FI810669L - Nya karbostyrilderivat foerfarande foer deras framstaellning och dessa innehaollande farmaceutiska kompositioner - Google Patents

Nya karbostyrilderivat foerfarande foer deras framstaellning och dessa innehaollande farmaceutiska kompositioner

Info

Publication number
FI810669L
FI810669L FI810669A FI810669A FI810669L FI 810669 L FI810669 L FI 810669L FI 810669 A FI810669 A FI 810669A FI 810669 A FI810669 A FI 810669A FI 810669 L FI810669 L FI 810669L
Authority
FI
Finland
Prior art keywords
carbostyrilderivat
nya
pharmaceutical composition
foerfarande foer
deras framstaellning
Prior art date
Application number
FI810669A
Other languages
English (en)
Other versions
FI76323B (fi
FI76323C (fi
Inventor
Kazuo Banno
Takafumi Fujioka
Masaaki Osaki
Kazuyuki Nakagawa
Original Assignee
Otsuka Pharma Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from JP2880580A external-priority patent/JPS56125370A/ja
Priority claimed from JP11502280A external-priority patent/JPS5738772A/ja
Application filed by Otsuka Pharma Co Ltd filed Critical Otsuka Pharma Co Ltd
Publication of FI810669L publication Critical patent/FI810669L/fi
Publication of FI76323B publication Critical patent/FI76323B/fi
Application granted granted Critical
Publication of FI76323C publication Critical patent/FI76323C/fi

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D215/00Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/20Oxygen atoms
    • C07D215/22Oxygen atoms attached in position 2 or 4
    • C07D215/227Oxygen atoms attached in position 2 or 4 only one oxygen atom which is attached in position 2

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
FI810669A 1980-03-06 1981-03-03 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara karbostyrilderivat. FI76323C (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
JP2880580 1980-03-06
JP2880580A JPS56125370A (en) 1980-03-06 1980-03-06 Carbostyril derivative
JP11502280A JPS5738772A (en) 1980-08-20 1980-08-20 Carbostyril derivative
JP11502280 1980-08-20

Publications (3)

Publication Number Publication Date
FI810669L true FI810669L (fi) 1981-09-07
FI76323B FI76323B (fi) 1988-06-30
FI76323C FI76323C (fi) 1988-10-10

Family

ID=26366952

Family Applications (1)

Application Number Title Priority Date Filing Date
FI810669A FI76323C (fi) 1980-03-06 1981-03-03 Foerfarande foer framstaellning av nya terapeutiskt anvaendbara karbostyrilderivat.

Country Status (21)

Country Link
US (4) US4460593A (fi)
AT (1) AT381307B (fi)
AU (1) AU523005B2 (fi)
BE (1) BE887800A (fi)
CA (1) CA1155119A (fi)
CH (1) CH647775A5 (fi)
DE (2) DE3152880C2 (fi)
DK (1) DK155282C (fi)
ES (4) ES8301962A1 (fi)
FI (1) FI76323C (fi)
FR (1) FR2477542A1 (fi)
GB (1) GB2071094B (fi)
IT (1) IT1144315B (fi)
MX (1) MX6980E (fi)
NL (1) NL184364C (fi)
NO (1) NO159531C (fi)
PH (1) PH17194A (fi)
PT (1) PT72622B (fi)
RU (1) RU1779249C (fi)
SE (1) SE447255B (fi)
SU (1) SU1367857A3 (fi)

Families Citing this family (57)

* Cited by examiner, † Cited by third party
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PH17194A (en) * 1980-03-06 1984-06-19 Otsuka Pharma Co Ltd Novel carbostyril derivatives,and pharmaceutical composition containing the same
FI77852C (fi) * 1981-02-17 1989-05-10 Otsuka Pharma Co Ltd Foerfarande foer framstaellning av nya, saosom hjaertmediciner anvaendbara substituerade amid- och (maettad heterocykel)karbonylkarbostyrilderivat.
AU532361B2 (en) * 1981-09-01 1983-09-29 Otsuka Pharmaceutical Co., Ltd. Carbostyril derivatives
US4578381A (en) * 1982-07-05 1986-03-25 Otsuka Pharmaceutical Co., Ltd. Carbostyril derivatives
CH655110A5 (de) * 1982-09-03 1986-03-27 Otsuka Pharma Co Ltd Carbostyrilderivate, verfahren zu deren herstellung und arzneimittel, welche diese enthalten.
DE3434271A1 (de) * 1984-09-19 1986-03-20 Beiersdorf Ag, 2000 Hamburg Substituierte 3,4-dihydro-chinolin-2(1h)-one verfahren zu ihrer herstellung und ihre verwendung sowie diese verbindungen enthaltende zubereitungen
DE3509131A1 (de) * 1985-03-14 1986-09-18 Fa. Carl Zeiss, 7920 Heidenheim Verfahren zur justierten montage der optischen bauteile eines optischen geraetes
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US5166367A (en) * 1991-06-21 1992-11-24 American Home Products Corporation Antipsychotic benzodioxan derivatives
US5189171A (en) * 1991-06-21 1993-02-23 American Home Products Corporation Antipsychotic benzodioxan derivatives
HUT70528A (en) * 1991-07-17 1995-10-30 Pfizer 2-(4-hydroxypiperidino)-1-alkanol derivatives as antiischemic agents and process for production thereof
US6255322B1 (en) 1992-06-19 2001-07-03 Pfizer Inc. 2-(4-hydroxypiperidino)-1-alkanol derivatives as antiischemic agents
DE69430861T2 (de) * 1993-04-07 2003-01-23 Otsuka Pharmaceutical Co., Ltd. N-acylierte 4-aminopiperidin derivate als aktive bestandteile von peripher gefässerweiternden wikstoffen
EP0709384B1 (de) * 1994-10-31 1998-12-23 MERCK PATENT GmbH Benzylpiperidinderivate mit hoher Affinität zu Bindungsstellen von Aminosäure-Rezeptoren
ZA9610745B (en) * 1995-12-22 1997-06-24 Warner Lambert Co 4-Subsituted piperidine analogs and their use as subtype selective nmda receptor antagonists
ZA9610736B (en) * 1995-12-22 1997-06-27 Warner Lambert Co 2-Substituted piperidine analogs and their use as subtypeselective nmda receptor antagonists
ZA9610738B (en) 1995-12-22 1997-06-24 Warner Lambert Co Subtype selective nmda receptor ligands and the use thereof
ZA9610741B (en) * 1995-12-22 1997-06-24 Warner Lambert Co 4-Substituted piperidine analogs and their use as subtype selective nmda receptor antagonists
DE19812331A1 (de) * 1998-03-20 1999-09-23 Merck Patent Gmbh Piperidinderivate
FR2823749B1 (fr) * 2001-04-20 2004-02-20 Sanofi Synthelabo Phenyl- et pyridyl-piperidines, procede pour leur preparation et compositions pharmaceutiques les contenant
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US7446109B2 (en) 2002-03-13 2008-11-04 Janssen Pharmaceutica N.V. Carbonylamino-derivatives as novel inhibitors of histone deacetylase
KR20040090979A (ko) 2002-03-13 2004-10-27 얀센 파마슈티카 엔.브이. 히스톤 데아세틸레이즈의 신규한 억제제
JP4725945B2 (ja) 2002-03-13 2011-07-13 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ ヒストンデアセチラーゼの新規な阻害剤としてのスルホニルアミノ誘導体
US7592450B2 (en) * 2002-03-13 2009-09-22 Janssen Pharmaceutica N.V. Piperazinyl-, piperidinyl- and morpholinyl-derivatives as inhibitors of histone deacetylase
MY142362A (en) * 2004-01-29 2010-11-30 Otsuka Pharma Co Ltd Pharmaceutical composition for promoting angiogenesis
SI1776358T1 (sl) * 2004-07-28 2009-10-31 Janssen Pharmaceutica Nv Substituirani propenil piperazinski derivati kot novi inhibitorji histon-deacetilaze
ME01058B (me) * 2004-07-28 2012-10-20 Janssen Pharmaceutica Nv Supstituisani derivati propenil piperazina kao novi inhibitori histonske deacetilaze
EP1781639B1 (en) 2004-07-28 2012-01-25 Janssen Pharmaceutica NV Substituted indolyl alkyl amino derivatives as novel inhibitors of histone deacetylase
TWI320783B (en) 2005-04-14 2010-02-21 Otsuka Pharma Co Ltd Heterocyclic compound
CA2605272C (en) 2005-05-18 2013-12-10 Janssen Pharmaceutica N.V. Substituted aminopropenyl piperidine or morpholine derivatives as novel inhibitors of histone deacetylase
US7834025B2 (en) * 2006-01-19 2010-11-16 Janssen Pharmaceutica N.V. Substituted indolyl-alkyl-amino-derivatives as inhibitors of histone deacetylase
CN101370789B (zh) * 2006-01-19 2012-05-30 詹森药业有限公司 作为组蛋白脱乙酰酶抑制剂的吡啶和嘧啶衍生物
JP5247470B2 (ja) * 2006-01-19 2013-07-24 ジヤンセン・フアーマシユーチカ・ナームローゼ・フエンノートシヤツプ ヒストンデアセチラーゼのインヒビターとしてのピリジン及びピリミジン誘導体
WO2007082878A1 (en) * 2006-01-19 2007-07-26 Janssen Pharmaceutica N.V. Aminophenyl derivatives as novel inhibitors of histone deacetylase
EP2520567A3 (en) * 2006-02-23 2012-12-12 Shionogi & Co., Ltd. Nitrogen-containing heterocycle derivatives substituted with cyclic group
WO2009034029A2 (de) * 2007-09-07 2009-03-19 Boehringer Ingelheim International Gmbh 1-substituierte 4 -heterocyclylpiperidine als cgrp antagonisten
EP2400968B1 (en) 2009-02-26 2016-09-28 Reviva Pharmaceuticals, Inc. Compositions, synthesis, and methods of utilizing arylpiperazine derivatives
EP2847193B1 (en) * 2012-05-09 2019-08-07 Sunovion Pharmaceuticals Inc. Heteroaryl compounds and methods of use thereof
CN106608875A (zh) 2015-10-26 2017-05-03 江苏恩华药业股份有限公司 一种稠和杂环类衍生物合成及其应用
CN108031471A (zh) * 2017-10-27 2018-05-15 苏州盖德精细材料有限公司 一种静电纺丝制备的负载型纳米纤维催化剂及其在3,5-二羟基甲苯制备中的应用
CN108250058B (zh) * 2018-01-19 2022-02-11 上海怡立舍生物技术有限公司 Ppar激动剂及其在治疗老年痴呆及其他疾病中的用途
CN116554127B (zh) * 2022-01-28 2025-03-21 成都麻沸散医药科技有限公司 哌嗪取代苯酚类衍生物及其用途

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US3629266A (en) * 1969-03-03 1971-12-21 Miles Lab (phenyl piperidino alkyl)3 4-dihydrocarbostyrils
US3910924A (en) * 1972-04-13 1975-10-07 Otsuka Pharma Co Ltd 3,4-Dihydrocarbostyril derivatives and a process for preparing the same
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FI77852C (fi) * 1981-02-17 1989-05-10 Otsuka Pharma Co Ltd Foerfarande foer framstaellning av nya, saosom hjaertmediciner anvaendbara substituerade amid- och (maettad heterocykel)karbonylkarbostyrilderivat.
AU532361B2 (en) * 1981-09-01 1983-09-29 Otsuka Pharmaceutical Co., Ltd. Carbostyril derivatives

Also Published As

Publication number Publication date
ES500137A0 (es) 1982-11-01
ES509659A0 (es) 1983-05-01
ES518667A0 (es) 1984-06-16
SU1367857A3 (ru) 1988-01-15
GB2071094B (en) 1984-09-26
US4455422A (en) 1984-06-19
IT8167311A0 (it) 1981-03-05
MX6980E (es) 1987-01-19
DE3107601A1 (de) 1982-02-04
US4567187A (en) 1986-01-28
CH647775A5 (de) 1985-02-15
NL184364B (nl) 1989-02-01
FI76323B (fi) 1988-06-30
ES8405782A1 (es) 1984-06-16
NO810765L (no) 1981-09-07
DK155282C (da) 1989-08-07
CA1155119A (en) 1983-10-11
US4460593A (en) 1984-07-17
DK155282B (da) 1989-03-20
DK99781A (da) 1981-09-07
ES8305356A1 (es) 1983-04-01
IT1144315B (it) 1986-10-29
GB2071094A (en) 1981-09-16
DE3107601C2 (fi) 1989-07-20
AT381307B (de) 1986-09-25
FR2477542A1 (fr) 1981-09-11
FI76323C (fi) 1988-10-10
ATA98481A (de) 1986-02-15
ES509658A0 (es) 1983-04-01
NO159531C (no) 1989-01-11
NL184364C (nl) 1989-07-03
AU523005B2 (en) 1982-07-08
NL8101099A (nl) 1981-10-01
FR2477542B1 (fi) 1983-09-09
ES8301962A1 (es) 1982-11-01
AU6797381A (en) 1981-09-10
PT72622B (en) 1982-06-15
DE3152880C2 (fi) 1990-03-22
ES8306141A1 (es) 1983-05-01
RU1779249C (ru) 1992-11-30
NO159531B (no) 1988-10-03
PT72622A (en) 1981-04-01
BE887800A (fr) 1981-09-07
SE447255B (sv) 1986-11-03
US4619932A (en) 1986-10-28
PH17194A (en) 1984-06-19
SE8101409L (sv) 1981-09-07

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Legal Events

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MM Patent lapsed

Owner name: OTSUKA PHARMACEUTICAL CO., LTD.