AT349482B - Verfahren zur herstellung von neuen morpholinderivaten, ihren n-oxiden und salzen - Google Patents

Verfahren zur herstellung von neuen morpholinderivaten, ihren n-oxiden und salzen

Info

Publication number
AT349482B
AT349482B AT25878A AT25878A AT349482B AT 349482 B AT349482 B AT 349482B AT 25878 A AT25878 A AT 25878A AT 25878 A AT25878 A AT 25878A AT 349482 B AT349482 B AT 349482B
Authority
AT
Austria
Prior art keywords
oxides
salts
producing new
morpholine derivatives
new morpholine
Prior art date
Application number
AT25878A
Other languages
English (en)
Other versions
ATA25878A (de
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Priority to AT25878A priority Critical patent/AT349482B/de
Publication of ATA25878A publication Critical patent/ATA25878A/de
Application granted granted Critical
Publication of AT349482B publication Critical patent/AT349482B/de

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D295/00Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/125Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/13Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/24Antidepressants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/26Psychostimulants, e.g. nicotine, cocaine

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • Psychiatry (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biomedical Technology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pain & Pain Management (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
AT25878A 1976-02-16 1978-01-13 Verfahren zur herstellung von neuen morpholinderivaten, ihren n-oxiden und salzen AT349482B (de)

Priority Applications (1)

Application Number Priority Date Filing Date Title
AT25878A AT349482B (de) 1976-02-16 1978-01-13 Verfahren zur herstellung von neuen morpholinderivaten, ihren n-oxiden und salzen

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
AT107076A AT345842B (de) 1976-02-16 1976-02-16 Verfahren zur herstellung von neuen morpholinderivaten, ihren n-oxyden und salzen
AT25878A AT349482B (de) 1976-02-16 1978-01-13 Verfahren zur herstellung von neuen morpholinderivaten, ihren n-oxiden und salzen

Publications (2)

Publication Number Publication Date
ATA25878A ATA25878A (de) 1978-09-15
AT349482B true AT349482B (de) 1979-04-10

Family

ID=3505951

Family Applications (5)

Application Number Title Priority Date Filing Date
AT107076A AT345842B (de) 1976-02-16 1976-02-16 Verfahren zur herstellung von neuen morpholinderivaten, ihren n-oxyden und salzen
AT25578A AT349479B (de) 1976-02-16 1978-01-13 Verfahren zur herstellung von neuen morpholin- derivaten, ihren n-oxiden und salzen
AT25778A AT349481B (de) 1976-02-16 1978-01-13 Verfahren zur herstellung von neuen morpholinderivaten, ihren n-oxiden und salzen
AT25878A AT349482B (de) 1976-02-16 1978-01-13 Verfahren zur herstellung von neuen morpholinderivaten, ihren n-oxiden und salzen
AT25678A AT349480B (de) 1976-02-16 1978-01-13 Verfahren zur herstellung von neuen morpholin- derivaten, ihren n-oxiden und salzen

Family Applications Before (3)

Application Number Title Priority Date Filing Date
AT107076A AT345842B (de) 1976-02-16 1976-02-16 Verfahren zur herstellung von neuen morpholinderivaten, ihren n-oxyden und salzen
AT25578A AT349479B (de) 1976-02-16 1978-01-13 Verfahren zur herstellung von neuen morpholin- derivaten, ihren n-oxiden und salzen
AT25778A AT349481B (de) 1976-02-16 1978-01-13 Verfahren zur herstellung von neuen morpholinderivaten, ihren n-oxiden und salzen

Family Applications After (1)

Application Number Title Priority Date Filing Date
AT25678A AT349480B (de) 1976-02-16 1978-01-13 Verfahren zur herstellung von neuen morpholin- derivaten, ihren n-oxiden und salzen

Country Status (28)

Country Link
JP (1) JPS52100476A (de)
AR (2) AR214307A1 (de)
AT (5) AT345842B (de)
AU (1) AU506427B2 (de)
BE (1) BE851422A (de)
CA (1) CA1076112A (de)
CH (5) CH623317A5 (de)
DE (1) DE2706179C2 (de)
DK (1) DK148824C (de)
ES (4) ES455907A1 (de)
FI (1) FI65426C (de)
FR (1) FR2340940A1 (de)
GB (1) GB1512194A (de)
GR (1) GR62413B (de)
HR (1) HRP930495B1 (de)
IE (1) IE44482B1 (de)
IL (1) IL51406A (de)
LU (2) LU76771A1 (de)
MC (1) MC1136A1 (de)
NL (2) NL179382C (de)
NO (2) NO148417C (de)
NZ (1) NZ183316A (de)
PH (1) PH12847A (de)
PT (1) PT66195B (de)
SE (1) SE426822B (de)
SI (1) SI7710060A8 (de)
YU (1) YU39983B (de)
ZA (1) ZA77746B (de)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP2005263787A (ja) * 2004-02-17 2005-09-29 Ishihara Sangyo Kaisha Ltd アミド系化合物又はその塩、並びにそれらを含有するサイトカイン産生抑制剤
ATE414694T1 (de) * 2005-05-03 2008-12-15 Bayer Cropscience Sa Neue heterocyclylethylbenzamid-derivate
RU2414462C1 (ru) * 2009-11-16 2011-03-20 Федеральное государственное унитарное предприятие "Государственный научный центр "Научно-исследовательский институт органических полупродуктов и красителей" (ФГУП "ГНЦ "НИОПИК") Способ получения 4-хлор-n-(2-морфолиноэтил)бензамида
RU2570898C2 (ru) * 2014-03-27 2015-12-20 Федеральное государственное бюджетное образовательное учреждение высшего профессионального образования "Российский химико-технологический университет имени Д.И. Менделеева (РХТУ им. Д.И. Менделеева)" Способ получения n-[2-(морфолин-4-ил)этил]-4-хлорбензамида (варианты)

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH451142A (de) * 1965-01-19 1968-05-15 Sandoz Ag Verfahren zur Herstellung neuer basisch substituierter Benzoesäureamide
FR1501846A (fr) * 1966-09-26 1967-11-18 Bellon Labor Sa Roger Procédé amélioré pour la préparation des thioamides
US3787419A (en) * 1971-07-01 1974-01-22 American Home Prod N-substituted-alpha,alpha,alpha-trifluoro-m-toluamides

Also Published As

Publication number Publication date
JPS6215547B2 (de) 1987-04-08
DK148824C (da) 1986-04-21
NO1994008I1 (no) 1994-08-03
AR212554A1 (es) 1978-07-31
CH623576A5 (en) 1981-06-15
PH12847A (en) 1979-09-12
NL930082I1 (nl) 1993-09-16
NL179382B (nl) 1986-04-01
CH622787A5 (en) 1981-04-30
ES455907A1 (es) 1978-05-01
CH623317A5 (en) 1981-05-29
ATA25778A (de) 1978-09-15
FR2340940B1 (de) 1981-01-09
SE426822B (sv) 1983-02-14
IL51406A (en) 1979-12-30
FI65426B (fi) 1984-01-31
DE2706179A1 (de) 1977-08-18
NO148417B (no) 1983-06-27
AT349481B (de) 1979-04-10
DK51677A (da) 1977-08-17
AT349479B (de) 1979-04-10
FI65426C (fi) 1984-05-10
ES467449A1 (es) 1978-10-16
YU39983B (en) 1985-06-30
GB1512194A (en) 1978-05-24
DK148824B (da) 1985-10-14
GR62413B (en) 1979-04-11
CH623577A5 (en) 1981-06-15
FI770356A7 (de) 1977-08-17
AU2109977A (en) 1978-07-13
PT66195A (fr) 1977-03-01
JPS52100476A (en) 1977-08-23
CH622786A5 (en) 1981-04-30
AU506427B2 (en) 1980-01-03
SI7710060A8 (en) 1996-12-31
BE851422A (fr) 1977-08-16
NL7701144A (nl) 1977-08-18
CA1076112A (en) 1980-04-22
AT349480B (de) 1979-04-10
YU6077A (en) 1983-01-21
FR2340940A1 (fr) 1977-09-09
ATA25878A (de) 1978-09-15
NZ183316A (en) 1979-04-26
NO148417C (no) 1983-10-12
ES467455A1 (es) 1978-10-16
HRP930495B1 (en) 1996-10-31
ZA77746B (en) 1977-12-28
NO770488L (no) 1977-08-17
PT66195B (fr) 1979-01-17
ES467448A1 (es) 1978-10-16
NL179382C (nl) 1986-09-01
MC1136A1 (fr) 1977-11-18
LU88300I2 (de) 1994-09-09
IE44482L (en) 1977-08-16
AR214307A1 (es) 1979-05-31
LU76771A1 (de) 1978-04-13
ATA25578A (de) 1978-09-15
SE7701669L (sv) 1977-08-17
ATA107076A (de) 1978-02-15
ATA25678A (de) 1978-09-15
IE44482B1 (en) 1981-12-16
AT345842B (de) 1978-10-10
DE2706179C2 (de) 1984-02-02
NL930082I2 (nl) 1994-08-16
IL51406A0 (en) 1977-04-29

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Legal Events

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REN Ceased due to non-payment of the annual fee