FR2559152B1 - Nouveaux derives de la furo-(3,4-c)-pyridine substitues en position 6, ainsi que leur procede de preparation - Google Patents
Nouveaux derives de la furo-(3,4-c)-pyridine substitues en position 6, ainsi que leur procede de preparationInfo
- Publication number
- FR2559152B1 FR2559152B1 FR8501401A FR8501401A FR2559152B1 FR 2559152 B1 FR2559152 B1 FR 2559152B1 FR 8501401 A FR8501401 A FR 8501401A FR 8501401 A FR8501401 A FR 8501401A FR 2559152 B1 FR2559152 B1 FR 2559152B1
- Authority
- FR
- France
- Prior art keywords
- furo
- well
- preparation process
- novel derivatives
- pyridine substituted
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Psychiatry (AREA)
- Medicinal Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pyridine Compounds (AREA)
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB848402740A GB8402740D0 (en) | 1984-02-02 | 1984-02-02 | Furo-(3 4-c)-pyridine derivatives |
Publications (2)
Publication Number | Publication Date |
---|---|
FR2559152A1 FR2559152A1 (fr) | 1985-08-09 |
FR2559152B1 true FR2559152B1 (fr) | 1987-05-22 |
Family
ID=10555953
Family Applications (2)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR8501402A Expired FR2559062B1 (fr) | 1984-02-02 | 1985-02-01 | Medicaments a base de nouveaux derives 6-substitues de la furo-(3,4-c)-pyridine |
FR8501401A Expired FR2559152B1 (fr) | 1984-02-02 | 1985-02-01 | Nouveaux derives de la furo-(3,4-c)-pyridine substitues en position 6, ainsi que leur procede de preparation |
Family Applications Before (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
FR8501402A Expired FR2559062B1 (fr) | 1984-02-02 | 1985-02-01 | Medicaments a base de nouveaux derives 6-substitues de la furo-(3,4-c)-pyridine |
Country Status (24)
Country | Link |
---|---|
US (1) | US4581362A (fr) |
JP (1) | JPS60181088A (fr) |
AT (1) | AT391700B (fr) |
BE (1) | BE901545A (fr) |
CA (1) | CA1300148C (fr) |
CH (1) | CH663023A5 (fr) |
DE (1) | DE3503435A1 (fr) |
DK (1) | DK158951C (fr) |
DZ (1) | DZ743A1 (fr) |
ES (1) | ES8607308A1 (fr) |
FI (1) | FI82051C (fr) |
FR (2) | FR2559062B1 (fr) |
GB (1) | GB8402740D0 (fr) |
HK (1) | HK92587A (fr) |
IE (1) | IE58229B1 (fr) |
IT (1) | IT1200587B (fr) |
LU (1) | LU85744A1 (fr) |
MA (1) | MA20342A1 (fr) |
NL (1) | NL8500241A (fr) |
NO (1) | NO160369C (fr) |
OA (1) | OA07947A (fr) |
PT (1) | PT79913B (fr) |
SE (2) | SE8500460L (fr) |
ZA (1) | ZA85508B (fr) |
Families Citing this family (25)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB8427218D0 (en) * | 1984-10-27 | 1984-12-05 | Scras | Pyridine derivatives |
GB8808001D0 (en) * | 1988-04-06 | 1988-05-05 | Scras | Stereospecific preparative process for furol(3,4-c)pyridine derivatives |
GB8907480D0 (en) * | 1989-04-03 | 1989-05-17 | Scaras Societe De Conseils De | Separation of insomers of furo(3,4-c)pyridine derivatives |
US5130252A (en) * | 1990-05-14 | 1992-07-14 | Synthetech, Inc. | Resolution of furopyridine enantiomers and synthetic precursors thereof |
JPH054664A (ja) * | 1991-06-21 | 1993-01-14 | Yoozuri:Kk | 運搬等用の包装体及び包装方法 |
CN104135859B (zh) | 2011-12-28 | 2017-06-27 | 全球血液疗法公司 | 取代的苯甲醛化合物及其用于增加组织氧合的方法 |
US9012450B2 (en) | 2011-12-28 | 2015-04-21 | Global Blood Therapeutics, Inc. | Substituted heteroaryl aldehyde compounds and methods for their use in increasing tissue oxygenation |
PE20160078A1 (es) | 2013-03-15 | 2016-03-02 | Global Blood Therapeutics Inc | Compuestos y sus usos para modular la hemoglobina |
US10100043B2 (en) | 2013-03-15 | 2018-10-16 | Global Blood Therapeutics, Inc. | Substituted aldehyde compounds and methods for their use in increasing tissue oxygenation |
US9422279B2 (en) | 2013-03-15 | 2016-08-23 | Global Blood Therapeutics, Inc. | Compounds and uses thereof for the modulation of hemoglobin |
US20140274961A1 (en) | 2013-03-15 | 2014-09-18 | Global Blood Therapeutics, Inc. | Compounds and uses thereof for the modulation of hemoglobin |
US10266551B2 (en) | 2013-03-15 | 2019-04-23 | Global Blood Therapeutics, Inc. | Compounds and uses thereof for the modulation of hemoglobin |
US9802900B2 (en) | 2013-03-15 | 2017-10-31 | Global Blood Therapeutics, Inc. | Bicyclic heteroaryl compounds and uses thereof for the modulation of hemoglobin |
US8952171B2 (en) | 2013-03-15 | 2015-02-10 | Global Blood Therapeutics, Inc. | Compounds and uses thereof for the modulation of hemoglobin |
AP2015008721A0 (en) | 2013-03-15 | 2015-09-30 | Global Blood Therapeutics Inc | Compounds and uses thereof for the modulation of hemoglobin |
US9458139B2 (en) | 2013-03-15 | 2016-10-04 | Global Blood Therapeutics, Inc. | Compounds and uses thereof for the modulation of hemoglobin |
MY183637A (en) | 2013-03-15 | 2021-03-04 | Global Blood Therapeutics Inc | Compounds and uses thereof for the modulation of hemoglobin |
US9604999B2 (en) | 2013-03-15 | 2017-03-28 | Global Blood Therapeutics, Inc. | Compounds and uses thereof for the modulation of hemoglobin |
EA201992707A1 (ru) | 2013-11-18 | 2020-06-30 | Глобал Блад Терапьютикс, Инк. | Соединения и их применения для модуляции гемоглобина |
PT3102208T (pt) | 2014-02-07 | 2021-04-05 | Global Blood Therapeutics Inc | Polimorfos cristalinos da base livre de 2-hidroxi-6-((2-(1-isopropil-1h-pirazol-5-il)piridin-3 il)metoxi)benzaldeído |
MA41841A (fr) | 2015-03-30 | 2018-02-06 | Global Blood Therapeutics Inc | Composés aldéhyde pour le traitement de la fibrose pulmonaire, de l'hypoxie, et de maladies auto-immunes et des tissus conjonctifs |
TW201731509A (zh) | 2015-12-04 | 2017-09-16 | 全球血液治療公司 | 針對2-羥基-6-((2-(1-異丙基-1h-吡唑-5-基)吡啶-3-基)甲氧基)-苯甲醛之劑量方案 |
AR108435A1 (es) | 2016-05-12 | 2018-08-22 | Global Blood Therapeutics Inc | Proceso para sintetizar 2-hidroxi-6-((2-(1-isopropil-1h-pirazol-5-il)-piridin-3-il)metoxi)benzaldehído |
TW202332423A (zh) | 2016-10-12 | 2023-08-16 | 美商全球血液治療公司 | 包含2-羥基-6-((2-(1-異丙基-1h-吡唑-5-基)吡啶-3-基)甲氧基)-苯甲醛之片劑 |
US11014884B2 (en) | 2018-10-01 | 2021-05-25 | Global Blood Therapeutics, Inc. | Modulators of hemoglobin |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
ZA786269B (en) * | 1977-11-25 | 1979-10-31 | Scras | New pyridine derivative,its preparation and use |
IN156817B (fr) * | 1981-02-10 | 1985-11-09 | Scras | |
GB8330517D0 (en) * | 1983-11-16 | 1983-12-21 | Scras | 6-vinyl-furo-(3,4-c)pyridine derivatives |
GB8330658D0 (en) * | 1983-11-17 | 1983-12-29 | Scras | 7-carboxymethoxy-furo-(3,4-c)-pyridine derivatives |
-
1984
- 1984-02-02 GB GB848402740A patent/GB8402740D0/en active Pending
-
1985
- 1985-01-22 FI FI850275A patent/FI82051C/fi not_active IP Right Cessation
- 1985-01-22 ZA ZA85508A patent/ZA85508B/xx unknown
- 1985-01-22 BE BE0/214370A patent/BE901545A/fr not_active IP Right Cessation
- 1985-01-23 US US06/693,715 patent/US4581362A/en not_active Expired - Lifetime
- 1985-01-24 CH CH312/85A patent/CH663023A5/fr not_active IP Right Cessation
- 1985-01-25 LU LU85744A patent/LU85744A1/fr unknown
- 1985-01-26 DZ DZ850024A patent/DZ743A1/fr active
- 1985-01-29 NL NL8500241A patent/NL8500241A/nl not_active Application Discontinuation
- 1985-01-31 AT AT0027585A patent/AT391700B/de not_active IP Right Cessation
- 1985-01-31 CA CA000473302A patent/CA1300148C/fr not_active Expired - Fee Related
- 1985-01-31 OA OA58520A patent/OA07947A/fr unknown
- 1985-02-01 JP JP60016713A patent/JPS60181088A/ja active Granted
- 1985-02-01 PT PT79913A patent/PT79913B/pt not_active IP Right Cessation
- 1985-02-01 DE DE19853503435 patent/DE3503435A1/de active Granted
- 1985-02-01 IE IE24185A patent/IE58229B1/en not_active IP Right Cessation
- 1985-02-01 FR FR8501402A patent/FR2559062B1/fr not_active Expired
- 1985-02-01 DK DK045585A patent/DK158951C/da not_active IP Right Cessation
- 1985-02-01 FR FR8501401A patent/FR2559152B1/fr not_active Expired
- 1985-02-01 SE SE8500460D patent/SE8500460L/xx not_active Application Discontinuation
- 1985-02-01 ES ES540080A patent/ES8607308A1/es not_active Expired
- 1985-02-01 MA MA20566A patent/MA20342A1/fr unknown
- 1985-02-01 SE SE8500460A patent/SE460903B/sv not_active IP Right Cessation
- 1985-02-01 NO NO850399A patent/NO160369C/no unknown
- 1985-02-01 IT IT19327/85A patent/IT1200587B/it active
-
1987
- 1987-12-03 HK HK925/87A patent/HK92587A/xx not_active IP Right Cessation
Also Published As
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
ST | Notification of lapse |