | 1961-06-01 | Verfahren zur Herstellung von epimeren a-Amino-benzylpenicillinen |
| ES0267993A ES267993A2 (es) | 1960-08-25 | 1961-06-05 | Procedimiento para la preparaciën de derivados penicilinicos de la fërmula general: |
| FR863883A FR12F (fr) | 1958-10-06 | 1961-06-05 | Dérivés de la pénicilline et leur procédé de préparation. |
| DK340861AA DK128166B (da) | 1960-08-25 | 1961-08-25 | Fremgangsmåde til fremstilling af 6-(D(-)-α-aminophenylacetamido) penicillansyre eller et salte deraf. |
| OA50918A OA060E (enrdf_load_stackoverflow) | 1960-08-25 | 1964-12-18 |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB29345/60A GB902703A (en) | 1960-08-25 | 1960-08-25 | Penicillins |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| GB902703A true GB902703A (en) | 1962-08-09 |
Family
ID=10290076
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| GB29345/60A Expired GB902703A (en) | 1958-10-06 | 1960-08-25 | Penicillins |
Country Status (6)
| Country | Link |
|---|---|
| BE (1) | BE604187R (enrdf_load_stackoverflow) |
| DK (1) | DK128166B (enrdf_load_stackoverflow) |
| ES (1) | ES267993A2 (enrdf_load_stackoverflow) |
| GB (1) | GB902703A (enrdf_load_stackoverflow) |
| OA (1) | OA060E (enrdf_load_stackoverflow) |
| SE (1) | SE219929C1 (enrdf_load_stackoverflow) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1208302B (de) * | 1962-08-28 | 1966-01-05 | Novo Terapeutisk Labor As | Verfahren zur Herstellung von D(-)- und L(ú½)-alpha-Aminobenzylpenicillin |
| US6544991B2 (en) | 2000-06-30 | 2003-04-08 | Pharmacia & Upjohn Company | Compositions and methods for treating bacterial infections |
-
1960
- 1960-08-25 GB GB29345/60A patent/GB902703A/en not_active Expired
-
1961
- 1961-05-23 SE SE539061A patent/SE219929C1/sv unknown
- 1961-05-25 BE BE604187A patent/BE604187R/fr active
- 1961-06-05 ES ES0267993A patent/ES267993A2/es not_active Expired
- 1961-08-25 DK DK340861AA patent/DK128166B/da unknown
-
1964
- 1964-12-18 OA OA50918A patent/OA060E/xx unknown
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE1208302B (de) * | 1962-08-28 | 1966-01-05 | Novo Terapeutisk Labor As | Verfahren zur Herstellung von D(-)- und L(ú½)-alpha-Aminobenzylpenicillin |
| US6544991B2 (en) | 2000-06-30 | 2003-04-08 | Pharmacia & Upjohn Company | Compositions and methods for treating bacterial infections |
Also Published As
| Publication number | Publication date |
|---|---|
| DK128166B (da) | 1974-03-11 |
| SE219929C1 (enrdf_load_stackoverflow) | 1968-04-09 |
| OA060E (enrdf_load_stackoverflow) | 1970-12-15 |
| BE604187R (fr) | 1961-09-18 |
| ES267993A2 (es) | 1961-10-16 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| GB1241844A (en) | Penicillins | |
| ES299038A1 (es) | Procedimiento de preparaciën de nuevas penicilinas | |
| CH385211A (de) | Verfahren zur Herstellung von am Iminostickstoff substituierten 2-Imino-1,3-di-N-heterocyclen | |
| GB902703A (en) | Penicillins | |
| PL238200A1 (en) | Process for preparing novel penicillins | |
| ES464000A1 (es) | Un procedimiento para preparar nuevas beta-lactamas monoci- clicas con actividad antibacteriana. | |
| ES8500957A1 (es) | Un procedimiento para preparar compuestos de cefalosporina. | |
| ES402674A1 (es) | Procedimiento para la preparacion de agentes antibacteria- nos. | |
| NL241461A (nl) | Werkwijze ter bereiding van alkalimetaalzouten van 1,2,5-thiadiazool 3,4-dicarbonzuur | |
| DK110173C (da) | Fremgangsmåde til fremstilling af 6-amino-penicillansyrederivater. | |
| GB965377A (en) | Penicillin derivatives | |
| GB894457A (en) | Improvements in or relating to penicillin derivatives | |
| GB940488A (en) | Penicillins | |
| ES395083A1 (es) | Un procedimiento para la preparacion de los acidos 7-(d- (alfa-amino-alfa-fenila-cetamido))-3-cefem-4-carboxilicos 3 - sustituidos. | |
| GB874414A (en) | Antibacterial agents | |
| GB1048907A (en) | Penicillins | |
| GB1267936A (en) | DERIVATIVES OF alpha-AMINOPENICILLINS | |
| OA01036A (fr) | Procédé de préparation de pénicillines et de leurs sels non toxiques. | |
| FI40539C (fi) | Menetelmä penisilliinien ja niiden myrkyttömien suolojen valmistamiseksi | |
| GB1030759A (en) | Penicillins | |
| GB894247A (en) | Antibacterial agents | |
| CA599513A (en) | Method for purification of glutamic acid | |
| GB1315443A (en) | Penicillins | |
| JPS5231088A (en) | Novel method of synthesis of penicillin derivatives | |
| JPS5481202A (en) | Elimination of protecting group |