ES402674A1 - Procedimiento para la preparacion de agentes antibacteria- nos. - Google Patents

Procedimiento para la preparacion de agentes antibacteria- nos.

Info

Publication number
ES402674A1
ES402674A1 ES402674A ES402674A ES402674A1 ES 402674 A1 ES402674 A1 ES 402674A1 ES 402674 A ES402674 A ES 402674A ES 402674 A ES402674 A ES 402674A ES 402674 A1 ES402674 A1 ES 402674A1
Authority
ES
Spain
Prior art keywords
formula
preparation
antibacterial agents
blocking group
dales
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES402674A
Other languages
English (en)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
R&L Molecular Research Ltd
Original Assignee
R&L Molecular Research Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by R&L Molecular Research Ltd filed Critical R&L Molecular Research Ltd
Publication of ES402674A1 publication Critical patent/ES402674A1/es
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/44—Iso-indoles; Hydrogenated iso-indoles
    • C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C247/00—Compounds containing azido groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
    • C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
    • C07D249/04—1,2,3-Triazoles; Hydrogenated 1,2,3-triazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/06—1,2,3-Thiadiazoles; Hydrogenated 1,2,3-thiadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
    • C07D285/01—Five-membered rings
    • C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
    • C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
    • C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
    • C07D285/125—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Cephalosporin Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Un procedimiento para la preparación de agentes antibacterianos de fórmula **fórmula** donde n es 0 o 1 y R representa **fórmula** y sus dales no tóxicas y farmacéuticamente aceptables, cuyo procedimiento consiste en hacer reaccionar un compuesto de fórmula**fórmula** **fórmula** don R es el definido anteriormente, o una sal o un éster fácilmente hidrolizable del mismo, con un ácido de fórmula **fórmula** donde B es un grupo bloqueante y n es el descrito anteriormente o con su equivalente funcional como agente acilante de un grupo amino primario y posteriormente separar dicho grupo bloqueante.
ES402674A 1971-05-11 1972-05-12 Procedimiento para la preparacion de agentes antibacteria- nos. Expired ES402674A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US14233871A 1971-05-11 1971-05-11
US14233771A 1971-05-11 1971-05-11

Publications (1)

Publication Number Publication Date
ES402674A1 true ES402674A1 (es) 1975-10-16

Family

ID=26840005

Family Applications (1)

Application Number Title Priority Date Filing Date
ES402674A Expired ES402674A1 (es) 1971-05-11 1972-05-12 Procedimiento para la preparacion de agentes antibacteria- nos.

Country Status (16)

Country Link
JP (1) JPS523390B1 (es)
AR (1) AR193397A1 (es)
AU (1) AU456536B2 (es)
BE (1) BE783223A (es)
CH (1) CH569023A5 (es)
DD (1) DD98933A5 (es)
DK (1) DK137192B (es)
ES (1) ES402674A1 (es)
FR (1) FR2137792B1 (es)
GB (1) GB1392241A (es)
HU (1) HU165964B (es)
IE (1) IE36346B1 (es)
IL (1) IL39388A (es)
NL (1) NL7206326A (es)
SE (1) SE390172B (es)
YU (1) YU36035B (es)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7311757A (es) * 1972-08-30 1974-03-04
KR780000197B1 (en) * 1972-12-26 1978-05-26 Bristol Myers Co Method for preparing antibacterial agent
US3910899A (en) * 1973-09-07 1975-10-07 Bristol Myers Co 7-(2-Aminomethylphenyl-acetamido)-3-{8 2-(5-hydroxymethyl-1,3,4-thiadiazolyl)-thiomethyl{9 -3-cephem-4-carboxylic acid
KR20040014498A (ko) * 2001-04-19 2004-02-14 바이오퍼마 무르시아, 에스.에이. 세팔로스포린 유도체의 제조 방법

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US382241A (en) * 1888-05-01 William e
NL7103331A (es) * 1970-03-13 1971-09-15

Also Published As

Publication number Publication date
FR2137792B1 (es) 1976-04-16
NL7206326A (es) 1972-11-14
SU440842A3 (es) 1974-08-25
DD98933A5 (es) 1973-07-12
AR193397A1 (es) 1973-04-23
IE36346L (en) 1972-11-11
DK137192B (da) 1978-01-30
YU36035B (en) 1981-11-13
IL39388A0 (en) 1972-07-26
DE2222954A1 (de) 1973-03-08
YU123772A (en) 1981-04-30
GB1392241A (en) 1975-04-30
IL39388A (en) 1975-02-10
JPS523390B1 (es) 1977-01-27
HU165964B (es) 1974-12-28
DE2222954B2 (de) 1975-07-10
BE783223A (fr) 1972-11-09
AU4187772A (en) 1973-11-08
SE390172B (sv) 1976-12-06
AU456536B2 (en) 1974-12-19
FR2137792A1 (es) 1972-12-29
DK137192C (es) 1978-07-03
CH569023A5 (es) 1975-11-14
IE36346B1 (en) 1976-10-13

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