FI880632A - Fusionerade azepinon- och azocinonderivat, foerfarande foer deras framstaellning, dessa innehaollande medel och deras anvaendning samt vid deras framstaellning anvaendbara mellanprodukter. - Google Patents

Fusionerade azepinon- och azocinonderivat, foerfarande foer deras framstaellning, dessa innehaollande medel och deras anvaendning samt vid deras framstaellning anvaendbara mellanprodukter. Download PDF

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Publication number
FI880632A
FI880632A FI880632A FI880632A FI880632A FI 880632 A FI880632 A FI 880632A FI 880632 A FI880632 A FI 880632A FI 880632 A FI880632 A FI 880632A FI 880632 A FI880632 A FI 880632A
Authority
FI
Finland
Prior art keywords
deras
och
framstaellning
fusionerade
azocinonderivat
Prior art date
Application number
FI880632A
Other languages
English (en)
Other versions
FI880632A0 (fi
FI86849C (fi
FI86849B (fi
Inventor
Hansjoerg Urbach
Rainer Henning
Bernward Schoelkens
Reinhard Becker
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of FI880632A0 publication Critical patent/FI880632A0/fi
Publication of FI880632A publication Critical patent/FI880632A/fi
Application granted granted Critical
Publication of FI86849B publication Critical patent/FI86849B/fi
Publication of FI86849C publication Critical patent/FI86849C/fi

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Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/02Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link
    • C07K5/022Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2
    • C07K5/0222Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing at least one abnormal peptide link containing the structure -X-C(=O)-(C)n-N-C-C(=O)-Y-; X and Y being heteroatoms; n being 1 or 2 with the first amino acid being heterocyclic, e.g. Pro, Trp
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P27/00Drugs for disorders of the senses
    • A61P27/02Ophthalmic agents
    • A61P27/06Antiglaucoma agents or miotics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/12Antihypertensives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Ophthalmology & Optometry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Cardiology (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
FI880632A 1987-02-14 1988-02-11 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara azepinonderivat och vid foerfarandet anvaendbara mellanprodukter FI86849C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3704661 1987-02-14
DE19873704661 DE3704661A1 (de) 1987-02-14 1987-02-14 Annelierte azepinon- und azocinon-derivate, verfahren zu ihrer herstellung, diese enthaltende mittel und ihre verwendung, sowie zwischenprodukte bei ihrer herstellung

Publications (4)

Publication Number Publication Date
FI880632A0 FI880632A0 (fi) 1988-02-11
FI880632A true FI880632A (fi) 1988-08-15
FI86849B FI86849B (fi) 1992-07-15
FI86849C FI86849C (fi) 1992-10-26

Family

ID=6320980

Family Applications (1)

Application Number Title Priority Date Filing Date
FI880632A FI86849C (fi) 1987-02-14 1988-02-11 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara azepinonderivat och vid foerfarandet anvaendbara mellanprodukter

Country Status (26)

Country Link
US (1) US4857520A (fi)
EP (1) EP0279350B1 (fi)
JP (1) JP2638034B2 (fi)
KR (1) KR960011376B1 (fi)
AR (1) AR246957A1 (fi)
AT (1) ATE97913T1 (fi)
AU (1) AU610124B2 (fi)
CA (1) CA1313371C (fi)
CZ (1) CZ280148B6 (fi)
DD (1) DD279877A5 (fi)
DE (2) DE3704661A1 (fi)
DK (1) DK172553B1 (fi)
ES (1) ES2061531T3 (fi)
FI (1) FI86849C (fi)
HU (2) HU208425B (fi)
IE (1) IE62354B1 (fi)
IL (1) IL85406A (fi)
JO (1) JO1524B1 (fi)
MA (1) MA21181A1 (fi)
MX (1) MX174166B (fi)
NO (1) NO176763C (fi)
NZ (1) NZ223500A (fi)
PH (1) PH25186A (fi)
PT (1) PT86748B (fi)
TN (1) TNSN88010A1 (fi)
ZA (1) ZA88991B (fi)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW483763B (en) * 1994-09-02 2002-04-21 Astra Ab Pharmaceutical composition comprising of ramipril and dihydropyridine compound
US5587375A (en) * 1995-02-17 1996-12-24 Bristol-Myers Squibb Company Azepinone compounds useful in the inhibition of ACE and NEP
SE9903028D0 (sv) 1999-08-27 1999-08-27 Astra Ab New use
TR200200515T2 (tr) * 1999-08-30 2002-11-21 Aventis Pharma Deutschland Gmbh Renin-anjiyotensin sistem önleyicilerinin kardiyovasküler vakaların engellenmesinde kullanılması.

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3354146A (en) * 1967-11-21 Process for the production of cyclo- pentano omega-oenantholactam
US4141893A (en) * 1976-11-02 1979-02-27 Eli Lilly And Company Decahydrocyclopent[c]azepines
CY1403A (en) * 1981-08-11 1987-12-18 Ciba Geigy Ag Benzazepin-2-ones
DE3373469D1 (en) * 1982-09-30 1987-10-15 Merck & Co Inc 1-n-alkylcarboxy-benzofused lactams useful as antihypertensive agents
US4470988A (en) * 1983-02-10 1984-09-11 Ciba-Geigy Corporation Benzazocinone and benzazoninone derivatives, and their pharmaceutical use
DE3426720A1 (de) * 1984-07-20 1986-01-23 Hoechst Ag, 6230 Frankfurt Benzthiazepinon- und benzthiazocinon-derivate, verfahren zu ihrer herstellung, diese enthaltende mittel und ihre verwendung, sowie zwischenprodukte bei ihrer herstellung

Also Published As

Publication number Publication date
JP2638034B2 (ja) 1997-08-06
AR246957A1 (es) 1994-10-31
JO1524B1 (en) 1989-01-25
FI880632A0 (fi) 1988-02-11
NZ223500A (en) 1990-11-27
NO880628L (no) 1988-08-15
EP0279350A3 (en) 1990-09-05
DD279877A5 (de) 1990-06-20
AU1167288A (en) 1988-08-18
DE3885914D1 (de) 1994-01-13
PH25186A (en) 1991-03-27
PT86748B (pt) 1992-04-30
ZA88991B (en) 1988-08-10
NO880628D0 (no) 1988-02-12
MX174166B (es) 1994-04-26
HUT48602A (en) 1989-06-28
NO176763C (no) 1995-05-24
FI86849C (fi) 1992-10-26
CZ89288A3 (en) 1994-12-15
TNSN88010A1 (fr) 1990-07-10
HU203727B (en) 1991-09-30
DK72488A (da) 1988-08-15
ATE97913T1 (de) 1993-12-15
DK172553B1 (da) 1999-01-11
HU208425B (en) 1993-10-28
IL85406A0 (en) 1988-07-31
US4857520A (en) 1989-08-15
EP0279350B1 (de) 1993-12-01
NO176763B (no) 1995-02-13
IL85406A (en) 1992-06-21
JPS63203665A (ja) 1988-08-23
MX10408A (es) 1993-07-01
CA1313371C (en) 1993-02-02
MA21181A1 (fr) 1988-10-01
CZ280148B6 (cs) 1995-11-15
KR880009939A (ko) 1988-10-06
ES2061531T3 (es) 1994-12-16
EP0279350A2 (de) 1988-08-24
IE880390L (en) 1988-08-14
FI86849B (fi) 1992-07-15
PT86748A (pt) 1988-03-01
DK72488D0 (da) 1988-02-12
IE62354B1 (en) 1995-01-25
AU610124B2 (en) 1991-05-16
KR960011376B1 (ko) 1996-08-22
HUT50785A (en) 1990-03-28
DE3704661A1 (de) 1988-08-25

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Owner name: HOECHST AKTIENGESELLSCHAFT