FI943775A0 - Hypolipideemiset bentsotiatsepiiniyhdisteet - Google Patents

Hypolipideemiset bentsotiatsepiiniyhdisteet

Info

Publication number
FI943775A0
FI943775A0 FI943775A FI943775A FI943775A0 FI 943775 A0 FI943775 A0 FI 943775A0 FI 943775 A FI943775 A FI 943775A FI 943775 A FI943775 A FI 943775A FI 943775 A0 FI943775 A0 FI 943775A0
Authority
FI
Finland
Prior art keywords
integer
pct
alkyl
phenylalkoxy
alkoxy
Prior art date
Application number
FI943775A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI943775A7 (fi
FI943775L (fi
Inventor
Lawrence Edward Brieaddy
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of FI943775A7 publication Critical patent/FI943775A7/fi
Publication of FI943775L publication Critical patent/FI943775L/fi
Publication of FI943775A0 publication Critical patent/FI943775A0/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D281/00Heterocyclic compounds containing rings of more than six members having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D281/02Seven-membered rings
    • C07D281/04Seven-membered rings having the hetero atoms in positions 1 and 4
    • C07D281/08Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D281/10Seven-membered rings having the hetero atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Thiazole And Isothizaole Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Saccharide Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Hydrogenated Pyridines (AREA)
  • Steroid Compounds (AREA)
FI943775A 1992-02-17 1993-02-16 Hypolipideemiset bentsotiatsepiiniyhdisteet FI943775A0 (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB929203347A GB9203347D0 (en) 1992-02-17 1992-02-17 Hypolipidaemic compounds
PCT/GB1993/000328 WO1993016055A1 (en) 1992-02-17 1993-02-16 Hypolipidaemic benzothiazepine compounds

Publications (3)

Publication Number Publication Date
FI943775A7 FI943775A7 (fi) 1994-08-16
FI943775L FI943775L (fi) 1994-08-16
FI943775A0 true FI943775A0 (fi) 1994-08-16

Family

ID=10710542

Family Applications (1)

Application Number Title Priority Date Filing Date
FI943775A FI943775A0 (fi) 1992-02-17 1993-02-16 Hypolipideemiset bentsotiatsepiiniyhdisteet

Country Status (21)

Country Link
US (2) US5663165A (OSRAM)
EP (1) EP0626952B1 (OSRAM)
JP (1) JP2904926B2 (OSRAM)
KR (1) KR100265529B1 (OSRAM)
AT (1) ATE178897T1 (OSRAM)
AU (1) AU675419B2 (OSRAM)
CA (1) CA2117485A1 (OSRAM)
DE (1) DE69324479T2 (OSRAM)
DK (1) DK0626952T3 (OSRAM)
ES (1) ES2131106T3 (OSRAM)
FI (1) FI943775A0 (OSRAM)
GB (1) GB9203347D0 (OSRAM)
GR (1) GR3030491T3 (OSRAM)
HU (1) HUT71487A (OSRAM)
IL (1) IL104740A (OSRAM)
MX (1) MX9300821A (OSRAM)
MY (1) MY129970A (OSRAM)
NZ (1) NZ249189A (OSRAM)
TW (1) TW274547B (OSRAM)
WO (1) WO1993016055A1 (OSRAM)
ZA (1) ZA931073B (OSRAM)

Families Citing this family (126)

* Cited by examiner, † Cited by third party
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TW202313579A (zh) 2021-06-03 2023-04-01 瑞典商艾爾比瑞歐公司 苯并噻(二)氮呯(benzothia(di)azepine)化合物及其作為膽酸調節劑之用途
JP2025516153A (ja) 2022-04-22 2025-05-27 アルビレオ・アクチボラグ Asbt阻害剤の皮下投与
JP2025524362A (ja) 2022-06-09 2025-07-30 アルビレオ・アクチボラグ 肝炎の処置
KR20250029896A (ko) 2022-07-05 2025-03-05 알비레오 에이비 벤조티아(디)아제핀 화합물 및 담즙산 조절제로서의 이의 용도
EP4629997A1 (en) 2022-12-09 2025-10-15 Albireo AB Asbt inhibitors in the treatment of renal diseases
WO2025146507A1 (en) 2024-01-05 2025-07-10 Albireo Ab Benzothia(di)azepine compounds and their use as bile acid modulators
WO2025146508A1 (en) 2024-01-05 2025-07-10 Albireo Ab Benzothia(di)azepine compounds and their use as bile acid modulators

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US3362962A (en) * 1964-01-24 1968-01-09 Hoffmann La Roche Certain benzothiazepine derivatives
US5276025A (en) * 1992-09-09 1994-01-04 Merck & Co., Inc. Heterobicyclic sulfonamides

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US5859240A (en) 1999-01-12
DK0626952T3 (da) 1999-10-25
JP2904926B2 (ja) 1999-06-14
KR100265529B1 (ko) 2000-11-01
HK1004217A1 (en) 1998-11-20
FI943775A7 (fi) 1994-08-16
ZA931073B (en) 1994-08-16
AU3508293A (en) 1993-09-03
ATE178897T1 (de) 1999-04-15
GR3030491T3 (en) 1999-10-29
WO1993016055A1 (en) 1993-08-19
KR950700265A (ko) 1995-01-16
TW274547B (OSRAM) 1996-04-21
DE69324479T2 (de) 1999-09-16
FI943775L (fi) 1994-08-16
AU675419B2 (en) 1997-02-06
MX9300821A (es) 1993-09-01
HU9402365D0 (en) 1994-10-28
GB9203347D0 (en) 1992-04-01
DE69324479D1 (de) 1999-05-20
JPH07503724A (ja) 1995-04-20
IL104740A0 (en) 1993-06-10
CA2117485A1 (en) 1993-08-19
US5663165A (en) 1997-09-02
NZ249189A (en) 1996-02-27
HUT71487A (en) 1995-11-28
ES2131106T3 (es) 1999-07-16
MY129970A (en) 2007-05-31
EP0626952B1 (en) 1999-04-14
IL104740A (en) 1996-09-12
EP0626952A1 (en) 1994-12-07

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