FR2360587A1 - Nouveaux derives d'amino-alcoyl-furannes utiles comme medicaments - Google Patents

Nouveaux derives d'amino-alcoyl-furannes utiles comme medicaments

Info

Publication number
FR2360587A1
FR2360587A1 FR7724021A FR7724021A FR2360587A1 FR 2360587 A1 FR2360587 A1 FR 2360587A1 FR 7724021 A FR7724021 A FR 7724021A FR 7724021 A FR7724021 A FR 7724021A FR 2360587 A1 FR2360587 A1 FR 2360587A1
Authority
FR
France
Prior art keywords
alcoyl
amino
medicinal products
new derivatives
furans
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
FR7724021A
Other languages
English (en)
Other versions
FR2360587B1 (fr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Allen and Hanburys Ltd
Original Assignee
Allen and Hanburys Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=27516213&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FR2360587(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Allen and Hanburys Ltd filed Critical Allen and Hanburys Ltd
Priority claimed from KR7701808A external-priority patent/KR810000355B1/ko
Publication of FR2360587A1 publication Critical patent/FR2360587A1/fr
Application granted granted Critical
Publication of FR2360587B1 publication Critical patent/FR2360587B1/fr
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/02—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings
    • C07D275/03—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings not condensed with other rings with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/34—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having five-membered rings with one oxygen as the only ring hetero atom, e.g. isosorbide
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/52—Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/56—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D307/64—Sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Furan Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

Abstract

L'invention concerne des nouveaux dérivés d'amino-alcoylfurannes. Il s'agit notamment de composés de formule générale :
FR7724021A 1976-08-04 1977-08-04 Nouveaux derives d'amino-alcoyl-furannes utiles comme medicaments Expired FR2360587B1 (fr)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
GB32465/76A GB1565966A (en) 1976-08-04 1976-08-04 Aminoalkyl furan derivatives
GB5068576 1976-12-06
GB2018777 1977-05-13
GB28187/78A GB1565967A (en) 1976-08-04 1977-07-22 Aminoalkyl furan derivatives
KR7701808A KR810000355B1 (ko) 1977-05-13 1977-08-04 아미노 알킬푸란 유도체의 제조방법

Publications (2)

Publication Number Publication Date
FR2360587A1 true FR2360587A1 (fr) 1978-03-03
FR2360587B1 FR2360587B1 (fr) 1981-07-17

Family

ID=27516213

Family Applications (3)

Application Number Title Priority Date Filing Date
FR7724021A Expired FR2360587B1 (fr) 1976-08-04 1977-08-04 Nouveaux derives d'amino-alcoyl-furannes utiles comme medicaments
FR7814250A Expired FR2384765B1 (fr) 1976-08-04 1978-05-12 Derives amino-substitues du furanne et procede pour leur preparation
FR7814251A Expired FR2384753B1 (fr) 1976-08-04 1978-05-12 Nouveaux thiols et leur procede de preparation

Family Applications After (2)

Application Number Title Priority Date Filing Date
FR7814250A Expired FR2384765B1 (fr) 1976-08-04 1978-05-12 Derives amino-substitues du furanne et procede pour leur preparation
FR7814251A Expired FR2384753B1 (fr) 1976-08-04 1978-05-12 Nouveaux thiols et leur procede de preparation

Country Status (10)

Country Link
US (3) US4128658A (fr)
JP (3) JPS5840956B2 (fr)
AU (1) AU515628B2 (fr)
BE (1) BE857388A (fr)
CA (1) CA1099268A (fr)
DE (1) DE2734070C2 (fr)
FR (3) FR2360587B1 (fr)
GB (2) GB1565966A (fr)
LU (1) LU77911A1 (fr)
NL (1) NL178320C (fr)

Cited By (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2391209A1 (fr) * 1977-05-17 1978-12-15 Allen & Hanburys Ltd Aminoalkyl thiophenes, utiles comme medicaments, leur preparation et compositions en contenant
FR2437409A1 (fr) * 1978-09-26 1980-04-25 Bristol Myers Co Furannes substitues, leur procede de production et medicament les contenant
EP0060182A1 (fr) * 1981-03-11 1982-09-15 Sanofi S.A. Thioalkylamide de l'acide nicotinique 1-oxyde, ses sels, procédé pour leur préparation et compositions pharmaceutiques
FR2537582A1 (fr) * 1982-12-08 1984-06-15 Degussa Nouveaux derives de l'ethylene-diamine et de la guanidine
FR2547727A1 (fr) * 1983-05-13 1984-12-28 Glaxo Group Ltd Compositions pharmaceutiques
EP0571575A1 (fr) * 1991-11-15 1993-12-01 Baxter International Inc. Formulation de ranitidine premelangee non tamponnee

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* Cited by examiner, † Cited by third party
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US5021429A (en) * 1977-05-17 1991-06-04 Allen & Hansburys Limited Pharmacologically active aminoalkylphenyl compounds and their use
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JPS5461167A (en) * 1977-10-11 1979-05-17 Glaxo Group Ltd Novel substituted heterocyclic compounds* their manufacture and medical composition containing them
US4233302A (en) * 1977-12-23 1980-11-11 Glaxo Group Limited Amine derivatives and pharmaceutical compositions containing them
IN151188B (fr) * 1978-02-13 1983-03-05 Smith Kline French Lab
US4539207A (en) * 1978-02-13 1985-09-03 Smith Kline & French Laboratories Limited Pyrimidine compounds
AR228941A1 (es) 1978-04-26 1983-05-13 Glaxo Group Ltd Procedimiento para preparar nuevos derivados de 3,5-diamino-1,2,4-triazol que son activos contra receptores histaminicos
US4405624A (en) * 1978-05-30 1983-09-20 Smith Kline & French Laboratories Limited Nitro-substituted dihydropyrroles and tetrahydropyridines, compositions, compounds, and medicinal use
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IL57415A (en) * 1978-05-30 1984-08-31 Smith Kline French Lab Nitropyrrole compounds,process for preparing them and pharmaceutical compositions containing them
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US4282363A (en) * 1978-11-24 1981-08-04 Bristol-Myers Company 1-Nitro-2-(2-alkynylamino)-2-[(2-pyridylmethylthio)-ethylamino]ethylene derivatives
DE3067920D1 (en) * 1979-03-02 1984-06-28 Glaxo Group Ltd 1,2,4-triazole derivatives, processes for their production and pharmaceutical compositions containing them
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US4431802A (en) * 1979-12-10 1984-02-14 G. D. Searle & Co. N-Heterocyclyl-N-cyano-N-(heterocyclythioalkyl)-guanidines
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FR2384765A1 (fr) 1978-10-20
FR2384753A1 (fr) 1978-10-20
DE2734070C2 (de) 1983-12-29
FR2360587B1 (fr) 1981-07-17
FR2384753B1 (fr) 1981-06-12
LU77911A1 (fr) 1979-05-23
DE2734070A1 (de) 1978-02-09
JPS6132315B2 (fr) 1986-07-25
CA1099268A (fr) 1981-04-14
GB1565966A (en) 1980-04-23
NL178320C (nl) 1986-03-03
US4255440A (en) 1981-03-10
NL7708601A (nl) 1978-02-07
FR2384765B1 (fr) 1982-09-10
JPS5840956B2 (ja) 1983-09-08
AU2751977A (en) 1979-02-08
AU515628B2 (en) 1981-04-16
BE857388A (fr) 1978-02-02
US4279819A (en) 1981-07-21
GB1565967A (en) 1980-04-23
JPS55153779A (en) 1980-11-29
US4128658A (en) 1978-12-05
JPS55153761A (en) 1980-11-29
JPS5318557A (en) 1978-02-20

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