FR2439191A1 - Derives 2-amino ou 2-thio substitues de 4,5-diphenyloxazole et procede pour leur preparation - Google Patents
Derives 2-amino ou 2-thio substitues de 4,5-diphenyloxazole et procede pour leur preparationInfo
- Publication number
- FR2439191A1 FR2439191A1 FR7925705A FR7925705A FR2439191A1 FR 2439191 A1 FR2439191 A1 FR 2439191A1 FR 7925705 A FR7925705 A FR 7925705A FR 7925705 A FR7925705 A FR 7925705A FR 2439191 A1 FR2439191 A1 FR 2439191A1
- Authority
- FR
- France
- Prior art keywords
- amino
- diphenyloxazole
- preparation
- hydroxyalkyl
- thio derivatives
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- GOJUJUVQIVIZAV-UHFFFAOYSA-N 2-amino-4,6-dichloropyrimidine-5-carbaldehyde Chemical compound NC1=NC(Cl)=C(C=O)C(Cl)=N1 GOJUJUVQIVIZAV-UHFFFAOYSA-N 0.000 title abstract 2
- ODKHOKLXMBWVOQ-UHFFFAOYSA-N 4,5-diphenyl-1,3-oxazole Chemical compound O1C=NC(C=2C=CC=CC=2)=C1C1=CC=CC=C1 ODKHOKLXMBWVOQ-UHFFFAOYSA-N 0.000 title abstract 2
- 239000002253 acid Substances 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- SCVJRXQHFJXZFZ-KVQBGUIXSA-N 2-amino-9-[(2r,4s,5r)-4-hydroxy-5-(hydroxymethyl)oxolan-2-yl]-3h-purine-6-thione Chemical group C1=2NC(N)=NC(=S)C=2N=CN1[C@H]1C[C@H](O)[C@@H](CO)O1 SCVJRXQHFJXZFZ-KVQBGUIXSA-N 0.000 abstract 1
- -1 AMINO Chemical group 0.000 abstract 1
- OKTJSMMVPCPJKN-UHFFFAOYSA-N Carbon Chemical compound [C] OKTJSMMVPCPJKN-UHFFFAOYSA-N 0.000 abstract 1
- VEXZGXHMUGYJMC-UHFFFAOYSA-M Chloride anion Chemical compound [Cl-] VEXZGXHMUGYJMC-UHFFFAOYSA-M 0.000 abstract 1
- 150000007513 acids Chemical class 0.000 abstract 1
- 150000008064 anhydrides Chemical class 0.000 abstract 1
- 229910052799 carbon Inorganic materials 0.000 abstract 1
- 239000007858 starting material Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/46—Sulfur atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/30—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D263/34—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D263/48—Nitrogen atoms not forming part of a nitro radical
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Hematology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Steroid Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| IT28825/78A IT1099996B (it) | 1978-10-17 | 1978-10-17 | Derivati del 4,5-difenil-ossazolo 2-ammino o 2-tio sostituiti e procedimento per il loro ottenimento |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| FR2439191A1 true FR2439191A1 (fr) | 1980-05-16 |
| FR2439191B1 FR2439191B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1982-06-18 |
Family
ID=11224263
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FR7925705A Granted FR2439191A1 (fr) | 1978-10-17 | 1979-10-16 | Derives 2-amino ou 2-thio substitues de 4,5-diphenyloxazole et procede pour leur preparation |
Country Status (22)
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1099996B (it) * | 1978-10-17 | 1985-09-28 | Anic Spa | Derivati del 4,5-difenil-ossazolo 2-ammino o 2-tio sostituiti e procedimento per il loro ottenimento |
| GB2422782A (en) * | 2003-10-21 | 2006-08-09 | Inspire Pharmaceuticals Inc | Non-nucleotide compositions and method for treating pain |
| USD1012421S1 (en) | 2020-08-07 | 2024-01-30 | Zuru (Singapore) Pte. Ltd. | Confectionery |
| AU2020329071A1 (en) | 2019-08-09 | 2022-02-24 | Zuru (Singapore) Pte. Ltd. | Gummy confectionery-coated non-edible container |
Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1538009A (fr) * | 1966-08-10 | 1968-08-30 | Serono Ist Farm | 4, 5-diphényl-oxazols 2-amino-substitués et les procédés de préparation par synthèse propres à les obtenir |
| FR2281115A1 (fr) * | 1974-08-06 | 1976-03-05 | Serono Lab | Derives de 2-thiol-4,5-diphenyloxazole substitues sur le soufre et compositions les contenant |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CH506548A (de) * | 1966-08-10 | 1971-04-30 | Serono Ist Farm | Verfahren zur Herstellung von 2-aminsubstituiertem 4,5-Diphenyl-Oxazol |
| DE2129012A1 (de) * | 1971-06-11 | 1973-01-04 | Merck Patent Gmbh | Azol-derivate |
| DE2428249C3 (de) * | 1973-07-09 | 1978-12-14 | Serna Ag, Glarus (Schweiz) | Verfahren zur Herstellung von |
| GB1497536A (en) * | 1973-12-17 | 1978-01-12 | Lilly Industries Ltd | 2-acylaminooxazoles methods for their preparation and their use |
| IT1085524B (it) * | 1977-03-22 | 1985-05-28 | Snam Progetti | Materiali e fibre porose biocompatibili in grado di inglobare sostanze di interesse biologico e metodi per il loro ottenimento |
| IT1099996B (it) * | 1978-10-17 | 1985-09-28 | Anic Spa | Derivati del 4,5-difenil-ossazolo 2-ammino o 2-tio sostituiti e procedimento per il loro ottenimento |
-
1978
- 1978-10-17 IT IT28825/78A patent/IT1099996B/it active
-
1979
- 1979-10-11 AU AU51712/79A patent/AU533275B2/en not_active Ceased
- 1979-10-12 GB GB7935584A patent/GB2036006B/en not_active Expired
- 1979-10-15 LU LU81788A patent/LU81788A1/fr unknown
- 1979-10-15 NO NO793322A patent/NO793322L/no unknown
- 1979-10-15 SE SE7908532A patent/SE446533B/sv not_active IP Right Cessation
- 1979-10-15 YU YU2503/79A patent/YU41184B/xx unknown
- 1979-10-16 BE BE0/197669A patent/BE879440A/fr not_active IP Right Cessation
- 1979-10-16 DD DD79216260A patent/DD146598A5/de not_active IP Right Cessation
- 1979-10-16 CA CA000337867A patent/CA1122221A/en not_active Expired
- 1979-10-16 ZA ZA00795525A patent/ZA795525B/xx unknown
- 1979-10-16 FR FR7925705A patent/FR2439191A1/fr active Granted
- 1979-10-16 CH CH930179A patent/CH645364A5/it not_active IP Right Cessation
- 1979-10-16 IL IL58458A patent/IL58458A/xx unknown
- 1979-10-16 SU SU792834908A patent/SU982540A3/ru active
- 1979-10-16 JP JP13248079A patent/JPS5589271A/ja active Granted
- 1979-10-16 DK DK436879A patent/DK151880C/da active
- 1979-10-16 HU HU79EE2699A patent/HU181426B/hu not_active IP Right Cessation
- 1979-10-17 CS CS797044A patent/CS213305B2/cs unknown
- 1979-10-17 DE DE2942050A patent/DE2942050C2/de not_active Expired
- 1979-10-17 NL NL7907661A patent/NL7907661A/nl not_active Application Discontinuation
-
1983
- 1983-11-17 US US06/552,987 patent/US4591596A/en not_active Expired - Fee Related
Patent Citations (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| FR1538009A (fr) * | 1966-08-10 | 1968-08-30 | Serono Ist Farm | 4, 5-diphényl-oxazols 2-amino-substitués et les procédés de préparation par synthèse propres à les obtenir |
| FR2281115A1 (fr) * | 1974-08-06 | 1976-03-05 | Serono Lab | Derives de 2-thiol-4,5-diphenyloxazole substitues sur le soufre et compositions les contenant |
Non-Patent Citations (1)
| Title |
|---|
| EXBK/71 * |
Also Published As
| Publication number | Publication date |
|---|---|
| IL58458A (en) | 1983-06-15 |
| HU181426B (en) | 1983-07-28 |
| CA1122221A (en) | 1982-04-20 |
| YU250379A (en) | 1983-04-30 |
| DE2942050C2 (de) | 1986-12-04 |
| DK151880C (da) | 1988-06-06 |
| SE446533B (sv) | 1986-09-22 |
| JPH0231072B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1990-07-11 |
| NL7907661A (nl) | 1980-04-21 |
| GB2036006A (en) | 1980-06-25 |
| FR2439191B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) | 1982-06-18 |
| IT7828825A0 (it) | 1978-10-17 |
| AU5171279A (en) | 1980-04-24 |
| CS213305B2 (en) | 1982-04-09 |
| JPS5589271A (en) | 1980-07-05 |
| IL58458A0 (en) | 1980-01-31 |
| US4591596A (en) | 1986-05-27 |
| CH645364A5 (it) | 1984-09-28 |
| DK436879A (da) | 1980-04-18 |
| LU81788A1 (fr) | 1980-01-24 |
| GB2036006B (en) | 1983-01-06 |
| SE7908532L (sv) | 1980-04-18 |
| SU982540A3 (ru) | 1982-12-15 |
| ZA795525B (en) | 1980-10-29 |
| NO793322L (no) | 1980-04-18 |
| DD146598A5 (de) | 1981-02-18 |
| BE879440A (fr) | 1980-04-16 |
| YU41184B (en) | 1986-12-31 |
| DE2942050A1 (de) | 1980-04-24 |
| AU533275B2 (en) | 1983-11-17 |
| IT1099996B (it) | 1985-09-28 |
| DK151880B (da) | 1988-01-11 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| ST | Notification of lapse |