FI65426C - Analogifoerfarande foer framstaellning av nya farmakologiskt verkande n-(2-morfolinoetyl)bensamider - Google Patents

Analogifoerfarande foer framstaellning av nya farmakologiskt verkande n-(2-morfolinoetyl)bensamider Download PDF

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Publication number
FI65426C
FI65426C FI770356A FI770356A FI65426C FI 65426 C FI65426 C FI 65426C FI 770356 A FI770356 A FI 770356A FI 770356 A FI770356 A FI 770356A FI 65426 C FI65426 C FI 65426C
Authority
FI
Finland
Prior art keywords
morpholinoethyl
formula
benzamide
compound
compounds
Prior art date
Application number
FI770356A
Other languages
English (en)
Finnish (fi)
Other versions
FI770356A (de
FI65426B (fi
Inventor
Willy Burkard
Pierre-Charles Wyss
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of FI770356A publication Critical patent/FI770356A/fi
Application granted granted Critical
Publication of FI65426B publication Critical patent/FI65426B/fi
Publication of FI65426C publication Critical patent/FI65426C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/24—Antidepressants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/26—Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychiatry (AREA)
  • Medicinal Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
FI770356A 1976-02-16 1977-02-01 Analogifoerfarande foer framstaellning av nya farmakologiskt verkande n-(2-morfolinoetyl)bensamider FI65426C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
AT107076A AT345842B (de) 1976-02-16 1976-02-16 Verfahren zur herstellung von neuen morpholinderivaten, ihren n-oxyden und salzen
AT107076 1976-02-16

Publications (3)

Publication Number Publication Date
FI770356A FI770356A (de) 1977-08-17
FI65426B FI65426B (fi) 1984-01-31
FI65426C true FI65426C (fi) 1984-05-10

Family

ID=3505951

Family Applications (1)

Application Number Title Priority Date Filing Date
FI770356A FI65426C (fi) 1976-02-16 1977-02-01 Analogifoerfarande foer framstaellning av nya farmakologiskt verkande n-(2-morfolinoetyl)bensamider

Country Status (28)

Country Link
JP (1) JPS52100476A (de)
AR (2) AR214307A1 (de)
AT (5) AT345842B (de)
AU (1) AU506427B2 (de)
BE (1) BE851422A (de)
CA (1) CA1076112A (de)
CH (5) CH623317A5 (de)
DE (1) DE2706179C2 (de)
DK (1) DK148824C (de)
ES (4) ES455907A1 (de)
FI (1) FI65426C (de)
FR (1) FR2340940A1 (de)
GB (1) GB1512194A (de)
GR (1) GR62413B (de)
HR (1) HRP930495B1 (de)
IE (1) IE44482B1 (de)
IL (1) IL51406A (de)
LU (2) LU76771A1 (de)
MC (1) MC1136A1 (de)
NL (2) NL179382C (de)
NO (2) NO148417C (de)
NZ (1) NZ183316A (de)
PH (1) PH12847A (de)
PT (1) PT66195B (de)
SE (1) SE426822B (de)
SI (1) SI7710060A8 (de)
YU (1) YU39983B (de)
ZA (1) ZA77746B (de)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4829506B2 (ja) * 2004-02-17 2011-12-07 石原産業株式会社 チオアミド系化合物又はその塩、並びにそれらを含有するサイトカイン産生抑制剤
US7960391B2 (en) 2005-05-03 2011-06-14 Bayer Cropscience Ag Heterocyclylethylbenzamide derivatives
RU2570898C2 (ru) * 2014-03-27 2015-12-20 Федеральное государственное бюджетное образовательное учреждение высшего профессионального образования "Российский химико-технологический университет имени Д.И. Менделеева (РХТУ им. Д.И. Менделеева)" Способ получения n-[2-(морфолин-4-ил)этил]-4-хлорбензамида (варианты)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH451142A (de) * 1965-01-19 1968-05-15 Sandoz Ag Verfahren zur Herstellung neuer basisch substituierter Benzoesäureamide
FR1501846A (fr) * 1966-09-26 1967-11-18 Bellon Labor Sa Roger Procédé amélioré pour la préparation des thioamides
US3787419A (en) * 1971-07-01 1974-01-22 American Home Prod N-substituted-alpha,alpha,alpha-trifluoro-m-toluamides

Also Published As

Publication number Publication date
BE851422A (fr) 1977-08-16
JPS6215547B2 (de) 1987-04-08
AR212554A1 (es) 1978-07-31
PT66195A (fr) 1977-03-01
AT345842B (de) 1978-10-10
CH623577A5 (en) 1981-06-15
CA1076112A (en) 1980-04-22
ATA25778A (de) 1978-09-15
NO148417C (no) 1983-10-12
NO770488L (no) 1977-08-17
GR62413B (en) 1979-04-11
NO148417B (no) 1983-06-27
ES455907A1 (es) 1978-05-01
FR2340940B1 (de) 1981-01-09
ATA107076A (de) 1978-02-15
DK148824C (da) 1986-04-21
NO1994008I1 (no) 1994-08-03
FI770356A (de) 1977-08-17
ZA77746B (en) 1977-12-28
CH622787A5 (en) 1981-04-30
NL930082I1 (nl) 1993-09-16
MC1136A1 (fr) 1977-11-18
HRP930495B1 (en) 1996-10-31
ES467449A1 (es) 1978-10-16
CH622786A5 (en) 1981-04-30
YU6077A (en) 1983-01-21
IE44482L (en) 1977-08-16
YU39983B (en) 1985-06-30
IE44482B1 (en) 1981-12-16
FR2340940A1 (fr) 1977-09-09
ES467455A1 (es) 1978-10-16
PH12847A (en) 1979-09-12
SE426822B (sv) 1983-02-14
NL179382C (nl) 1986-09-01
LU76771A1 (de) 1978-04-13
CH623576A5 (en) 1981-06-15
GB1512194A (en) 1978-05-24
DE2706179C2 (de) 1984-02-02
IL51406A0 (en) 1977-04-29
LU88300I2 (de) 1994-09-09
NL179382B (nl) 1986-04-01
DK148824B (da) 1985-10-14
NL930082I2 (nl) 1994-08-16
ES467448A1 (es) 1978-10-16
NZ183316A (en) 1979-04-26
ATA25678A (de) 1978-09-15
DK51677A (da) 1977-08-17
NL7701144A (nl) 1977-08-18
AU2109977A (en) 1978-07-13
AU506427B2 (en) 1980-01-03
FI65426B (fi) 1984-01-31
IL51406A (en) 1979-12-30
AT349479B (de) 1979-04-10
AT349481B (de) 1979-04-10
JPS52100476A (en) 1977-08-23
AT349482B (de) 1979-04-10
PT66195B (fr) 1979-01-17
SE7701669L (sv) 1977-08-17
ATA25878A (de) 1978-09-15
ATA25578A (de) 1978-09-15
CH623317A5 (en) 1981-05-29
DE2706179A1 (de) 1977-08-18
AR214307A1 (es) 1979-05-31
AT349480B (de) 1979-04-10
SI7710060A8 (en) 1996-12-31

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Legal Events

Date Code Title Description
MA Patent expired
ND Supplementary protection certificate (spc) granted
SPCG Supplementary protection certificate granted

Spc suppl protection certif: L16

Extension date: 20020201

MA Patent expired

Owner name: F. HOFFMANN-LA ROCHE AG